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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T0137 Mirtazapine 85650-52-8 98%
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T0031L Ziprasidone hydrochloride 122883-93-6 98%
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T0211 Azelastine 58581-89-8 98%
Azelastine is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
T68150 Talastine 16188-61-7 98%
Talastine is an antihistamine compound that can induce an allergic rash.
T22746 Tesmilifene fumarate 1185241-83-1 98%
Tesmilifene fumarate (DPPE fumarate) is an H1C receptor antagonist。
T21428 Mianserin 24219-97-4 98%
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, an...
T0089 Cetirizine dihydrochloride 83881-52-1 98%
Cetirizine dihydrochloride is an effective second-generation histamine H1 antagonist that is potent in the therapy of allergic rhinitis, confirmed urticaria, and...
T0236 Azatadine dimaleate 3978-86-7 98%
Azatadine dimaleate is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
T31488 Dimethindene 5636-83-9 98%
Dimethindene is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.
T7564 Chlorphenoxamine 77-38-3 98%
Chlorphenoxamine is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
T1393 Sodium butanoate 156-54-7 98%
Sodium Butyrate is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds to the zinc sites ...
T4563 Thonzylamine 91-85-0 98%
Thonzylamine is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of sympt...
T2004 Ciproxifan maleate 184025-19-2 98%
Ciproxifan maleate(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other rec...
T8439 Clobenpropit dihydrobromide 145231-35-2 98%
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
T21419 Diphenhydramine 58-73-1 98%
Diphenhydramine, a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the treatment o...
T9353 OXOMEMAZINE 3689-50-7 98%
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
T68921 Impromidine hydrochloride 65573-02-6 98%
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.
T1336 Benztropine mesylate 132-17-2 98%
Benztropine mesylate is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISEASE. Benztropine also inhibits ...
T3963 VUF10460 1028327-66-3 98%
VUF10460 is a non-imidazole histamine H4 receptor agonist.
T0031L2 Ziprasidone 146939-27-7 98%
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Mirtazapine
T0137
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
Ziprasidone hydrochloride
T0031L
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Azelastine
T0211
Azelastine is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
Talastine
T68150
Talastine is an antihistamine compound that can induce an allergic rash.
Tesmilifene fumarate
T22746
Tesmilifene fumarate (DPPE fumarate) is an H1C receptor antagonist。
Mianserin
T21428
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, an...
Cetirizine dihydrochloride
T0089
Cetirizine dihydrochloride is an effective second-generation histamine H1 antagonist that is potent in the therapy of allergic rhinitis, confirmed urticaria, and...
Azatadine dimaleate
T0236
Azatadine dimaleate is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
Dimethindene
T31488
Dimethindene is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.
Chlorphenoxamine
T7564
Chlorphenoxamine is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
Sodium butanoate
T1393
Sodium Butyrate is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds to the zinc sites ...
Thonzylamine
T4563
Thonzylamine is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of sympt...
Ciproxifan maleate
T2004
Ciproxifan maleate(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other rec...
Clobenpropit dihydrobromide
T8439
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
Diphenhydramine
T21419
Diphenhydramine, a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the treatment o...
OXOMEMAZINE
T9353
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
Impromidine hydrochloride
T68921
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.
Benztropine mesylate
T1336
Benztropine mesylate is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISEASE. Benztropine also inhibits ...
VUF10460
T3963
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Ziprasidone
T0031L2
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
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