Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T23297	(S)-(+)-Dimethindene maleate	136152-65-3	99.43%
T23297	(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M...
T0236	Azatadine dimaleate	3978-86-7	99.4%
T0236	Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.
T21428	Mianserin	24219-97-4	99.39%
T21428	Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, an...
T22746	Tesmilifene fumarate	1185241-83-1	99.38%
T22746	Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
T68150	Talastine	16188-61-7	99.37%
T68150	Talastine is an antihistamine compound that can induce an allergic rash.
T1266	Terfenadine	50679-08-8	99.36%
T1266	Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist...
T0211	Azelastine	58581-89-8	99.35%
T0211	Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
T0031L	Ziprasidone hydrochloride	122883-93-6	99.34%
T0031L	Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
T0137	Mirtazapine	85650-52-8	99.3%
T0137	Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T0205	Brompheniramine maleate	980-71-2	99.3%
T0205	Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
T68146	Sufotidine	80343-63-1	99.28%
T68146	Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.
T9084	Cetirizine Impurity B dihydrochloride	1000690-91-4	99.24%
T9084	Cetirizine Impurity B dihydrochloride (De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride) is an impurity of Cetirizine dihydrochloride. Cetirizine is a s...
T0059	Diphenylpyraline hydrochloride	132-18-3	99.22%
T0059	Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) is used in the treatment of Parkinsonism.It is a first-generation antihistami...
T68100	Mifentidine	83184-43-4	99.20%
T68100	Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.
T0383	Fenspiride hydrochloride	5053-08-7	99.18%
T0383	Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use i...
T22501	2-Pyridylethylamine dihydrochloride	3343-39-3	99.17%
T22501	2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
T0074L	Chlorprothixene hydrochloride	6469-93-8	99.16%
T0074L	Chlorprothixene hydrochloride (Truxal hydrochloride) brings strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrener...
T4087	S 38093 HCl	1222097-72-4	99.16%
T4087	S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
T15005	CP-66948	101189-47-3	99.14%
T15005	CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.
T0865	Ranitidine Hydrochloride	66357-59-3	99.13%
T0865	Ranitidine Hydrochloride (AH19065) is a member of the class of histamine H2-receptor antagonists with antacid activity. Ranitidine is a competitive and reversibl...