T68056 |
Donetidine
|
99248-32-5
|
99.12%
|
|
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
|
T0445 |
Promethazine
|
60-87-7
|
99.11%
|
|
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
|
T10499 |
H3 receptor-MO-1
|
1240914-03-7
|
99.11%
|
|
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
|
T3610 |
Ranitidine
|
66357-35-5
|
99.1%
|
|
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestina...
|
T12489 |
Pimethixene
|
314-03-4
|
99.1%
|
|
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist...
|
T8548 |
Metoprine
|
7761-45-7
|
99.09%
|
|
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
|
T9770 |
Samelisant
|
1394808-82-2
|
99.09%
|
|
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects...
|
T1110 |
Meclizine dihydrochloride
|
1104-22-9
|
99.08%
|
|
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation si...
|
T17072 |
Thiethylperazine dimaleate
|
1179-69-7
|
99.07%
|
|
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 an...
|
T10680 |
Carebastine
|
90729-42-3
|
99.06%
|
|
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
|
TN1008 |
Psoralenoside
|
905954-17-8
|
99.03%
|
|
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
|
T3723 |
Dioxopromethazine hydrochloride
|
15374-15-9
|
99%
|
|
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
|
T5495 |
Decloxizine dihydrochloride
|
13073-96-6
|
99%
|
|
Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.
|
T27244 |
Efletirizine
|
150756-35-7
|
98.98%
|
|
Efletirizine (UCB-28754) is a histamine receptor antagonist with inhibitory effects on the enzyme 5-lipoxygenase (5-LO), and is useful in the topical treatment o...
|
T10000 |
(±)-Tazifylline
|
79712-55-3
|
98.97%
|
|
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptor...
|
T22713 |
Decloxizine
|
3733-63-9
|
98.95%
|
|
Decloxizine is a H1 receptor antagonist
|
T19839 |
Oxatomide
|
60607-34-3
|
98.93%
|
|
Oxatomide (Oxatomida) is a potent and orally active dual H1 histamine receptor and P2X7 receptor antagonist with antihistamine and antiallergic activity.Oxatomid...
|
T0797 |
Cimetidine
|
51481-61-9
|
98.85%
|
|
Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological ...
|
T26526 |
Abt-288
|
948845-91-8
|
98.84%
|
|
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.
|
T1822 |
Clemizole
|
442-52-4
|
98.81%
|
|
Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
|