T0942 |
Quinacrine dihydrochloride
|
69-05-6
|
98%
|
|
Quinacrine Hydrochloride is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and antiparasitic activities.
|
T7176 |
Pitolisant hydrochloride
|
903576-44-3
|
98%
|
|
Pitolisant hydrochloride is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
|
T27462 |
GSK-239512
|
720691-69-0
|
98%
|
|
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
|
T26690 |
AVN-101
|
1061354-48-0
|
98%
|
|
AVN-101 is a potent 5-HT7 receptor antagonist.
|
T7085 |
Mebhydrolin
|
524-81-2
|
98%
|
|
Mebhydrolin is a specific histamine H1 receptor antagonist.
|
T0468 |
Lidocaine
|
137-58-6
|
98%
|
|
Lidocaine is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation of intracellul...
|
T1627 |
Famotidine
|
76824-35-6
|
98%
|
|
Famotidine is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors located on the b...
|
T1266 |
Terfenadine
|
50679-08-8
|
98%
|
|
Terfenadine is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistamin...
|
T1097 |
Loratadine
|
79794-75-5
|
98%
|
|
Loratadine is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical antihistamines...
|
T22354 |
Levocetirizine Dihydrochloride
|
130018-87-0
|
98%
|
|
Levocetirizine Dihydrochloride is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine ...
|
T7893 |
Bepotastine
|
125602-71-3
|
98%
|
|
Bepotastine free base is a histamine 1 (H1) receptor antagonis.
|
T0092 |
Antazoline hydrochloride
|
2508-72-7
|
98%
|
|
Antazoline hydrochloride, a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous histamine.
|
T0113 |
Mebhydrolin napadisylate
|
6153-33-9
|
98%
|
|
Mebhydrolin (napadisylate) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.
|
T0118 |
Mizolastine
|
108612-45-9
|
98%
|
|
Mizolastine (IC50= 47 nM) is a histamine H1-receptor antagonist.It is used in the treatment of allergic reactions such as hay fever (seasonal allergic rhinitis),...
|
T32191 |
Irdabisant
|
1005402-19-6
|
98%
|
|
Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R K...
|
T1170 |
Olopatadine hydrochloride
|
140462-76-6
|
98%
|
|
Olopatadine hydrochloride is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.
|
T2200 |
Hydroxyzine dihydrochloride
|
2192-20-3
|
98%
|
|
Hydroxyzine hydrochloride is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruri...
|
T1110 |
Meclizine dihydrochloride
|
1104-22-9
|
98%
|
|
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
|
T0370 |
Pheniramine maleate
|
132-20-7
|
98%
|
|
Pheniramine Maleate, an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase ...
|
T0147 |
Clemastine fumarate
|
14976-57-9
|
98%
|
|
Clemastine Fumarate is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
|