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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T68056 Donetidine 99248-32-5 99.12%
Donetidine
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
T0445 Promethazine 60-87-7 99.11%
Promethazine
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
T10499 H3 receptor-MO-1 1240914-03-7 99.11%
H3 receptor-MO-1
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
T3610 Ranitidine 66357-35-5 99.1%
Ranitidine
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestina...
T12489 Pimethixene 314-03-4 99.1%
Pimethixene
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist...
T8548 Metoprine 7761-45-7 99.09%
Metoprine
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
T9770 Samelisant 1394808-82-2 99.09%
Samelisant
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects...
T1110 Meclizine dihydrochloride 1104-22-9 99.08%
Meclizine dihydrochloride
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation si...
T17072 Thiethylperazine dimaleate 1179-69-7 99.07%
Thiethylperazine dimaleate
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 an...
T10680 Carebastine 90729-42-3 99.06%
Carebastine
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
TN1008 Psoralenoside 905954-17-8 99.03%
Psoralenoside
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
T3723 Dioxopromethazine hydrochloride 15374-15-9 99%
Dioxopromethazine hydrochloride
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
T5495 Decloxizine dihydrochloride 13073-96-6 99%
Decloxizine dihydrochloride
Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.
T27244 Efletirizine 150756-35-7 98.98%
Efletirizine
Efletirizine (UCB-28754) is a histamine receptor antagonist with inhibitory effects on the enzyme 5-lipoxygenase (5-LO), and is useful in the topical treatment o...
T10000 (±)-Tazifylline 79712-55-3 98.97%
(±)-Tazifylline
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptor...
T22713 Decloxizine 3733-63-9 98.95%
Decloxizine
Decloxizine is a H1 receptor antagonist
T19839 Oxatomide 60607-34-3 98.93%
Oxatomide
Oxatomide (Oxatomida) is a potent and orally active dual H1 histamine receptor and P2X7 receptor antagonist with antihistamine and antiallergic activity.Oxatomid...
T0797 Cimetidine 51481-61-9 98.85%
Cimetidine
Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological ...
T26526 Abt-288 948845-91-8 98.84%
Abt-288
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.
T1822 Clemizole 442-52-4 98.81%
Clemizole
Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
Donetidine
T68056
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
Promethazine
T0445
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
H3 receptor-MO-1
T10499
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
Ranitidine
T3610
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestina...
Pimethixene
T12489
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist...
Metoprine
T8548
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
Samelisant
T9770
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects...
Meclizine dihydrochloride
T1110
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation si...
Thiethylperazine dimaleate
T17072
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 an...
Carebastine
T10680
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Psoralenoside
TN1008
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
Dioxopromethazine hydrochloride
T3723
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
Decloxizine dihydrochloride
T5495
Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.
Efletirizine
T27244
Efletirizine (UCB-28754) is a histamine receptor antagonist with inhibitory effects on the enzyme 5-lipoxygenase (5-LO), and is useful in the topical treatment o...
(±)-Tazifylline
T10000
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptor...
Decloxizine
T22713
Decloxizine is a H1 receptor antagonist
Oxatomide
T19839
Oxatomide (Oxatomida) is a potent and orally active dual H1 histamine receptor and P2X7 receptor antagonist with antihistamine and antiallergic activity.Oxatomid...
Cimetidine
T0797
Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological ...
Abt-288
T26526
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.
Clemizole
T1822
Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
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TargetMol