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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T0942 Quinacrine dihydrochloride 69-05-6 98%
Quinacrine Hydrochloride is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and antiparasitic activities.
T7176 Pitolisant hydrochloride 903576-44-3 98%
Pitolisant hydrochloride is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
T27462 GSK-239512 720691-69-0 98%
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
T26690 AVN-101 1061354-48-0 98%
AVN-101 is a potent 5-HT7 receptor antagonist.
T7085 Mebhydrolin 524-81-2 98%
Mebhydrolin is a specific histamine H1 receptor antagonist.
T0468 Lidocaine 137-58-6 98%
Lidocaine is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation of intracellul...
T1627 Famotidine 76824-35-6 98%
Famotidine is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors located on the b...
T1266 Terfenadine 50679-08-8 98%
Terfenadine is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistamin...
T1097 Loratadine 79794-75-5 98%
Loratadine is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical antihistamines...
T22354 Levocetirizine Dihydrochloride 130018-87-0 98%
Levocetirizine Dihydrochloride is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine ...
T7893 Bepotastine 125602-71-3 98%
Bepotastine free base is a histamine 1 (H1) receptor antagonis.
T0092 Antazoline hydrochloride 2508-72-7 98%
Antazoline hydrochloride, a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous histamine.
T0113 Mebhydrolin napadisylate 6153-33-9 98%
Mebhydrolin (napadisylate) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.
T0118 Mizolastine 108612-45-9 98%
Mizolastine (IC50= 47 nM) is a histamine H1-receptor antagonist.It is used in the treatment of allergic reactions such as hay fever (seasonal allergic rhinitis),...
T32191 Irdabisant 1005402-19-6 98%
Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R K...
T1170 Olopatadine hydrochloride 140462-76-6 98%
Olopatadine hydrochloride is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.
T2200 Hydroxyzine dihydrochloride 2192-20-3 98%
Hydroxyzine hydrochloride is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruri...
T1110 Meclizine dihydrochloride 1104-22-9 98%
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
T0370 Pheniramine maleate 132-20-7 98%
Pheniramine Maleate, an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase ...
T0147 Clemastine fumarate 14976-57-9 98%
Clemastine Fumarate is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
Quinacrine dihydrochloride
T0942
Quinacrine Hydrochloride is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and antiparasitic activities.
Pitolisant hydrochloride
T7176
Pitolisant hydrochloride is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
GSK-239512
T27462
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
AVN-101
T26690
AVN-101 is a potent 5-HT7 receptor antagonist.
Mebhydrolin
T7085
Mebhydrolin is a specific histamine H1 receptor antagonist.
Lidocaine
T0468
Lidocaine is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation of intracellul...
Famotidine
T1627
Famotidine is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors located on the b...
Terfenadine
T1266
Terfenadine is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistamin...
Loratadine
T1097
Loratadine is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical antihistamines...
Levocetirizine Dihydrochloride
T22354
Levocetirizine Dihydrochloride is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine ...
Bepotastine
T7893
Bepotastine free base is a histamine 1 (H1) receptor antagonis.
Antazoline hydrochloride
T0092
Antazoline hydrochloride, a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous histamine.
Mebhydrolin napadisylate
T0113
Mebhydrolin (napadisylate) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.
Mizolastine
T0118
Mizolastine (IC50= 47 nM) is a histamine H1-receptor antagonist.It is used in the treatment of allergic reactions such as hay fever (seasonal allergic rhinitis),...
Irdabisant
T32191
Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R K...
Olopatadine hydrochloride
T1170
Olopatadine hydrochloride is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.
Hydroxyzine dihydrochloride
T2200
Hydroxyzine hydrochloride is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruri...
Meclizine dihydrochloride
T1110
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
Pheniramine maleate
T0370
Pheniramine Maleate, an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase ...
Clemastine fumarate
T0147
Clemastine Fumarate is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
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