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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T2200 Hydroxyzine dihydrochloride 2192-20-3 98%
Hydroxyzine hydrochloride is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruri...
T1110 Meclizine dihydrochloride 1104-22-9 98%
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
T0370 Pheniramine maleate 132-20-7 98%
Pheniramine Maleate, an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase ...
T0147 Clemastine fumarate 14976-57-9 98%
Clemastine Fumarate is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T2520 Desloratadine 100643-71-8 98%
Desloratadine is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histamin...
T0263 Chloropyramine hydrochloride 6170-42-9 98%
Chloropyramine hydrochloride is a histamine receptor H1 antagonist.
T2222 Carbinoxamine Maleate Salt 3505-38-2 98%
Carbinoxamine Maleate is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.
T4566 Lodoxamide 53882-12-5 98%
Lodoxamide is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.
T22879 JNJ 10191584 maleate 869497-75-6 98%
JNJ 10191584 maleate is an orally active and selective antagonist of H4 receptor (Ki = 26 nM). JNJ 10191584 maleate inhibits chemotaxis of eosinophils and mast c...
T19966 Clemastine 15686-51-8 98%
Clemastine is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
T0246L Betahistine mesylate 54856-23-4 98%
Betahistine mesilate is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may ...
T21014 Thonzylamine hydrochloride 63-56-9 98%
Thonzylamine hydrochloride is an anticholinergic and antihistamine used as an antipruritic.
T4551 Acrivastine 87848-99-5 98%
Acrivastine is a short-acting histamine 1 receptor antagonist.
T8514 LML134 1542135-76-1 98%
LML-134 is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).
T6405 Bepotastine Besilate 190786-44-8 98%
Bepotastine is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
T20712 Conessine 546-06-5 98%
Conessine, a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
T4195 Betahistine 5638-76-6 98%
Betahistine is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbat...
T1575 Nizatidine 76963-41-2 98%
Nizatidine is a competitive and reversible histamine H2-receptor antagonist with antacid activity.
T0678 Amitriptyline hydrochloride 549-18-8 98%
Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.
T21390 Fexofenadine 83799-24-0 98%
Fexofenadine, an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. Compared to first-gene...
Hydroxyzine dihydrochloride
T2200
Hydroxyzine hydrochloride is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruri...
Meclizine dihydrochloride
T1110
Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
Pheniramine maleate
T0370
Pheniramine Maleate, an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase ...
Clemastine fumarate
T0147
Clemastine Fumarate is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
Desloratadine
T2520
Desloratadine is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histamin...
Chloropyramine hydrochloride
T0263
Chloropyramine hydrochloride is a histamine receptor H1 antagonist.
Carbinoxamine Maleate Salt
T2222
Carbinoxamine Maleate is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.
Lodoxamide
T4566
Lodoxamide is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.
JNJ 10191584 maleate
T22879
JNJ 10191584 maleate is an orally active and selective antagonist of H4 receptor (Ki = 26 nM). JNJ 10191584 maleate inhibits chemotaxis of eosinophils and mast c...
Clemastine
T19966
Clemastine is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
Betahistine mesylate
T0246L
Betahistine mesilate is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may ...
Thonzylamine hydrochloride
T21014
Thonzylamine hydrochloride is an anticholinergic and antihistamine used as an antipruritic.
Acrivastine
T4551
Acrivastine is a short-acting histamine 1 receptor antagonist.
LML134
T8514
LML-134 is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).
Bepotastine Besilate
T6405
Bepotastine is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
Conessine
T20712
Conessine, a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
Betahistine
T4195
Betahistine is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbat...
Nizatidine
T1575
Nizatidine is a competitive and reversible histamine H2-receptor antagonist with antacid activity.
Amitriptyline hydrochloride
T0678
Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.
Fexofenadine
T21390
Fexofenadine, an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. Compared to first-gene...
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