Home Tools
Log in
Cart

Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T9717 Chlorcyclizine 82-93-9 98.75%
Chlorcyclizine
CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
T22842 HTMT dimaleate 195867-54-0 98.51%
HTMT dimaleate
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.
T27462 GSK-239512 720691-69-0 98.50%
GSK-239512
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
T6562 Latrepirdine dihydrochloride 97657-92-6 98.45%
Latrepirdine dihydrochloride
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
T31195 Dalcotidine 120958-90-9 98.34%
Dalcotidine
Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for bin...
T34709 ST-1006 1196994-11-2 98.31%
ST-1006
ST-1006 is a potent histamine H4 receptor agonist (pKi: 7.94).ST-1006 has anti-inflammatory effects.ST-1006 is a potent inducer of basophil migration and induces...
T11095L DREADD agonist 21 56296-18-5 98.27%
DREADD agonist 21
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
T16778 Rocastine 91833-49-7 98.26%
Rocastine
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
T1278 Astemizole 68844-77-9 98.24%
Astemizole
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 ...
T22624L Carcinine ditrifluoroacetate Acetate 98.18%
Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.
T79500L KSK94 FA 98.13%
KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.
TQ0066 GSK189254A 720690-73-3 98.04%
GSK189254A
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
T1045 Trimipramine maleate 521-78-8 98.02%
Trimipramine maleate
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
T11723L JNJ-39758979 1046447-90-8 98.00%
JNJ-39758979
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, res...
T1030 Triprolidine hydrochloride monohydrate 6138-79-0 98%
Triprolidine hydrochloride monohydrate
Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
T20884 Hydroxyzine 68-88-2 98%
Hydroxyzine
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
T1182 Levocarnitine propionate hydrochloride 119793-66-7 98%
Levocarnitine propionate hydrochloride
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudica...
T7413 JNJ-5207852 398473-34-2 98%
JNJ-5207852
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T7524 Metiamide 34839-70-8 98%
Metiamide
Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .
T4196 Betahistine EP Impurity C 5452-87-9 98%
Betahistine EP Impurity C
Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
Chlorcyclizine
T9717
CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
HTMT dimaleate
T22842
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.
GSK-239512
T27462
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
Latrepirdine dihydrochloride
T6562
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
Dalcotidine
T31195
Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for bin...
ST-1006
T34709
ST-1006 is a potent histamine H4 receptor agonist (pKi: 7.94).ST-1006 has anti-inflammatory effects.ST-1006 is a potent inducer of basophil migration and induces...
DREADD agonist 21
T11095L
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
Rocastine
T16778
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
Astemizole
T1278
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 ...
Carcinine ditrifluoroacetate Acetate
T22624L
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.
KSK94 FA
T79500L
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.
GSK189254A
TQ0066
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
Trimipramine maleate
T1045
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
JNJ-39758979
T11723L
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, res...
Triprolidine hydrochloride monohydrate
T1030
Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
Hydroxyzine
T20884
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
Levocarnitine propionate hydrochloride
T1182
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudica...
JNJ-5207852
T7413
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
Metiamide
T7524
Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .
Betahistine EP Impurity C
T4196
Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
1 2 3 4 5 6 7 8 9 10 11 12
TargetMol