Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T2200	Hydroxyzine dihydrochloride	2192-20-3	98%
T2200	Hydroxyzine hydrochloride is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruri...
T1110	Meclizine dihydrochloride	1104-22-9	98%
T1110	Meclizine hydrochloride is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
T0370	Pheniramine maleate	132-20-7	98%
T0370	Pheniramine Maleate, an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase ...
T0147	Clemastine fumarate	14976-57-9	98%
T0147	Clemastine Fumarate is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T2520	Desloratadine	100643-71-8	98%
T2520	Desloratadine is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histamin...
T0263	Chloropyramine hydrochloride	6170-42-9	98%
T0263	Chloropyramine hydrochloride is a histamine receptor H1 antagonist.
T2222	Carbinoxamine Maleate Salt	3505-38-2	98%
T2222	Carbinoxamine Maleate is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.
T4566	Lodoxamide	53882-12-5	98%
T4566	Lodoxamide is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.
T22879	JNJ 10191584 maleate	869497-75-6	98%
T22879	JNJ 10191584 maleate is an orally active and selective antagonist of H4 receptor (Ki = 26 nM). JNJ 10191584 maleate inhibits chemotaxis of eosinophils and mast c...
T19966	Clemastine	15686-51-8	98%
T19966	Clemastine is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
T0246L	Betahistine mesylate	54856-23-4	98%
T0246L	Betahistine mesilate is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may ...
T21014	Thonzylamine hydrochloride	63-56-9	98%
T21014	Thonzylamine hydrochloride is an anticholinergic and antihistamine used as an antipruritic.
T4551	Acrivastine	87848-99-5	98%
T4551	Acrivastine is a short-acting histamine 1 receptor antagonist.
T8514	LML134	1542135-76-1	98%
T8514	LML-134 is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).
T6405	Bepotastine Besilate	190786-44-8	98%
T6405	Bepotastine is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
T20712	Conessine	546-06-5	98%
T20712	Conessine, a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
T4195	Betahistine	5638-76-6	98%
T4195	Betahistine is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbat...
T1575	Nizatidine	76963-41-2	98%
T1575	Nizatidine is a competitive and reversible histamine H2-receptor antagonist with antacid activity.
T0678	Amitriptyline hydrochloride	549-18-8	98%
T0678	Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.
T21390	Fexofenadine	83799-24-0	98%
T21390	Fexofenadine, an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. Compared to first-gene...