Cat. No. | Product name | CAS No. | Purity | Chemical Structure |
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T26559 | ACT-462206 | 1361321-96-1 | 98% |
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ACT-462206 is an orally available Orexin 1/Orexin 2 receptor antagonist that crosses the blood-brain barrier.ACT-462206 is highly potent and can be used in studi... | ||||
TP1973L | OXA (17-33) acetate | 98% |
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OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM). | ||||
T2710 | TCS 1102 | 916141-36-1 | 98% |
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TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors). |