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Results for "

adenosine kinase inhibitor (hydrate)

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    77
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    2
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Adenosine Kinase Inhibitor (hydrate)
T22554
Adenosine kinase is the key metabolizing enzyme regulating cellular adenosine concentrations. Inhibition of adenosine kinase can selectively enhance the protective actions of adenosine during tissue trauma without producing the nonspecific effects associa
  • $80
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AKT Kinase Inhibitor
T10276842148-40-7In house
AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.
  • $138
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AKT Kinase Inhibitor HCl
T10276L In house
AKT Kinase Inhibitor HCl is an Akt inhibitor with antitumor activity.
  • $138
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FLT3 kinase inhibitor 2HCl
T500722411178-94-2
3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride is used in the synthesis of various compounds.
  • $95
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mTOR kinase Inhibitor 2
T93151021917-65-6In house
2H-Imidazo[4,5-b]pyrazin-2-one, 1,3-dihydro-6-[6-(1-hydroxy-1-methylethyl)-3-pyridinyl]-1-[(tetrahydro-2H-pyran-4-yl)methyl]- is a potent mTOR inhibitor with IC50 of 0.176 μM and >30 μM for mTOR and PI3Kα, respectively.
  • $148
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mTOR kinase Inhibitor 1
T9311321557-16-8In house
can be used in research in the fields of chemistry and life sciences.
  • $148
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CaM kinase II inhibitor TFA salt
TP1216
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
  • $177
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Pim-1 kinase inhibitor 4
T77526
Pim-1 kinase inhibitor 4 is a potent Pim-1 kinase inhibitor with an IC50 value of 17.01 nM.Pim-1 kinase inhibitor 4 also possesses antioxidant activity and potential anticancer activity, and inhibits DPPH.Pim-1 kinase inhibitor 4 promotes apoptosis and inhibits the growth of PC-3 cells with an IC50 value of 16 nM. Pim-1 kinase inhibitor 4 promotes apoptosis and inhibits PC-3 cell growth with an IC50 of 16 nM. Pim-1 kinase inhibitor 4 can be used in prostate cancer research.
  • $195
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Casein Kinase II Inhibitor IV
T10687863598-09-8In house
Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.
  • $79
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RIP2 Kinase Inhibitor 3
T127281398053-50-3In house
RIP2 Kinase Inhibitor 3 is a potent and selective inhibitor of RIP2, demonstrating an IC50 of 1 nM.
  • $53
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EML4-ALK kinase inhibitor 1
T111841373409-08-5In house
EML4-ALK kinase inhibitor 1 (EML4 ALK kinase inhibitor 1) is a potent oral active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (EML4-ALK), with an IC50 of 1 nM.
  • $88
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Thymidylate Kinase Inhibitor, YMU1
T8864902589-96-2
YMU1 is a human thymidylate kinase (hTMPK) inhibitor. YMU1 stabilizes the conformation of ligand-induced degradation (LID) region of hTMPK and blocks the catalytic site or ATP-binding site.
  • $31
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Protein kinase G inhibitor-2
T9940612829-80-8
Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities.
  • $33
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Multi-kinase inhibitor 1
T4191778274-97-8
Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.
  • $33
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ALK kinase inhibitor-1
T64091462949-64-9
SAR348830 is an ALK inhibitor, targeting anaplastic lymphoma kinase.
  • $41
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TAO Kinase inhibitor 1
T16987850467-66-2
TAO Kinase inhibitor 1 delays mitosis and induces mitotic cell death. TAO Kinase inhibitor 1 is a selective and ATP-competitive thousand-and-one amino acid kinases inhibitor (IC50s: 11 to 15 nM for TAOK1 and 2, respectively).
  • $64
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Protein kinase inhibitor 6
T9779348-45-8
Protein kinase inhibitor 6 (PKI 6) is a compound that acts as an inhibitor of protein kinases.
  • $50
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Protein kinase inhibitor H-7
T6010984477-87-2
Protein kinase inhibitor H-7 (5-(2-methylpiperazine-1-sulfonyl)isoquinoline) is a potent inhibitor of protein kinase C (PKC) with a Ki of 6 μM. Protein kinase inhibitor H-7 is also a cyclic nucleotide dependent protein kinase inhibitor.
  • $52
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Aurora kinase inhibitor-3
T5524879127-16-9
Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK, IGF-1R, c-Src, TRKB, SYK, and EGFR.
  • $71
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IRAK-4 protein kinase inhibitor 2
T9631301675-24-1
IRAK-4 protein kinase inhibitor 2 is a potent inhibitor of interleukin-1 receptor-associated kinase-4 (IC50 = 4 μM).
  • $39
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Aurora kinase inhibitor-2
T9040331770-21-9
Aurora kinase inhibitor-2 (IUN-70219) is a cell-permeable anilinoquinazoline that inhibit the activity of Aurora A (IC50 = 0.39 M).
  • $100
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Adenosine receptor inhibitor 1
T618502550400-52-5
Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR), exhibiting exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory, and peripheral analgesic properties, holding great promise for investigating cancer and neurodegenerative diseases [1].
  • $1,520
6-8 weeks
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Tie2 kinase inhibitor 1
T6335948557-43-5
Tie2 kinase inhibitor 1 (Tie2 kinase inhibitor), an optimized compound of SB-203580, is selective to Tie2 with IC50 of 0.25 μM, which is 200-fold more effective than p38.
  • $62
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Tyrosine kinase inhibitor
T171841021950-26-4
Tyrosine kinase inhibitor is a tyrosine kinase inhibitor used in combination with fragmenting aromatic nitrogen compounds as antiproliferative agents.
    7-10 days
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    Protein kinase inhibitor H-7 dihydrochloride
    T22831108930-17-2
    Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor. Protein kinase inhibitor H-7 dihydrochloride (100 μM) significantly inhibits TPA (skin tumor promoter, 12-O-tetradecanoylphorbol-13-acetate) and phospholipase C-induced ODC (ornithine decarboxylase) inhibited PMA-induced promiscuity cell lysis activity.
    • $45
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    Casein Kinase inhibitor A86
    T394822079069-01-3
    Casein Kinase inhibitor A86 is a highly effective and orally bioavailable inhibitor of casein kinase 1α (CK1α) and also inhibits CDK7 (TFIIH) and CDK9 (P-TEFb). It induces apoptosis in leukemia cells, exhibiting substantial anti-leukemic effects.
      7-10 days
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      Adenosine 5’-methylenediphosphate (hydrate)
      T35573
      Adenosine 5’-methylenediphosphate is an inhibitor of ecto-5’-nucleotidase, also known as CD73, with a Kivalue of 37 nM.1It inhibits cAMP accumulation induced by adenosine 5’-monophosphate , adenosine 5’-diphosphate , or adenosine 5’-triphosphate but not adenosine in VA-13 human fibroblasts when used at a concentration of 100 μM. Adenosine 5’-methylenediphosphate reduces proliferation of U138MG glioma cells, as well as inhibits the invasion and migration of MHCC97H hepatocellular carcinoma (HCC) cells in a migration assay.2,3It increases tumor infiltration of CD3+CD8+T cells and reduces tumor growth in a K1735 murine melanoma model when administered at a dose of 400 μg/mouse.4 1.Bruns, R.F.Adenosine receptor activation by adenine nucleotides requires conversion of the nucleotides to adenosineNaunyn Schmiedebergs Arch. Pharmacol.315(1)5-13(1980) 2.Braganhol, E., Tamajusuku, A.S.K., Bernardi, A., et al.Ecto-5′-nucleotidase/CD73 inhibition by quercetin in the human U138MG glioma cell lineBiochim. Biophys. Acta1770(9)1352-1359(2007) 3.Shali, S., Yu, J., Zhang, X., et al.Ecto\5′\nucleotidase (CD73) is a potential target of hepatocellular carcinomaJ. Cell Physiol.234(7)10248-10259(2018) 4.Forte, G., Sorrentino, R., Montinaro, A., et al.Inhibition of CD73 improves B cell-mediated anti-tumor immunity in a mouse model of melanomaJ. Immunol.189(5)2226-2233(2021)
      • $57
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      Adenosine 3’-monophosphate (sodium salt hydrate)
      T35571
      Adenosine 3’-monophosphate is a nucleotide and metabolite formedviahydrolysis of 2’,3’-cAMP by metal-dependent phosphodiesterases.1It reduces proliferation of rat preglomerular vascular smooth muscles cells (PGVSMCs) and glomerular mesangial cells (GMCs) in a concentration-dependent manner, an effect that is abolished by the adenosine A2Breceptor antagonist MRS1754.2Adenosine 3’-monophosphate is also a metabolic intermediate in the biosynthesis of adenosine .
      • $51
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      RIP2 kinase inhibitor 2
      T167531581270-11-2
      RIP2 kinase inhibitor 2 is a compound that inhibits receptor-interacting protein-2 kinase (RIP2).
      • $196
      5 days
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      EGFR kinase inhibitor 1
      T636482413958-04-8
      EGFR kinase inhibitor 1 is a potent inhibitor of EGFR that acts on WT (IC50: 37 nM), l885R T790M (IC50: 1.7 nM), and L858R T790M C797S (IC50>300 nM). It is capable of blocking the cell cycle in G0 G1 phase, inducing apoptosis, and has an inhibitory effect on cell metastasis. Additionally, EGFR kinase inhibitor 1 exhibits anti-proliferative and anti-tumor effects.
      • $1,520
      8-10 weeks
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      RIP1 kinase inhibitor 7
      T790442428401-23-2
      RIP1 Kinase Inhibitor 7 (Compound 41) serves as a potent inhibitory agent for receptor interacting protein 1 kinase (RIP1) with an IC50 of under 100 nM. Additionally, it demonstrates an EC50 ranging from 1 to 100 nM in cell necrosis assays [1].
      • $1,520
      6-8 weeks
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      RIP1 kinase inhibitor 4
      T790412919836-00-1
      RIP1 Kinase Inhibitor 4 (Compound 3) is an effective inhibitor of RIP1K, exhibiting an EC50 of ≤ 1000 nM [1].
      • $1,820
      8-10 weeks
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      PDGFRα kinase inhibitor 1
      T123962209053-93-8
      PDGFRα kinase inhibitor 1 is a highly selective inhibitor of type II PDGFRα kinase (PDGFRα and PDGFRβ) with IC50 values of 132 nM and 6115 nM, respectively.
      • $399
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      Pim-1 kinase inhibitor 1
      T609722803505-57-7
      Pim-1 kinase inhibitor 1 can be used in cancer research, showing anticancer activity against a variety of cancer cell lines by promoting cell apoptosis. Pim-1 kinase inhibitor 1 is an inhibitor of Pim-1 kinase with an IC 50 value of 0.11 μM [1].
      • $1,520
      6-8 weeks
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      AKT Kinase Inhibitor hydrochloride
      T72104
      AKT Kinase Inhibitor hydrochloride is an Akt kinase inhibitor exhibiting anti-tumor activity.
      • $1,530
      1-2 weeks
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      Pim-1 kinase inhibitor 6
      T872132928606-69-1
      • Inquiry Price
      10-14 weeks
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      EGFR kinase inhibitor 3
      T863412922402-03-5
      • Inquiry Price
      10-14 weeks
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      Adenosine receptor inhibitor 2
      T620182550401-76-6
      Adenosine receptor inhibitor 2 (compound 14b) is a potent inhibitor of AR (adenosine receptor), exhibiting dual affinity towards A1 A2A ARs with higher affinity for A1- than A2A AR, and Ki values of 52.2 nM for A1 AR and 167 nM for A2A AR.
      • $1,520
      6-8 weeks
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      Tpl2 Kinase Inhibitor 1
      T17145871307-18-5
      Tpl2 Kinase Inhibitor 1 is an effective and selective Tpl2 inhibitor.
      • $143
      35 days
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      p38 MAP Kinase Inhibitor IV
      T360111638-41-1
      p38 MAPK inhibitor IV is an ATP-competitive inhibitor of p38 MAP kinases with IC50 values of 0.13, 0.55, 5.47, and 8.63 μM for p38α, p38β, p38x, and p38δ, respectively, in vitro.[1] It also inhibits LPS-induced TNF-α and IL-1β cytokine production (IC50s = 22 and 44 nM, respectively) in human peripheral blood mononuclear cells.
      • $155
      35 days
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      Pim-1 kinase inhibitor 10
      T872122918764-57-3
        10-14 weeks
        Inquiry
        TAO Kinase inhibitor 2
        T77501850467-77-5
        TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
        • $30
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        Protein kinase inhibitor peptide
        TP2349128022-93-5
        Protein kinase inhibitor peptide matches the inhibitory domain of the heat-stable protein kinase inhibitor.
        • Inquiry Price
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        Protein kinase G inhibitor-1
        T67755354544-70-0
        Protein kinase G inhibitor-1 is a potent Protein kinase G inhibitor, IC50= 0.9 uM.
        • $195
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        Protein kinase D inhibitor 1
        T611632489320-03-6
        Protein kinase D inhibitor 1 (compound 17m) is a potent pan-PKD inhibitor with IC50 values between 17 and 35 nM, demonstrating inhibitory activity in the low nanomolar range. By inhibiting protein kinase D, it effectively suppresses PKD-dependent cortactin phosphorylation [1].
        • $1,520
        6-8 weeks
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        RIP2 kinase inhibitor 1
        T127272380028-10-2
        RIP2 kinase inhibitor 1 is a potent and selective receptor interacting inhibitor of protein 2 (RIP2) kinase(RIP2 FP with an IC50 of 0.03 μM ),and is used for autoinflammatory disorders.
        • $2,120
        8-10 weeks
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        Pim-1 kinase inhibitor 5
        T789802928606-67-9
        Pim-1 kinase inhibitor 5 (Compound 4c) has an IC50 of 0.61 μM and exhibits cytotoxicity against cancer cell lines HepG2, MCF-7, PC3, and HCT-116, with IC50 values ranging from 6.95 to 20.19 μM [1].
        • Inquiry Price
        8-10 weeks
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        Protein kinase inhibitor 5 sulfate hydrate
        T79126
        Protein kinase inhibitor 5 sulfate hydrate, a potent TRK-A inhibitor, exhibits an IC50 of 1.8 nM and impairs cell viability [1].
        • Inquiry Price
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        Aurora kinase inhibitor-9
        T627892419107-09-6
        Aurora kinase inhibitor-9 (compound 9d) is a potent AURKA B bipolar kinase inhibitor with an IC50 of 0.093 μM for Aurora A and 0.09 μM for Aurora B, demonstrating broad-spectrum anti-proliferative activity.
        • $1,520
        6-8 weeks
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        Pim-1/2 kinase inhibitor 2
        T872142918764-16-4
        • Inquiry Price
        10-14 weeks
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