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Search Result

Search Results for " antiestrogenic "

Targets

Estrogen Receptor/ERR Estrogen/progestogen Receptor

12

Compounds

5

Natural Products

5

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T8984 FLTX1 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under permeabilized and non-permeabilized conditions. Additionally,...
T2569 Chlorotrianisene tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE Estrogen Receptor/ERR , Estrogen/progestogen Receptor , COX
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor modulator (SERM), with predominantly estrogenic but...
T11200 Endoxifen (E-isomer) E-Endoxifen,Endoxifen E-isomer Estrogen Receptor/ERR
Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.
T13415 Zuclomiphene citrate Others
Zuclomiphene citrate is a cis isomer of Clomiphene citrate, and has an antiestrogenic effect and can inhibit the secretion of luteinizing hormone (LH) more than the trans isomer.
T26154 RU 45144 RU45144,RU-45144
RU 45144 is an estradiol derivative with antiestrogenic activity.
T27884 LY 183648 LY-183648,LY183648
LY 183648 has antiestrogenic activity. LY117018 inhibited PAIII metastasis to the gluteal (97%) and iliac lymph nodes (88%).
T12312 OP-1074 Estrogen/progestogen Receptor
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
T61161 HIF-1α-IN-3
HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].
T9796 22393-62-0_peak 2
22393-62-0_peak 2 exhibits some aspects of the antiestrogenic activity and other actions that may be connected to the estrogenic properties. A mixture of the (Z)- and (E)-isomers (Broparestrol, INN) is used in dermatol...
T39259 Arzoxifene LY353381,Arzoxifene,SERMIII
Arzoxifene (LY353381) is an orally active selective estrogen receptor modulator (SERM) exhibiting a fixed ring structure analogous to raloxifene. This compound demonstrates potent antiestrogenic effects on breast cancer ...
T12148L N-Desmethyltamoxifen Others
N-Desmethyltamoxifen, the principal metabolite of tamoxifen in humans, serves as an efficacious modulator of ceramide metabolism within human AML cells by inhibiting ceramide glycosylation, hydrolysis, and sphingosine ph...
T69696 TAS-108 citrate
TAS-108, also known as SR16234, is a synthetic, antiestrogenic steroidal compound with potential antitumor activity. TAS-108 binds to and inhibits estrogenic receptor alpha (ERa), mainly expressed in the mammary gland an...
Cat No. Product Name Synonyms Targets
T3855 Tracheloside Estrogen Receptor/ERR , Phosphorylase
Tracheloside significantly decreases the activity of alkaline phosphatase (IC50: 0.31 μg/ml), a level of inhibition comparable to that of tamoxifen (IC50: 0.43 μg/ml).
T7999 7-Hydroxyflavanone Anti-infection
7-Hydroxyflavanone shows antimicrobial activity against Streptococcus pneumoniae clinical isolates.
TN4565 Millewanin G Others
Millewanin G shows antiestrogenic activity.
TN4566 Millewanin H Others
Millewanins H shows antiestrogenic activity.
TN4731 Pachyaximine A Antifection
Pachyaximine A possesses significant antibacterial activity against Escherichia coli, Staphylococcus aureus, Corynebacterium diphtheriae and Corynebacterium pyrogenes. (-)-Pachyaximine A demonstrates significant activity...

Natural Products

Tracheloside
T3855
Synonym:
Target: Estrogen Receptor/ERR, Phosphorylase
7-Hydroxyflavanone
T7999
Synonym:
Target: Anti-infection
Millewanin G
TN4565
Synonym:
Target: Others
Millewanin H
TN4566
Synonym:
Target: Others
Pachyaximine A
TN4731
Synonym:
Target: Antifection

Recombinant Proteins

Species：
Human (3)
Rat (1)
Rhesus (1)
Expression System：
HEK293 (4)
Baculovirus-Insect Cells (1)
Tag：
hFc (3)
His (1)
His,hFc (1)
Cat No. Product Name Species Expression System
TMPY-05157 TGFBR2 Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
TGFBR2 is a member of the Ser/Thr protein kinase family and the TGFB receptor subfamily. It is a transmembrane protein. TGFBR2 is comprised of a C-terminal protein kinase domain and an N-terminal ectodomain. The ectodoma...
TMPY-05508 TGFBR2 Protein, Human, Recombinant (hFc) Human HEK293
TGFBR2 is a member of the Ser/Thr protein kinase family and the TGFB receptor subfamily. It is a transmembrane protein. TGFBR2 is comprised of a C-terminal protein kinase domain and an N-terminal ectodomain. The ectodoma...
TMPY-03082 TGFBR2 Protein, Rat, Recombinant (hFc) Rat HEK293
TGFBR2 is a member of the Ser/Thr protein kinase family and the TGFB receptor subfamily. It is a transmembrane protein. TGFBR2 is comprised of a C-terminal protein kinase domain and an N-terminal ectodomain. The ectodoma...
TMPY-03171 TGFBR2 Protein, Rhesus, Recombinant (hFc) Rhesus HEK293
TGFBR2 is a member of the Ser/Thr protein kinase family and the TGFB receptor subfamily. It is a transmembrane protein. TGFBR2 is comprised of a C-terminal protein kinase domain and an N-terminal ectodomain. The ectodoma...
TMPY-05810 TGFBR2 Protein, Human, Recombinant (His & hFc), Biotinylated Human HEK293
TGFBR2 is a member of the Ser/Thr protein kinase family and the TGFB receptor subfamily. It is a transmembrane protein. TGFBR2 is comprised of a C-terminal protein kinase domain and an N-terminal ectodomain. The ectodoma...
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