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ar-c126313

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  • Inhibitors & Agonists
    3
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AR-C126313
ARC126313,AR C126313
T30120216657-60-2
AR-C126313 is a thiouracil derivative.
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AR-C 141990 hydrochloride
T37822
Monocarboxylate transporter (MCT1) inhibitor (pKi = 7.6. Exhibits approximately 10-fold selectivity for MCT1 over MCT2 and no significant activity against MCT3 or 4. Inhibits graft versus host response and prolongs cardiac graft survival in a rat model. Immunosuppressant. Also inhibits brain penetration of GHB analog HOCPCA.
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AR-C 102222
T22580253771-21-0
AR-C 102222 is an iNOS inhibitor.
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6-8 weeks
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