bp3

163-bp3 is an effective photoaffinity probe and can be used as a target γ Secretory enzyme.

PROTAC HSP90 degrader BP3 potently and selectively degrades HSP90 through a CRBN-dependent mechanism. It effectively diminishes HSP90 protein levels in MCF-7 cells with a half-maximal degradation concentration (DC50) of 0.99 µM. Additionally, this compound impedes the proliferation of breast cancer cells [1].

MGB-BP-3 is a synthetic antibiotic with bactericidal activity that inhibits bacterial DNA replication and can be used to study recurrent C. difficile infections.

SGC-CBP30 is an effective CREBBP/EP300 inhibitor (IC50: 21/38 nM).

UBP310 (UBP 310) is a GLUK5 kainate receptor antagonist

BIBP3226 is a potent and selective antagonist for the Neuropeptide Y receptor Y1 and the neuropeptide FF receptor.

UBP301 is a kainate receptor antagonist.

BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF).

GluR5-containing kainate receptor antagonist