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Inhibitors & Agonists

cmpd 101

" in TargetMol Product Catalog

Inhibitors & Agonists
1

CMPD101

T14989865608-11-3

CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2 3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with IC50s of 3.1 μM , 2.3 μM, 1.4 μM and 8.1 μM, respectively.

ROCK GRK PKC

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