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(1)
By Target- Apelin receptor
- Arrestin(1)
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Results for "
ml221
" in TargetMol Product Catalog- Inhibitors & Agonists1
ML221
Cited
T4390877636-42-5
ML221 is a potent apelin APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.
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