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protein kinase inhibitor h-7

" in TargetMol Product Catalog
  • Inhibitor Products
    138
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    124
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Protein kinase inhibitor H-7
T6010984477-87-2
Protein kinase inhibitor H-7 (5-(2-methylpiperazine-1-sulfonyl)isoquinoline) is a potent inhibitor of protein kinase C (PKC) with a Ki of 6 μM. Protein kinase inhibitor H-7 is also a cyclic nucleotide dependent protein kinase inhibitor.
  • $52
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Protein kinase inhibitor H-7 dihydrochloride
T22831108930-17-2
Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor. Protein kinase inhibitor H-7 dihydrochloride (100 μM) significantly inhibits TPA (skin tumor promoter, 12-O-tetradecanoylphorbol-13-acetate) and phospholipase C-induced ODC (ornithine decarboxylase) inhibited PMA-induced promiscuity cell lysis activity.
  • $45
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AKT Kinase Inhibitor
T10276842148-40-7In house
AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.
  • $138
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Tyrosine kinase-IN-7
T77746345615-74-9
Tyrosine kinase-IN-7 is a potent inhibitor of the tyrosine kinase EGFR, inhibiting EGFR(WT) and EGFR(T790M) and showing anti-cancer and anti-tumor activity in a variety of cancer cell lines. Tyrosine kinase-IN-7 has potential anti-inflammatory and antiviral activities.
  • $30
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AKT Kinase Inhibitor HCl
T10276L In house
AKT Kinase Inhibitor HCl is an Akt inhibitor with antitumor activity.
  • $138
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Protein kinase inhibitors 1 hydrochlorid
T4692
Protein kinase inhibitors 1 hydrochlorid (Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))) is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
  • $37
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T.cruzi Inhibitor (1350920-22-7(free base))
T4248
T.cruzi Inhibitor is a Trypanosoma cruzi inhibitor.
  • $35
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URAT1 inhibitor 7
T775171632002-28-8
URAT1 inhibitor 7 is a novel and potent inhibitor of the human uric acid transporter protein URAT1 (IC50:12 nM).URAT1 inhibitor 7 inhibits CYP2C9 with an IC50 of 4.2 μM.URAT1 inhibitor 7 can be used to study hyperuricemia and gout.
  • $195
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FLT3 kinase inhibitor 2HCl
T500722411178-94-2
3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride is used in the synthesis of various compounds.
  • $95
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mTOR kinase Inhibitor 2
T93151021917-65-6In house
2H-Imidazo[4,5-b]pyrazin-2-one, 1,3-dihydro-6-[6-(1-hydroxy-1-methylethyl)-3-pyridinyl]-1-[(tetrahydro-2H-pyran-4-yl)methyl]- is a potent mTOR inhibitor with IC50 of 0.176 μM and >30 μM for mTOR and PI3Kα, respectively.
  • $148
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CaM kinase II inhibitor TFA salt
TP1216
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
  • $177
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Calmodulin-Dependent Protein Kinase II 290-309 acetate
TP1271L
Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).
  • $221
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mTOR kinase Inhibitor 1
T9311321557-16-8In house
can be used in research in the fields of chemistry and life sciences.
  • $148
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Pim-1 kinase inhibitor 4
T77526
Pim-1 kinase inhibitor 4 is a potent Pim-1 kinase inhibitor with an IC50 value of 17.01 nM.Pim-1 kinase inhibitor 4 also possesses antioxidant activity and potential anticancer activity, and inhibits DPPH.Pim-1 kinase inhibitor 4 promotes apoptosis and inhibits the growth of PC-3 cells with an IC50 value of 16 nM. Pim-1 kinase inhibitor 4 promotes apoptosis and inhibits PC-3 cell growth with an IC50 of 16 nM. Pim-1 kinase inhibitor 4 can be used in prostate cancer research.
  • $195
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Protein Kinase C 19-31 acetate
TP1053L
Protein Kinase C 19-31 acetate, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate
  • $51
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Protein Kinase C Peptide Substrate acetate
TP1051L
Protein Kinase C Peptide Substrate acetate targets specific cell spacers ina manner that is dependent on second messengers and specific adaptor proteins in response to extracellular signals that activate g protein-coupled receptors, tyrosine Kinase recept
  • $133
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PI3Kα Inhibitor 7
T93121239978-63-2In house
PI3Kα Inhibitor 7 is a useful organic compound for research related to life sciences. The catalog number is T9312 and the CAS number is 1239978-63-2.
    8-10 weeks
    Inquiry
    Casein Kinase II Inhibitor IV
    T10687863598-09-8In house
    Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.
    • $79
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    PROTAC(H-PGDS)-7
    T412672761281-50-7In house
    PROTAC(H-PGDS)-7 is a selective and potent small molecule hematopoietic prostaglandin D synthase (H-PGDS) PROTAC degradation agent that exhibits degradation activity in KU812 cells with a DC50 of 17.3 pM. PROTAC(H-PGDS)-7 is a pharmacological compound that effectively inhibits prostaglandin D2 (PGD2) PROTAC(H-PGDS)-7 is a candidate compound for the treatment of DMD and other H-PGDS-related diseases.
    • $493
    35 days
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    RIP2 Kinase Inhibitor 3
    T127281398053-50-3In house
    RIP2 Kinase Inhibitor 3 is a potent and selective inhibitor of RIP2 with an IC50 of 1 nM.
    • $53
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    c-Myc inhibitor 7
    T720402883535-99-5In house
    C-Myc Inhibitor 7, serving as both a c-Myc inhibitor and a multi-target protein degrader, effectively degrades proteins c-MYC, CK1α, GSPT1, and IKZF1/2/3 across various tumor cell types. It holds potential for research into diseases associated with high c-Myc expression, including cancer, cardiovascular and cerebrovascular conditions, and viral infections.
    • $1,520
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    EML4-ALK kinase inhibitor 1
    T111841373409-08-5In house
    EML4-ALK kinase inhibitor 1 (EML4 ALK kinase inhibitor 1) is a potent oral active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (EML4-ALK), with an IC50 of 1 nM.
    • $88
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    Thymidylate Kinase Inhibitor, YMU1
    T8864902589-96-2
    YMU1 is a human thymidylate kinase (hTMPK) inhibitor. YMU1 stabilizes the conformation of ligand-induced degradation (LID) region of hTMPK and blocks the catalytic site or ATP-binding site.
    • $31
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    Protein kinase G inhibitor-2
    T9940612829-80-8
    Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities.
    • $33
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    KRAS G12D inhibitor 7
    T402822648552-34-3
    KRAS G12D inhibitor 7, is a highly potent inhibitor specifically targeting KRAS G12D.
    • $970
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    pTH-Related Protein (7-34) amide (human, mouse, rat)
    T81349115695-30-2
    PTH-Related Protein (7-34) amide (human, mouse, rat) serves as a potent antagonist of parathyroid hormone (PTH) [1].
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    prostate apoptosis response protein PAR-4 (2-7) [Homo sapiens]
    T23189
    Prostate apoptosis response protein PAR-4 (2-7) [Homo sapiens] is a peptide with the sequence H2N-Ala-Thr-Gly-Gly-Tyr-Arg-OH, MW= 623.66.
    • $50
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    KRAS mutant protein inhibitor 1
    T402722642305-16-4
    KRAS mutant protein inhibitor 1 is a KRAS mutant protein inhibitor for potential treatment in cancer.
    • $970
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    TAO Kinase inhibitor 2
    T77501850467-77-5
    TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
    • $30
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    Protein kinase inhibitor peptide
    TP2349128022-93-5
    Protein kinase inhibitor peptide matches the inhibitory domain of the heat-stable protein kinase inhibitor.
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    JAMM protein inhibitor 2 
    T9892848249-35-4
    JAMM protein inhibitor 2 (Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-) is an inhibitor of JAMM protease and can be used for anticancer studies. The IC50s are 10 μM, 46 μM, and 89 μM for thrombin, Rpn11, and MMP2, respectively.
    • $116
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    Multi-kinase inhibitor 1
    T4191778274-97-8
    Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.
    • $33
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    Multi-target kinase inhibitor 2
    T81739
    Compound 5K (Multi-target kinase inhibitor 2) is a multi-targeted kinase inhibitor demonstrating activity against EGFR, Her2, VEGFR2, and CDK2 with IC50 values between 40 to 204 nM. It exhibits cytotoxic effects on HepG2, HeLa, MDA-MB-231, and MCF-7 cell lines, with IC50 values of 41, 57, 51, and 59 μM, respectively. Additionally, it induces cell cycle arrest and apoptosis specifically in HepG2 cells.
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    Pim-1 kinase inhibitor 8
    T83627916038-47-6
    Pim-1 kinase inhibitor 8 is a potent Pim-1 kinase inhibitor with anticancer activity and can effectively inhibit cell migration.Pim-1 kinase inhibitor 8 is cytotoxic to MCF-7 and HepG2 cells, and is a candidate compound for breast cancer research.
    • $57
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    (Asn10,Leu11,D-Trp12)-pTH-Related Protein (7-34) amide (human, mouse, rat)
    T76586129622-68-0
    (Asn10,Leu11,D-Trp12)-pTH-Related Protein (7-34) amide (human, mouse, rat) is a potent antagonist of the PTH-1R [1] [2].
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    Protein kinase G inhibitor-1
    T67755354544-70-0
    Protein kinase G inhibitor-1 is a potent Protein kinase G inhibitor, IC50= 0.9 uM.
    • $195
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    KRAS G12C mutant protein inhibitor A-1
    T778052658538-04-4
    KRAS G12C mutant protein inhibitor A-1 can be used in studies about Ras.
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    Protein kinase inhibitor 6
    T9779348-45-8
    Protein kinase inhibitor 6 is a protein kinase inhibitor.
    • $50
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    Tpl2 Kinase Inhibitor (hydrochloride)
    T35536
    Tpl2 kinase inhibitor is an inhibitor of tumor progression locus 2 (Tpl2; IC50= 0.05 μM).1It is selective for Tpl2 over MEK, p38 MAPK, Src, MK2, and PKC (IC50s = >40, 180, >400, 110, and >400 μM, respectively). Tpl2 kinase inhibitor inhibits LPS-induced TNF-α production in isolated human monocytes and whole blood (IC50s = 0.7 and 8.5 μM, respectively). It enhances differentiation induced by calcitriol in HL-60 and U937 leukemia cells when used at a concentration of 5 μM.2Tpl2 kinase inhibitor (5 μM) inhibits the proliferation of KG-1a leukemia cells.3 1.Garvin, L.K., Green, N., Hu, Y., et al.Inhibition of Tpl2 kinase and TNF-α production with 1,7-naphthyridine-3-carbonitriles: Synthesis and structure-activity relationshipsBioor. Med. Chem. Lett.15(23)5288-5292(2005) 2.Wang, X., and Studzinski, G.P.Expression of MAP3 kinase COT1 is up-regulated by 1,25-dihydroxyvitamin D3 in parallel with activated c-jun during differentiation of human myeloid leukemia cellsJ. Steroid. Biochem. Mol. Biol.121(1-2)395-398(2010) 3.Wang, X., Gocek, E., Novik, V., et al.Inhibition of Cot1/Tlp2 oncogene in AML cells reduces ERK5 activation and up-regulates p27Kip1 concomitant with enhancement of differentiation and cell cycle arrest induced by silibinin and 1,25-dihydroxyvitamin D3Cell Cycle9(22)4542-4551(2010)
    • $143
    35 days
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    IRAK-4 protein kinase inhibitor 2
    T9631301675-24-1
    IRAK-4 protein kinase inhibitor 2 is a potent interleukin-1 receptor-associated kinase-4 (IRAK-4) inhibitor(IC50 = 4 μM).
    • $39
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    Protein Kinase C (19-31) (TFA)(121545-65-1,free)
    TP1052
    Protein Kinase C (19-31) TFA, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate p
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    RIP2 Kinase Inhibitor 4
    T395742126803-41-4
    RIP2 Kinase Inhibitor 4 is a highly potent and selective RIPK2 PROTAC compound that efficiently degrades RIPK2 (with a pIC50 value of 8) and effectively inhibits the release of TNF-α.
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    Tie2 kinase inhibitor 1
    T6335948557-43-5
    Tie2 kinase inhibitor 1 (Tie2 kinase inhibitor), an optimized compound of SB-203580, is selective to Tie2 with IC50 of 0.25 μM, which is 200-fold more effective than p38.
    • $62
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    Tyrosine kinase inhibitor
    T171841021950-26-4
    Tyrosine kinase inhibitor is a tyrosine kinase inhibitor used in combination with fragmenting aromatic nitrogen compounds as antiproliferative agents.
      7-10 days
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      Calmodulin-Dependent Protein Kinase II (290-309)
      TP1271115044-69-4
      Calmodulin-Dependent Protein Kinase II (290-309) is a potent CaMK antagonist with an IC50 of 52 nM for inhibition of Ca2+/calmodulin-dependent protein kinase II.
      • $270
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      PI3K/mTOR Inhibitor-7
      T640412456295-65-9
      PI3K/mTOR Inhibitor-7 is a potent dual PI3K/mTOR inhibitor. PI3K/mTOR Inhibitor-7 is 4.7-fold more potent than gedatolisib, with IC50 values of 1.4 μM and 0.3 μM, respectively. 10 μM of PI3K/mTOR Inhibitor-7 is able to significantly inhibit the PI3K/Akt/mTOR signalling pathway. PI3K/mTOR Inhibitor-7 has shown potential for research in cancer diseases.
      • $1,520
      8-10 weeks
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      Topoisomerase I inhibitor 7
      T620022408639-81-4
      Topoisomerase I inhibitor 7 (Compound 8) is a potent inhibitor of Topoisomerase I. Topoisomerase I inhibitor 7 significantly inhibits tumor growth (up to 79%) and increases the lifespan (153%) of mice bearing P388 lymphoma transplants.
      • $1,520
      6-8 weeks
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      Protein kinase affinity probe 1
      T125622098621-90-8
      Protein kinase affinity probe 1 is a protein kinase affinity probe for the functional identification of protein kinases (PKs).
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      Protein kinase C α peptide TFA
      T76388159939-84-1
      Protein Kinase C (alpha) Peptide (TFA) is a PKC-α-associated peptide functioning as a lipid-dependent serine/threonine protein kinase. It plays a pivotal role in regulating several cellular functions such as survival, proliferation, differentiation, migration, and adhesion [1].
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      Protein Kinase C (19-35) Peptide
      T76456309247-48-1
      Protein Kinase C (19-35) Peptide, serving as the PKC pseudosubstrate inhibitor/region, potentially inhibits PKC activity by obstructing the substrate-binding site within its kinase domain, rendering the cytoplasmic form of PKC inactive [1] [2].
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