T15809 |
LY2812223
|
1311385-20-2
|
98%
|
|
LY2812223 is a highly effective and functionally selective mGlu2 receptor agonist. It has a mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, res...
|
T7128 |
TH-257
|
2244678-29-1
|
98%
|
|
TH 257 is a Potent and selective allosteric LIMK 1/2 inhibitor(LIMK1 and LIMK2, IC50 of 84 nM and 39 nM).
|
T3960 |
T56-LIMKi
|
924473-59-6
|
98%
|
|
T56-LIMKi is a selective inhibitor of LIMK2.
|
T4598 |
BMS-5
|
1338247-35-0
|
98%
|
|
BMS-5 is a potent LIMK inhibitor with IC50s of 7 nM and 8 nM for LIMK1 and LIMK2, respectively.
|
T12609 |
R-10015
|
2097938-51-5
|
98%
|
|
R-10015 is a potent and selective inhibitor of LIM domain kinase (LIMK) and binds to the ATP-binding pocket(IC50 of 38 nM for human LIMK1),and a broad-spectrum a...
|
T24410 |
LIMK-IN-22j
|
1116571-01-7
|
98%
|
|
LIMK-IN-22j is an effective and selective inhibitor of LIMK.
|
T4600 |
BMS-3
|
1338247-30-5
|
98%
|
|
BMS-3 is a potent LIMK inhibitor with IC50s of 5 nM and 6 nM for LIMK1 and LIMK2, respectively.
|
T15798 |
LX7101
|
1192189-69-7
|
98%
|
|
LX7101 is an effective inhibitor of LIMK and ROCK2 (IC50: 24, 1.6, and 10 nM for LIMK1, LIMK2, and ROCK2, respectively). It also inhibits PKA (IC50 <1 nM).
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