Apalutamide-COOH is a metabolite derived from Apalutamide, which acts as a highly potent and competitive antagonist of the androgen receptor (AR). It effectively binds to the AR with an IC50 value of 16 nM.

Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.

Apalutamide-d4 is a deuterated compound of Apalutamide.

Apalutamide-d7 is a deuterated compound of Apalutamide. Apalutamide has a CAS number of 956104-40-8. Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.

N-desmethyl Apalutamide-d4 is a deuterated compound of N-desmethyl Apalutamide. N-desmethyl Apalutamide has a CAS number of 1332391-11-3. N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.

Apalutamide-13C-d3 is the 13C and deuterated compound of Apalutamide. Apalutamide has a CAS number of 956104-40-8. Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.

N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.