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  • HIV Protease
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gsk-1349572

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  • Inhibitors & Agonists
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Dolutegravir
S GSK1349572,GSK1349572
T61981051375-16-6
Dolutegravir (GSK1349572) (IC50=2.7 nM), a two-metal-binding HIV integrase inhibitor, exhibits medium activity against raltegravir-resistant signature mutants Y143R, Q148K, N155H, and G140S Q148H.
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Dolutegravir sodium
GSK1349572,GSK-1349572A
T23291051375-19-9
Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature mutants Y143R, Q148K, N155H, and G140S Q148H.
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