rp camps triethylammonium salt

Rp-cAMPS triethylammonium salt is an analog of cAMP.It acts as a potent, competitive and cell-permeable antagonist of cAMP-induced activation of cAMP-dependent PKA I and II with Kis of 6.05 µM and 9.75 µM, respectively.

BzATP triethylammonium salt is a P2X7 receptor agonist.

Rp-cAMPS competitively inhibits the cAMP-induced activation of cAMP-dependent protein kinase (PKA).

Rp-8-CPT-cAMP is a structural combination of the lipophilic and non-hydrolyzable cAMP analogs, 8-CPT-cyclic AMP and Rp-cyclic AMPS .[1] It functions as a site-selective inhibitor of protein kinase A (PKA) type I and II, with preference towards site A of type I and site B of type II.2 By occupying cAMP binding sites at the regulatory subunit of PKA, Rp-8-CPT-cAMP prevents the kinase holoenzyme from dissociative activation.[2],[3]

P2X receptor antagonist

Rp-8-bromo-Cyclic AMPS (Rp-8-bromo-cAMPS) is a cell-permeable cAMP analog that combines an exocyclic sulfur substitution in the equatorial position of the cyclophosphate ring with a bromine substitution in the adenine base of cAMP. It acts as an antagonist of cAMP-dependent protein kinases (PKAs) and is resistant to hydrolysis by cyclic nucleotide phosphodiesterases. Rp-8-bromo-cAMPS more effectively antagonizes cAMP-dependent activation of purified PKA type I from rabbit muscle than PKA type II from bovine heart.

Adenosine 5’-monophosphate triethylammonium salt is a useful organic compound for research related to life sciences and the catalog number is TNU1647.

2'-O-Methyl-5-methyluridine 5'-triphosphate triethylammonium salt is a Nucleoside Triphosphate.

2’-O-Methyl-N6-methyladenosine 5’-monophosphate triethylammonium salt (60091-05-6 neutral molecule) is a useful organic compound for research related to life sciences and the catalog number is TNU1630.

Rp-8-CPT-cAMPS is a powerful and competitive antagonist of cAMP-induced activation of cAMP-dependent protein kinase (PKA) I and II. Acting as a potent cAMP analog, Rp-8-CPT-cAMPS exhibits a preference for site A of RI over site A of RII. Additionally, it favors site B of RII over site B of RI. This compound effectively inhibits cAMP-dependent PKA activation and demonstrates selectivity in binding to specific sites within the protein kinase.

MRS 2957 triethylammonium salt is a P2Y6 agonist.

MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).

N6-Methyladenosine 5’-monophos phate triethylammonium salt (neutral 4229-50-9) is a useful organic compound for research related to life sciences and the catalog number is TNU1631.

Rp-cAMPS sodium salt, a cAMP analog, is a potent and competitive antagonist of cAMP-induced activation of cAMP-dependent PKA I and II (Kis of 12.5 μM and 4.5 μM, respectively). It is resistant to hydrolysis by phosphodiesterases[1][2][3][4][5][6].

(Methoxycarbonylsulfamoyl)triethylammonium hydroxide, inner salt is a useful organic compound for research related to life sciences. The catalog number is T65053 and the CAS number is 29684-56-8.