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Apelin receptor

The apelin receptor (also known as the APJ receptor) is a G protein-coupled receptor which binds apelin and Apela/ELABELA/Toddler.
Cat No. product name
T35374L (Ala13)-Apelin-13 acetate (Ala13)-Apelin-13 acetate,一种APJ拮抗剂,可调节CRF诱导的增强的结肠运动、内脏敏感性和肠屏障。
TP1922L1 ELA-11 (human) acetate(1784687-32-6 free base) ELA-11 (human) acetate high affinity apelin receptor agonist (Ki = 14 nM). Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulate...
TP1923L1 ELA-14(human) acetate ELA-14(human) acetate is a fragment of ELA that binds to APJ, activates the Gαi1 and β-arrestin-2 signaling pathways, and induces receptor internalization simila...
TP1260 [Pyr1]-Apelin-13 [Pyr1]-Apelin-13 is a potent and selective endogenous Apelin receptor (APJ) agonist.
T4390 ML221 ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the...
(Ala13)-Apelin-13 acetate
T35374L
(Ala13)-Apelin-13 acetate,一种APJ拮抗剂,可调节CRF诱导的增强的结肠运动、内脏敏感性和肠屏障。
ELA-11 (human) acetate(1784687-32-6 free base)
TP1922L1
ELA-11 (human) acetate high affinity apelin receptor agonist (Ki = 14 nM). Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulate...
ELA-14(human) acetate
TP1923L1
ELA-14(human) acetate is a fragment of ELA that binds to APJ, activates the Gαi1 and β-arrestin-2 signaling pathways, and induces receptor internalization simi...
[Pyr1]-Apelin-13
TP1260
[Pyr1]-Apelin-13 is a potent and selective endogenous Apelin receptor (APJ) agonist.
ML221
T4390
ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in t...