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GNRH Receptor

The gonadotropin-releasing hormone receptor (GnRHR), also known as the luteinizing hormone releasing hormone receptor (LHRHR), is a member of the seven-transmembrane, G-protein coupled receptor (GPCR) family. It is the receptor of gonadotropin-releasing hormone (GnRH). The GnRHR is expressed on the surface of pituitary gonadotrope cells as well as lymphocytes, breast, ovary, and prostate.
Cat. No. Product name CAS No. Purity Chemical Structure
T10988 Degarelix 214766-78-6 98%
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
T21309 Nafarelin acetate(76932-56-4 free base) 76932-60-0 98%
Nafarelin acetate is a GnRH agonist that acts as an analog of GnRH. Nafarelin causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (...
T5031 Elagolix sodium 832720-36-2 98%
Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
TP2107L Histrelin acetate 220810-26-4 98%
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called ...
T21410 Triptorelin acetate(57773-63-4 free base) 140194-24-7 98%
Triptorelin Acetate is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) ...
TP2323L Deslorelin acetate(57773-65-6 free base) TP2323L 98%
Deslorelin acetate is a gonadotropin releasing hormone super-agonist (GnRH agonist)
T27837 Linzagolix 935283-04-8 98%
Linzagolix is an antagonist of gonadotrophin releasing hormone (GnRH) .
T3630 Relugolix 737789-87-6 98%
Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential an...
TP1700L LGnRH-III, lamprey acetate(147859-97-0 free base) TP1700L 98%
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion of...
TP1307 Buserelin Acetate (57982-77-1 free base) 68630-75-1 98%
Buserelin Acetate is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
T10988L Degarelix acetate(214766-78-6 free base) T10988L 98%
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
TP1434L Lecirelin acetate(61012-19-9 free base) TP1434L 98%
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts....
T5520 Cetrorelix Acetate 145672-81-7 98%
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
TP2337 Ganirelix Acetate 123246-29-7 98%
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
T4102 Goserelin acetate 145781-92-6 98%
Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
T10217L Abarelix 183552-38-7 98%
Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
T1494 Alarelin Acetate 79561-22-1 98%
Alarelin acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
T22025 AG 045572 263847-55-8 98%
AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is ...
T11174 (R)-Elagolix 834153-87-6 98%
(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable dep...
T5520L Cetrorelix diacetate 130143-01-0 98%
Cetrorelix diacetate is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the ...
Degarelix
T10988
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
Nafarelin acetate(76932-56-4 free base)
T21309
Nafarelin acetate is a GnRH agonist that acts as an analog of GnRH. Nafarelin causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (...
Elagolix sodium
T5031
Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
Histrelin acetate
TP2107L
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called ...
Triptorelin acetate(57773-63-4 free base)
T21410
Triptorelin Acetate is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) ...
Deslorelin acetate(57773-65-6 free base)
TP2323L
Deslorelin acetate is a gonadotropin releasing hormone super-agonist (GnRH agonist)
Linzagolix
T27837
Linzagolix is an antagonist of gonadotrophin releasing hormone (GnRH) .
Relugolix
T3630
Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential an...
LGnRH-III, lamprey acetate(147859-97-0 free base)
TP1700L
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion of...
Buserelin Acetate (57982-77-1 free base)
TP1307
Buserelin Acetate is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
Degarelix acetate(214766-78-6 free base)
T10988L
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
Lecirelin acetate(61012-19-9 free base)
TP1434L
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts....
Cetrorelix Acetate
T5520
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
Ganirelix Acetate
TP2337
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
Goserelin acetate
T4102
Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
Abarelix
T10217L
Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
Alarelin Acetate
T1494
Alarelin acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
AG 045572
T22025
AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is ...
(R)-Elagolix
T11174
(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable dep...
Cetrorelix diacetate
T5520L
Cetrorelix diacetate is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the ...