GNRH Receptor

The gonadotropin-releasing hormone receptor (GnRHR), also known as the luteinizing hormone releasing hormone receptor (LHRHR), is a member of the seven-transmembrane, G-protein coupled receptor (GPCR) family. It is the receptor of gonadotropin-releasing hormone (GnRH). The GnRHR is expressed on the surface of pituitary gonadotrope cells as well as lymphocytes, breast, ovary, and prostate.

Cat. No.	Product name	CAS No.	Purity
T27837	Linzagolix	935283-04-8	98%
T27837	Linzagolix is an antagonist of gonadotrophin releasing hormone (GnRH) .
T10988	Degarelix	214766-78-6	98%
T10988	Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
T10217L	Abarelix	183552-38-7	100%
T10217L	Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
T1494	Alarelin Acetate	79561-22-1	100%
T1494	Alarelin acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
T4102	Goserelin acetate	145781-92-6	100%
T4102	Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
TP2337	Ganirelix Acetate	123246-29-7	96.05%
TP2337	Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
T11174	(R)-Elagolix	834153-87-6	97.63%
T11174	(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable dep...
T5520	Cetrorelix Acetate	145672-81-7	97.96%
T5520	Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
TP1434L	Lecirelin acetate(61012-19-9 free base)	TP1434L	98.1%
TP1434L	Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts....
T5520L	Cetrorelix diacetate	130143-01-0	98.38%
T5520L	Cetrorelix diacetate is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the ...
T10988L	Degarelix acetate(214766-78-6 free base)	T10988L	98.66%
T10988L	Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
T3630	Relugolix	737789-87-6	98.85%
T3630	Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential an...
TP1700L	LGnRH-III, lamprey acetate(147859-97-0 free base)	TP1700L	99.66%
TP1700L	LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion of...
TP1307	Buserelin Acetate (57982-77-1 free base)	68630-75-1	99.78%
TP1307	Buserelin Acetate is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
TP2323L	Deslorelin acetate(57773-65-6 free base)	TP2323L	99.84%
TP2323L	Deslorelin acetate is a gonadotropin releasing hormone super-agonist (GnRH agonist)
T5031	Elagolix sodium	832720-36-2	99.93%
T5031	Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
T21410	Triptorelin acetate(57773-63-4 free base)	140194-24-7	99.93%
T21410	Triptorelin Acetate is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) ...
T21309	Nafarelin acetate(76932-56-4 free base)	76932-60-0	99.98%
T21309	Nafarelin acetate is a GnRH agonist that acts as an analog of GnRH. Nafarelin causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (...
TP2107L	Histrelin acetate	220810-26-4
TP2107L	Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called ...