benzazepine

SKF83959, a benzazepine analog, is a selective and potent partial agonist of the dopamine D1 receptor with Ki values of 1.18, 7.56, 920, and 399 nM for rat D1, D5, D2, and D3 receptors, respectively.SKF83959 is a potent variant modulator of the sigma (σ)-1 receptor, which ameliorates cognitive dysfunction for the study depression and Alzheimer's disease.

Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4 BETA2 NICOTINIC RECEPTOR partial agonist. It is used for SMOKING CESSATION.

SQ-31765 is a blocker of benzazepine calcium channel.

Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).

Trimopam is a dopamine receptor agonist of the benzazepine group.

Mozavaptan (OPC-31260) is a competitive antagonist of vasopressin receptors, targeting both V1 and V2 receptors, with IC50 values of 1.2 μM and 14 nM, respectively.