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CaSR

The calcium-sensing receptor (CaSR) is a Class C G-protein coupled receptor which senses extracellular levels of calcium ion. It is primarily expressed in the parathyroid gland and the renal tubules of the kidney.
Cat. No. Product name CAS No. Purity Chemical Structure
T34385 Ronacaleret HCl 702686-96-2 98%
Ronacaleret HCl is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.
T10666 Calhex 231 hydrochloride 2387505-78-2 98%
Calhex 231 hydrochloride is a CaSR inhibitor with the potential for diabetic cardiomyopathy treatment. It blocks Ca2+-induced accumulation of [3H]inositol phosph...
T2406 Cinacalcet hydrochloride 364782-34-3 98%
Cinacalcet hydrochloride is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-sensing receptors to seru...
T15261 Evocalcet 870964-67-3 98%
Evocalcet has an activating effect on the calcium-sensing receptor (CaSR).
T3802 Ligustroflavone 260413-62-5 98%
Ligustroflavone has anti-inflammatory activity.
T13918 Tecalcet Hydrochloride 177172-49-5 98%
Tecalcet Hydrochloride is an allosteric and positive modulator of the calcium-sensing receptor(CaSR). Tecalcet Hydrochloride increases the sensitivity to the act...
T4967 NPS-2143 hydrochloride 324523-20-8 98%
NPS-2143 is a selective potent calcium ion-sensing receptor antagonist.
T29067L Upacicalcet HCl 98%
Upacicalcet HCl is an intravesical calcium mimetic that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on calcium-sensitive receptors ...
T1730 NPS-2143 284035-33-2 98%
NPS-2143 is a novel potent and selective antagonist of Ca(2+) receptor.
TP1236 Etelcalcetide hydrochloride 1334237-71-6 98%
Etelcalcetide hydrochloride is a synthetic peptide as an allosteric modulator of the calcium (Ca)-sensing receptor (CaSR). Etelcalcetide hydrochloride is effecti...
T1641 Strontium ranelate 135459-87-9 98%
Strontium ranelate, a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoarthritis o...
T22795 Gadolinium chloride 10138-52-0 98%
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
T12846 SB-423562 351490-27-2 98%
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
T23401 Strontium chloride 10476-85-4 98%
Strontium chloride is an agonist of Calcium sensing receptor (CaSR) and directly affects C-type nerve fibers.
T8403 Cinacalcet 226256-56-0 98%
Cinacalcet is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .
Ronacaleret HCl
T34385
Ronacaleret HCl is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.
Calhex 231 hydrochloride
T10666
Calhex 231 hydrochloride is a CaSR inhibitor with the potential for diabetic cardiomyopathy treatment. It blocks Ca2+-induced accumulation of [3H]inositol phosph...
Cinacalcet hydrochloride
T2406
Cinacalcet hydrochloride is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-sensing receptors to seru...
Evocalcet
T15261
Evocalcet has an activating effect on the calcium-sensing receptor (CaSR).
Ligustroflavone
T3802
Ligustroflavone has anti-inflammatory activity.
Tecalcet Hydrochloride
T13918
Tecalcet Hydrochloride is an allosteric and positive modulator of the calcium-sensing receptor(CaSR). Tecalcet Hydrochloride increases the sensitivity to the act...
NPS-2143 hydrochloride
T4967
NPS-2143 is a selective potent calcium ion-sensing receptor antagonist.
Upacicalcet HCl
T29067L
Upacicalcet HCl is an intravesical calcium mimetic that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on calcium-sensitive receptors ...
NPS-2143
T1730
NPS-2143 is a novel potent and selective antagonist of Ca(2+) receptor.
Etelcalcetide hydrochloride
TP1236
Etelcalcetide hydrochloride is a synthetic peptide as an allosteric modulator of the calcium (Ca)-sensing receptor (CaSR). Etelcalcetide hydrochloride is effecti...
Strontium ranelate
T1641
Strontium ranelate, a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoarthritis o...
Gadolinium chloride
T22795
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
SB-423562
T12846
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
Strontium chloride
T23401
Strontium chloride is an agonist of Calcium sensing receptor (CaSR) and directly affects C-type nerve fibers.
Cinacalcet
T8403
Cinacalcet is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .