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GHSR

Growth hormone secretagogue receptor(GHS-R), also known as ghrelin receptor, is a G protein-coupled receptor that binds growth hormone secretagogues (GHSs), such as ghrelin, the "hunger hormone". The role of GHS-R is thought to be in regulating energy homeostasis and body weight. In the brain, they are most highly expressed in the hypothalamus, specifically the ventromedial nucleus and arcuate nucleus. GSH-Rs are also expressed in other areas of the brain, including the ventral tegmental area, hippocampus, and substantia nigra. Outside the central nervous system, too, GSH-Rs are also found in the liver, in skeletal muscle, and even in the heart.
Cat No. product name
T17103 TM-N1324 TM-N1324 是一种 GPR39 激动剂。 TM-N1324 在没有和存在 Zn2+ 的情况下分别以 280 nM 和 9 nM 的高效率和效力激活人 GPR39。 TM-N1324 对鼠 GPR39 表现出相似的效力,EC50 分别为 180 nM 和 5 nM。
TP2279L Obestatin (rat) acetate Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39). Obestatin (rat) acetate has anti-inflammatory, anti-myocardial infarcti...
T11560 HGPR91 antagonist 1 hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
T16508 PF-5190457 PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
T7325 GHRP-6 acetate GHRP-6 acetate is a synthetic growth hormone (GH) secretagogue and an agonist of the GH secretagogue receptor (GHS-R), which is also known as the ghrelin recepto...
T7225 AnaMorelin hydrochloride Anamorelin hydrochloride is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
T7112 Ibutamoren Mesylate Ibutamoren Mesylate is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
T11719 JMV 2959 hydrochloride (925238-89-7 free base) JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
T10319 Anamorelin Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
TP2328L CJC-1295 acetate(863288-34-0 free base) CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone se...
TQ0022 Capromorelin Tartrate Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).
T4648 TC-G-1008 TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
T5025L Pralmorelin acetate 158861-67-7(free base) Pralmorelin acetate stimulates growth hormone secretion.Pralmorelin acetate is an oral active synthetic peptide analogue of MEK. Pralmorelin acetate, an auxin re...
TM-N1324
T17103
TM-N1324 是一种 GPR39 激动剂。 TM-N1324 在没有和存在 Zn2+ 的情况下分别以 280 nM 和 9 nM 的高效率和效力激活人 GPR39。 TM-N1324 对...
Obestatin (rat) acetate
TP2279L
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39). Obestatin (rat) acetate has anti-inflammatory, anti-myocardial infarcti...
hGPR91 antagonist 1
T11560
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
PF-5190457
T16508
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
GHRP-6 acetate
T7325
GHRP-6 acetate is a synthetic growth hormone (GH) secretagogue and an agonist of the GH secretagogue receptor (GHS-R), which is also known as the ghrelin recepto...
AnaMorelin hydrochloride
T7225
Anamorelin hydrochloride is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
Ibutamoren Mesylate
T7112
Ibutamoren Mesylate is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
JMV 2959 hydrochloride (925238-89-7 free base)
T11719
JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
Anamorelin
T10319
Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
CJC-1295 acetate(863288-34-0 free base)
TP2328L
CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone se...
Capromorelin Tartrate
TQ0022
Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).
TC-G-1008
T4648
TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
Pralmorelin acetate 158861-67-7(free base)
T5025L
Pralmorelin acetate stimulates growth hormone secretion.Pralmorelin acetate is an oral active synthetic peptide analogue of MEK. Pralmorelin acetate, an auxin re...