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GHSR

Growth hormone secretagogue receptor(GHS-R), also known as ghrelin receptor, is a G protein-coupled receptor that binds growth hormone secretagogues (GHSs), such as ghrelin, the "hunger hormone". The role of GHS-R is thought to be in regulating energy homeostasis and body weight. In the brain, they are most highly expressed in the hypothalamus, specifically the ventromedial nucleus and arcuate nucleus. GSH-Rs are also expressed in other areas of the brain, including the ventral tegmental area, hippocampus, and substantia nigra. Outside the central nervous system, too, GSH-Rs are also found in the liver, in skeletal muscle, and even in the heart.
Cat. No. Product name CAS No. Purity Chemical Structure
T17103 TM-N1324 1144477-35-9 98%
TM-N1324 is a GPR39 agonist. TM-N1324 activates human GPR39 with high efficacy and potencies of 280 nM and 9 nM in the absence and presence of Zn2+, respectively...
TP2279L Obestatin (rat) acetate 98%
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39). Obestatin (rat) acetate has anti-inflammatory, anti-myocardial infarcti...
T7225 AnaMorelin hydrochloride 861998-00-7
Anamorelin hydrochloride is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
T12216L NF-56-EJ40 hydrochloride 2728500-80-7 97.02%
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almo...
T7112 Ibutamoren Mesylate 159752-10-0 98%
Ibutamoren Mesylate is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
TP2328L CJC-1295 acetate(863288-34-0 free base) TP2328L 98%
CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone se...
T11719 JMV 2959 hydrochloride (925238-89-7 free base) T11719 98.09%
JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
T5025L Pralmorelin acetate 158861-67-7(free base) T5025L 98.96%
Pralmorelin acetate stimulates growth hormone secretion.Pralmorelin acetate is an oral active synthetic peptide analogue of MEK. Pralmorelin acetate, an auxin re...
TQ0022 Capromorelin Tartrate 193273-69-7 98.98%
Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).
T4648 TC-G-1008 1621175-65-2 99%
TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
TP1155L Human growth hormone-releasing factor acetate 99.26%
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on c...
T10319 Anamorelin 249921-19-5 99.35%
Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
T11560 HGPR91 antagonist 1 1314796-00-3 99.85%
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
T16508 PF-5190457 1334782-79-4 98%
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
TM-N1324
T17103
TM-N1324 is a GPR39 agonist. TM-N1324 activates human GPR39 with high efficacy and potencies of 280 nM and 9 nM in the absence and presence of Zn2+, respectively...
Obestatin (rat) acetate
TP2279L
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39). Obestatin (rat) acetate has anti-inflammatory, anti-myocardial infarcti...
AnaMorelin hydrochloride
T7225
Anamorelin hydrochloride is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
NF-56-EJ40 hydrochloride
T12216L
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almo...
Ibutamoren Mesylate
T7112
Ibutamoren Mesylate is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
CJC-1295 acetate(863288-34-0 free base)
TP2328L
CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone se...
JMV 2959 hydrochloride (925238-89-7 free base)
T11719
JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
Pralmorelin acetate 158861-67-7(free base)
T5025L
Pralmorelin acetate stimulates growth hormone secretion.Pralmorelin acetate is an oral active synthetic peptide analogue of MEK. Pralmorelin acetate, an auxin re...
Capromorelin Tartrate
TQ0022
Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).
TC-G-1008
T4648
TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
Human growth hormone-releasing factor acetate
TP1155L
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on c...
Anamorelin
T10319
Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
hGPR91 antagonist 1
T11560
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
PF-5190457
T16508
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).