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GTPase

GTPases are a large family of hydrolase enzymes that bind to the nucleotide guanosine triphosphate (GTP) and hydrolyze it to guanosine diphosphate (GDP).
Cat No. product name
T5142 NAV-2729 NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.
T2267 BQU57 BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.
T14897 CCG-63802 CCG-63802 is a reversible inhibitor of the regulator of G-protein signaling (RGS) protein and has the greatest potency at RGS4.
T21798L Dynamin inhibitory peptide Acetate Dynamin inhibitory peptide Acetate is a peptide with the sequence Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro that inhibit the GTPase dynamin.
T6634 RBC8 RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.
T14898 CCG-63808 CCG-63808 is a reversible inhibitor of the regulator of G-protein signaling (RGS) proteins.
T24706 RBC10 RBC10 is an inhibitor of the binding of Ral to its effector RALBP1 that acts by inhibiting Ral-mediated cell spreading of murine embryonic fibroblasts and anchor...
T21970 ML-097 ML-097 (CID-2160985) is a pan activator of Ras-related GTPases
T25529 IMM-01 IMM-01 is a novel class of small-molecule agonists of the mammalian Diaphanous (mDia)-related formins, which act downstream of Rho GTPases to assemble actin fila...
T9200 Exo-1 Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate is a chemical compound.
T10705 CCG 203769 CCG 203769 is a selective inhibitor of G protein signaling (RGS4). It blocks the RGS4-Gαo protein-protein interaction in vitro (IC50: 17 nM).
TN4098 Gancaonin I Gancaonin I exhibits anti-BsFtsZ GTPase activities; it also shows significant inhibitory activity against B. subtilis, with a MIC value of 5 uM.
T6434 CCG-50014 CCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.
T4022 QS11 QS 11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor. Modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling p...
NAV-2729
T5142
NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.
BQU57
T2267
BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.
CCG-63802
T14897
CCG-63802 is a reversible inhibitor of the regulator of G-protein signaling (RGS) protein and has the greatest potency at RGS4.
Dynamin inhibitory peptide Acetate
T21798L
Dynamin inhibitory peptide Acetate is a peptide with the sequence Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro that inhibit the GTPase dynamin.
RBC8
T6634
RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.
CCG-63808
T14898
CCG-63808 is a reversible inhibitor of the regulator of G-protein signaling (RGS) proteins.
RBC10
T24706
RBC10 is an inhibitor of the binding of Ral to its effector RALBP1 that acts by inhibiting Ral-mediated cell spreading of murine embryonic fibroblasts and anchor...
ML-097
T21970
ML-097 (CID-2160985) is a pan activator of Ras-related GTPases
IMM-01
T25529
IMM-01 is a novel class of small-molecule agonists of the mammalian Diaphanous (mDia)-related formins, which act downstream of Rho GTPases to assemble actin fila...
Exo-1
T9200
Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate is a chemical compound.
CCG 203769
T10705
CCG 203769 is a selective inhibitor of G protein signaling (RGS4). It blocks the RGS4-Gαo protein-protein interaction in vitro (IC50: 17 nM).
Gancaonin I
TN4098
Gancaonin I exhibits anti-BsFtsZ GTPase activities; it also shows significant inhibitory activity against B. subtilis, with a MIC value of 5 uM.
CCG-50014
T6434
CCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.
QS11
T4022
QS 11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor. Modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling ...