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Neurotensin Receptor

The neurotensin receptors are transmembrane receptors that bind the neurotransmitter neurotensin. Two of the receptors encoded by the NTSR1 and NTSR2 genes contain seven transmembrane helices and are G protein coupled. The third receptor has a single transmembrane domain and is encoded by the SORT1 gene.
Cat. No. Product name CAS No. Purity Chemical Structure
T7617 Neurotensin(8-13) 60482-95-3 98%
Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
TQ0075 ML314 1448895-09-7 98%
ML314 is an effective molecule agonist of NTR1 (EC50: 1.9 μM).
TP1819L Substance P 1-9 aceate 98%
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.
T38807L [Lys8, Lys9]-Neurotensin (8-13) acetate 98%
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, ...
T22476 (±)-AC 7954 hydrochloride 477313-09-0 98%
(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.
TP1310 Neurotensin 39379-15-2 98%
Neurotensin is a 13 amino acid neuropeptide that is implicated in the regulation of luteinizing hormone and prolactin release and has significant interaction wit...
TP1116L Kinetensin acetate(103131-69-7 free base) TP1116L 98%
Kinetensin acetate is isolated from pepsin-treated human plasma.Kinetensin acetate is a neurotensin-like peptide.
T7617L Neurotensin(8-13) 3TFA(60482-95-3(free base)) 2952825-79-3 98%
Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
T28217 NTRC-844 1811503-67-9 98%
NTRC-844 is a selective rat neurotensin receptor type 2 (NTS2) antagonist that shows analgesic activity in animal models of pain.
T12848 SB-657510 474960-44-6 98%
SB-657510 is a urotensin II (UII) receptor (UT) antagonist. The Ki values of UT for human, monkey, cat, rat and mouse were 61, 17, 30, 65 and 56 nM, respectively...
TP2106L Urantide acetate(669089-53-6 free base) TP2106L 98%
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. E...
T23323 SB 611812 345892-71-9 98%
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.
TQ0086 AF38469 1531634-31-7 98%
AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
T9044 SORT-PGRN interaction inhibitor 1 100957-85-5 98%
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
T16860 SBI-553 1849603-72-0 98%
SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
TP2104L UFP 803 acetate 98%
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.
T23386 SR 142948 184162-64-9 98%
SR 142948 is a neurotensin (NT) receptor antagonist.
Neurotensin(8-13)
T7617
Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
ML314
TQ0075
ML314 is an effective molecule agonist of NTR1 (EC50: 1.9 μM).
Substance P 1-9 aceate
TP1819L
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.
[Lys8, Lys9]-Neurotensin (8-13) acetate
T38807L
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, ...
(±)-AC 7954 hydrochloride
T22476
(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.
Neurotensin
TP1310
Neurotensin is a 13 amino acid neuropeptide that is implicated in the regulation of luteinizing hormone and prolactin release and has significant interaction wit...
Kinetensin acetate(103131-69-7 free base)
TP1116L
Kinetensin acetate is isolated from pepsin-treated human plasma.Kinetensin acetate is a neurotensin-like peptide.
Neurotensin(8-13) 3TFA(60482-95-3(free base))
T7617L
Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
NTRC-844
T28217
NTRC-844 is a selective rat neurotensin receptor type 2 (NTS2) antagonist that shows analgesic activity in animal models of pain.
SB-657510
T12848
SB-657510 is a urotensin II (UII) receptor (UT) antagonist. The Ki values of UT for human, monkey, cat, rat and mouse were 61, 17, 30, 65 and 56 nM, respectively...
Urantide acetate(669089-53-6 free base)
TP2106L
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. E...
SB 611812
T23323
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.
AF38469
TQ0086
AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
SORT-PGRN interaction inhibitor 1
T9044
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
SBI-553
T16860
SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
UFP 803 acetate
TP2104L
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.
SR 142948
T23386
SR 142948 is a neurotensin (NT) receptor antagonist.