T7617 |
Neurotensin(8-13)
|
60482-95-3
|
98%
|
|
Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
|
TQ0075 |
ML314
|
1448895-09-7
|
98%
|
|
ML314 is an effective molecule agonist of NTR1 (EC50: 1.9 μM).
|
TP1819L |
Substance P 1-9 aceate
|
|
98%
|
|
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.
|
T38807L |
[Lys8, Lys9]-Neurotensin (8-13) acetate
|
|
98%
|
|
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, ...
|
T22476 |
(±)-AC 7954 hydrochloride
|
477313-09-0
|
98%
|
|
(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.
|
TP1310 |
Neurotensin
|
39379-15-2
|
98%
|
|
Neurotensin is a 13 amino acid neuropeptide that is implicated in the regulation of luteinizing hormone and prolactin release and has significant interaction wit...
|
TP1116L |
Kinetensin acetate(103131-69-7 free base)
|
TP1116L
|
98%
|
|
Kinetensin acetate is isolated from pepsin-treated human plasma.Kinetensin acetate is a neurotensin-like peptide.
|
T7617L |
Neurotensin(8-13) 3TFA(60482-95-3(free base))
|
2952825-79-3
|
98%
|
|
Neurotensin(8-13)(3TFA) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
|
T28217 |
NTRC-844
|
1811503-67-9
|
98%
|
|
NTRC-844 is a selective rat neurotensin receptor type 2 (NTS2) antagonist that shows analgesic activity in animal models of pain.
|
T12848 |
SB-657510
|
474960-44-6
|
98%
|
|
SB-657510 is a urotensin II (UII) receptor (UT) antagonist. The Ki values of UT for human, monkey, cat, rat and mouse were 61, 17, 30, 65 and 56 nM, respectively...
|
TP2106L |
Urantide acetate(669089-53-6 free base)
|
TP2106L
|
98%
|
|
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. E...
|
T23323 |
SB 611812
|
345892-71-9
|
98%
|
|
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.
|
TQ0086 |
AF38469
|
1531634-31-7
|
98%
|
|
AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
|
T9044 |
SORT-PGRN interaction inhibitor 1
|
100957-85-5
|
98%
|
|
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
|
T16860 |
SBI-553
|
1849603-72-0
|
98%
|
|
SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
|
TP2104L |
UFP 803 acetate
|
|
98%
|
|
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.
|
T23386 |
SR 142948
|
184162-64-9
|
98%
|
|
SR 142948 is a neurotensin (NT) receptor antagonist.
|