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Thyroid hormone receptor(THR)

The thyroid hormone receptor (TR) is a type of nuclear receptor that is activated by binding thyroid hormone.TRs act as transcription factors, ultimately affecting the regulation of gene transcription and translation. These receptors also have non-genomic effects that lead to second messenger activation, and corresponding cellular response.
Cat No. product name
T9691L (D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate (D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate is a highly potent antagonist of parathyroid hormone (PTH) The Ki value is 69 nM in bovine renal cortical membr...
T7590 Taltirelin Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ conc...
T4461 NSC 90469 3, 5-Diiodo-L-thyronine is an iodinated thyronine hormone that regulates gene activity affecting processes such as homeostasis, lipid metabolism and insulin resi...
T1653 Liothyronine Liothyronine is an active form of thyroid hormone, binding to β1 thyroid hormone receptor (TRβ1), and activates its activity.
T1310 2-Thiouracil Deracil is a thiolated uracil derivative that is a known anti-hyperthyroid agent.
T8672 2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE 2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE is targets the thyroid stimulating hormone receptor (human)
T13492 3,5-Diiodothyropropionic acid 3,5-Diiodothyropropionic acid is a thyroid hormone analog. It induces α-myosin heavy chain mRNA expression, binds to thyroid hormone receptor (Ka: 2.40/M and 4.0...
T0864 L-Thyroxine Levothyroxine is the major hormone derived from the thyroid gland. Thyroxine is synthesized via the iodination of tyrosines (MONOIODOTYROSINE) and the coupling o...
T6956 Protirelin Protirelin is a tripeptide that stimulates the release of thyrotropin and prolactin.
T29011 Triiodothyronine Sulfate Triiodothyronine Sulfate is a prodrug to the Conventional Hormone Therapy of Hypothyroidism. Triiodothyronine sulfate is the main metabolite of thyroid hormone t...
T22355 L-Thyroxine sodium Levothyroxine, the major hormone derived from the thyroid gland, is the agonist of Thyroid hormone receptor alpha and beta.
T23673 AH-3960 AH-3960 is an thyroid hormone receptor-1 (PTHR1) agonist.
T7578 REVERSE T3 reverse T3 inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.
T13072 Taltirelin acetate Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic ...
T1309 Propylthiouracil Propylthiouracil is a thiourea derivative with an antithyroid property. Propylthiouracil (PTU) interferes with the oxidation of iodine possibly by interaction wi...
T10855 CO23 CO23 is a selective agonist of the thyroid hormone receptor (TR) α and can be transported through the blood-brain barrier. CO23 is used for growth and developmen...
T0840 Methimazole Methimazole is a thioureylene antithyroid agent that inhibits the formation of thyroid hormones by interfering with the incorporation of iodine into tyrosyl resi...
T0952 Carbimazole Carbimazole is an imidazole antithyroid agent. It is only found in individuals that have used or taken this drug. Carbimazole is metabolized to methimazole, whic...
TP1022 Protirelin Acetate Protirelin Acetate is a thyrotropin-releasing hormone, stimulating the release of thyrotropin and prolactin from the anterior pituitary.
T6956L Protirelin Acetate(24305-27-9 free base) Protirelin Acetate is a tripeptide that stimulates the release of thyrotropin and prolactin.
T5360 Eprotirome Eprotirome, a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.
T5313 Sobetirome Sobetirome is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).
T3595 Resmetirom MGL-3196 is a highly selective thyroid hormone receptor β (THR-β) agonist.
T1669 Liothyronine sodium Liothyronine Sodium is the sodium salt form of liothyronine, a synthetic form of the levorotatory isomer of the naturally occurring thyroid hormone triiodothyron...
T15699 L-Thyroxine sodium salt pentahydrate L-Thyroxine sodium salt pentahydrate is a synthetic hormone for the research of hypothyroidism. DIO enzymes convert biologically active thyroid hormone (Triiodot...
T15644 KAT681 KAT681 is a liver selective thyromimetic.
T16442 PCO371 PCO371 is an orally active full agonist of parathyroid hormone receptor 1. It has no effect on PTH type 2 receptor.
T1604 Tiratricol Tiratricol is a metabolite of T3 and T4 thyroid hormones; promoted for hyperlipidemia, localized lipodystrophy, and obesity. Tiratricol has been used in trials s...
T40548 NH-3 NH-3是一种可逆甲状腺激素受(THR)体拮抗剂,具有口服活性。
(D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate
T9691L
(D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate is a highly potent antagonist of parathyroid hormone (PTH) The Ki value is 69 nM in bovine renal cortical membr...
Taltirelin
T7590
Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ conc...
NSC 90469
T4461
3, 5-Diiodo-L-thyronine is an iodinated thyronine hormone that regulates gene activity affecting processes such as homeostasis, lipid metabolism and insulin resi...
Liothyronine
T1653
Liothyronine is an active form of thyroid hormone, binding to β1 thyroid hormone receptor (TRβ1), and activates its activity.
2-Thiouracil
T1310
Deracil is a thiolated uracil derivative that is a known anti-hyperthyroid agent.
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE
T8672
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE is targets the thyroid stimulating hormone receptor (human)
3,5-Diiodothyropropionic acid
T13492
3,5-Diiodothyropropionic acid is a thyroid hormone analog. It induces α-myosin heavy chain mRNA expression, binds to thyroid hormone receptor (Ka: 2.40/M and 4....
L-Thyroxine
T0864
Levothyroxine is the major hormone derived from the thyroid gland. Thyroxine is synthesized via the iodination of tyrosines (MONOIODOTYROSINE) and the coupling o...
Protirelin
T6956
Protirelin is a tripeptide that stimulates the release of thyrotropin and prolactin.
Triiodothyronine Sulfate
T29011
Triiodothyronine Sulfate is a prodrug to the Conventional Hormone Therapy of Hypothyroidism. Triiodothyronine sulfate is the main metabolite of thyroid hormone t...
L-Thyroxine sodium
T22355
Levothyroxine, the major hormone derived from the thyroid gland, is the agonist of Thyroid hormone receptor alpha and beta.
AH-3960
T23673
AH-3960 is an thyroid hormone receptor-1 (PTHR1) agonist.
REVERSE T3
T7578
reverse T3 inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.
Taltirelin acetate
T13072
Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic ...
Propylthiouracil
T1309
Propylthiouracil is a thiourea derivative with an antithyroid property. Propylthiouracil (PTU) interferes with the oxidation of iodine possibly by interaction wi...
CO23
T10855
CO23 is a selective agonist of the thyroid hormone receptor (TR) α and can be transported through the blood-brain barrier. CO23 is used for growth and developme...
Methimazole
T0840
Methimazole is a thioureylene antithyroid agent that inhibits the formation of thyroid hormones by interfering with the incorporation of iodine into tyrosyl resi...
Carbimazole
T0952
Carbimazole is an imidazole antithyroid agent. It is only found in individuals that have used or taken this drug. Carbimazole is metabolized to methimazole, whic...
Protirelin Acetate
TP1022
Protirelin Acetate is a thyrotropin-releasing hormone, stimulating the release of thyrotropin and prolactin from the anterior pituitary.
Protirelin Acetate(24305-27-9 free base)
T6956L
Protirelin Acetate is a tripeptide that stimulates the release of thyrotropin and prolactin.
Eprotirome
T5360
Eprotirome, a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.
Sobetirome
T5313
Sobetirome is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).
Resmetirom
T3595
MGL-3196 is a highly selective thyroid hormone receptor β (THR-β) agonist.
Liothyronine sodium
T1669
Liothyronine Sodium is the sodium salt form of liothyronine, a synthetic form of the levorotatory isomer of the naturally occurring thyroid hormone triiodothyron...
L-Thyroxine sodium salt pentahydrate
T15699
L-Thyroxine sodium salt pentahydrate is a synthetic hormone for the research of hypothyroidism. DIO enzymes convert biologically active thyroid hormone (Triiodot...
KAT681
T15644
KAT681 is a liver selective thyromimetic.
PCO371
T16442
PCO371 is an orally active full agonist of parathyroid hormone receptor 1. It has no effect on PTH type 2 receptor.
Tiratricol
T1604
Tiratricol is a metabolite of T3 and T4 thyroid hormones; promoted for hyperlipidemia, localized lipodystrophy, and obesity. Tiratricol has been used in trials s...
NH-3
T40548
NH-3是一种可逆甲状腺激素受(THR)体拮抗剂,具有口服活性。