Vasopressin Receptor

The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into the V1 (V1A), V2, and V3 (V1B) receptor subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.

Cat. No.	Product name	CAS No.	Purity
T80073	Dp[Tyr(methyl)2,Arg8]-Vasopressin	67269-08-3	98%
T80073	Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].
T80136	Val9-Oxytocin	1021701-88-1	98%
T80136	Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.
T80137	(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin	176714-12-8	98%
T80137	(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
T80138	(D-Arg8)-Inotocin	745816-74-4	98%
T80138	'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM. It dem...
T80197	Vasopressin Dimer (parallel) (TFA)		98%
T80197	Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, and O...
T80198	Vasopressin Dimer (anti-parallel) (TFA)		98%
T80198	Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate four G protein-coupled receptors: V1aR, V1bR, V...
T80270	Invopressin	1488411-60-4	98%
T80270	Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial p...
T83501	[Deamino-Pen1,Val4,D-Arg8]-vasopressin	64158-84-5	98%
T83501	[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP). It effectively reduces plasma aldosterone concentration in rats an...
T7434	Argipressin	113-79-1	98%
T7434	Argipressin (Vasopressin) is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, wi...
T4996	Atosiban	90779-69-4	98%
T4996	Atosiban (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt p...
TP2082L	D[Cha4]-AVP acetate(500170-27-4 free base)	TP2082L	99.86%
TP2082L	d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
T5148	Atosiban acetate	914453-95-5	99.84%
T5148	Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) t...
TP1192L	Conopressin S acetate(111317-90-9 free base)	TP1192L	99.79%
TP1192L	Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor...
T13920L	Terlipressin Acetate	1884420-36-3	99.69%
T13920L	Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal e...
T4355	Fuscoside	131631-89-5	99.66%
T4355	Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
T14494	Balovaptan	1228088-30-9	99.34%
T14494	Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mous...
T7303	LIXIVAPTAN	168079-32-1	99.33%
T7303	Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
T15273	Fedovapagon	347887-36-9	99.33%
T15273	Fedovapagon (VA106483) is a selective and potent agonist of the vasopressin V2 receptor (V2R) that inhibits the growth of intersegmental vessels in zebrafish. Fe...
T6288	Mozavaptan	137975-06-5	99.26%
T6288	Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
TP1927L1	D[Leu4,Lys8]-VP acetate	TP1927L1	98.86%
TP1927L1	d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respe...