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Vasopressin Receptor

The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into the V1 (V1A), V2, and V3 (V1B) receptor subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.
Cat No. product name
T2568L Felypressin acetate Felypressin acetate 是加压素 1 的激动剂,作用于所有精氨酸加压素受体 1AS。 Felypressin acetate 可用于牙科手术。
T2326 Tolvaptan Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
T4996 Atosiban Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
T5148 Atosiban acetate (90779-69-4 free base) Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
T7434 Argipressin Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values o...
T2568 Felypressin Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
T7303 LIXIVAPTAN Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
TP1192L Conopressin S acetate(111317-90-9 free base) Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
TP2082L D[Cha4]-AVP acetate(500170-27-4 free base) d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
T6453 Conivaptan hydrochloride Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
T6288 Mozavaptan Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T5144 Desmopressin acetate (16679-58-6 free base) Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
T4355 Fuscoside OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
T4141 RG7713 RO5028442 has been used in trials studying Autistic Disorder.
T14494 Balovaptan Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
T13920L Terlipressin Acetate Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
Felypressin acetate
T2568L
Felypressin acetate 是加压素 1 的激动剂,作用于所有精氨酸加压素受体 1AS。 Felypressin acetate 可用于牙科手术。
Tolvaptan
T2326
Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
Atosiban
T4996
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
Atosiban acetate (90779-69-4 free base)
T5148
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
Argipressin
T7434
Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values o...
Felypressin
T2568
Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
LIXIVAPTAN
T7303
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
Conopressin S acetate(111317-90-9 free base)
TP1192L
Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
d[Cha4]-AVP acetate(500170-27-4 free base)
TP2082L
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
Conivaptan hydrochloride
T6453
Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
Mozavaptan
T6288
Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
Desmopressin acetate (16679-58-6 free base)
T5144
Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
Fuscoside
T4355
OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
RG7713
T4141
RO5028442 has been used in trials studying Autistic Disorder.
Balovaptan
T14494
Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
Terlipressin Acetate
T13920L
Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...