TWS0787 |
Oroxin A
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Oroxin A is a partial PPARγ agonist that can activate PPARγ transcriptional activation in vitro and in vivo. Oroxin A also exhibited inhibitory activity against ...
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T10755L |
Celgosivir
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Celgosivir is an inhibitor of α-glucosidase I. In vitro assay, it inhibits bovine viral diarrhoea virus (BVDV) ( IC50: 1.27 μM ).
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T41044 |
Naringinase
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Naringinase, a hydrolytic enzymatic complex, possesses the activity of both α-L-rhamnosidase and β-D-glucosidase. Naringinase has wide occurrence in nature. Nari...
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TQ0308 |
Castanospermine
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Castanospermine is a natural compound that inhibits α- and β-glucosidases, especially glucosidase l.
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T21344 |
1-Deoxynojirimycin hydrochloride
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Duvoglustat is a potent and selective inhibitor of alpha-glucosidase, most commonly found in mulberry leaves. Duvoglustat is used to suppress the elevation of po...
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T8260 |
4',5-Dihydroxyflavone
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4',5-Dihydroxyflavone is a soybean LOX-1(Ki: 102.6 μM) and yeast α-Glucosidase inhibitor (IC50: 66 μM).
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T6S0535 |
Pinoresinol diglucoside
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1. Pinoresinol diglucoside is a putative α-glucosidase inhibiting compound. 2. Pinoresinol diglucoside is a important antihypertensive compound.
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T13130 |
Terphenyllin
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Terphenyllin has α-glucosidase inhibitory activity, and is a natural product isolated from the coral derived fungus Aspergillus candidus.
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T8319 |
Butyl isobutyl phthalate
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Butyl isobutyl phthalate is a non-competitive α-glucosidase inhibitor(IC50 :38 μM),it shows a hypoglycemic effect
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T3S1612 |
Kuwanon G
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1. Kuwanon G as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective treatment for ...
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T12142 |
N-Caffeoyl O-methyltyramine
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N-Caffeoyl O-methyltyramine is isolated from Cuscuta reflexa with strong inhibitory activity against α-glucosidase with IC50 of 103.58 μM.
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TN6784 |
Ethyl rosmarinate
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Methyl rosmarinate inhibit the activity of tyrosinase, α-glucosidase, and matrix metalloproteinase-1 (MMP-1).
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T5690 |
7,4'-Di-O-methylapigenin
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4',7-DIMETHOXY-5-HYDROXYFLAVONE can inhibit α-glucosidase and α-amylase enzymes and enhance 2-NBDG uptake in L6 cells, it has hypolipidemic effect on mouse pre-a...
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TN1451 |
Brevifolincarboxylic acid
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Brevifolincarboxylic acid is a natural product isolated from Polygonum capitatum, it has inhibitory effect on the aryl hydrocarbon receptor (AhR). Brevifolincarb...
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T4280 |
Gcase activator 1
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LTI-291 is a glucocerebrosidase (Gcase) activator.
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T7858 |
Ceftezole sodium
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Ceftezole sodium is a broad-spectrum cephalosporin antibiotic active gram-negative and gram-positive bacteria except for Proteus vulgaris, Pseudomonas aeruginosa...
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T3S2072 |
3-Butylidenephthalide
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1. (Z)-3-butylidenephthalide has antihyperglycemic effect is due to inhibition of α-glucosidase at the intestinal level, inhibited the activity of yeast-α-glucos...
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T6S2122 |
Ginkgolic Acid (C13:0)
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1.Ginkgolic acid C13: 0exhibits the highest α-glucosidase inhibitory activity.
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T3871 |
Daucosterol
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Eleutheroside A (Daucosterol) has proliferation-enhancing activity, may be involved in the IGF1-AKT pathway. Daucosterol has efficient and inexpensive neuroprote...
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T8202 |
Kaempferol 3-O-gentiobioside
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Kaempferol 3-O-gentiobioside is a flavonoid isolated from C. alata leaves with antidiabetic activity. It possesses activity against α-glucosidase and displays a ...
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T6S1371 |
Isovitexin
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1. Isovitexin exhibits a potential antioxidant activity. 2. Isovitexin shows a strong antihyperglycemic action, inhibits α-glucosidase in vivo.
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T6723 |
Voglibose
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Voglibose, an N-substituted derivative of valiolamine, exhibits excellent inhibitory activity against α-glucosidases and action against hyperglycemia and various...
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TQ0300 |
Conduritol B epoxide
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Conduritol B epoxide is an irreversible inhibitor of β-glucosidase (GCase).
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T3675 |
1-Deoxynojirimycin
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1-Deoxynojirimycin is a potent α-glucosidase inhibitor, suppressing postprandial blood glucose, thereby possibly preventing diabetes mellitus.
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T0247 |
Acarbose
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Acarbose is an inhibitor of α-Glucosidases with antihyperglycemic activity.
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T5489 |
Tryptophan, N-indol-3-ylacetyl- (6CI)
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Indole-3-acetyl-L-tryptophan is involved in regulatory mechanisms for the control of auxin activity during physiological and pathophysiological responses. It may...
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T7028 |
Licochalcone C
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Licochalcone C has potent antioxidant properties and inhibition of bacterial growth and cellular respiration. It has cardioprotection effect, via antioxidant, an...
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T3235 |
Rebaudioside A
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Rebaudioside A is a novel agent of glycoside clathration of pharmacons, acts as α-glucosidase inhibitor.
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TN2130 |
Manghaslin
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Manghaslin has considerable α-glucosidase inhibitory activity, illustrating the anti-diabetic potential of phenolic-rich litchi pulp extracts. Manghaslin also sh...
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TL0008 |
Gigantol
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Gigantol is a novel inhibitor of the Wnt/β-catenin pathway. It inhibits Wnt/β-catenin signaling through downregulation of phosphorylated LRP6 and cytosolic β-cat...
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