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Melanocortin Receptor

Melanocortin receptors are members of the rhodopsin family of 7-transmembrane G protein-coupled receptors. There are five known members of the melanocortin receptor system:MC1R,MC2R,MC3R,MC4R,MC5R.
Cat. No. Product name CAS No. Purity Chemical Structure
T12882 Setmelanotide 920014-72-8 98%
Setmelanotide is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
TP1011L ACTH (1-17) acetate 98%
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
T7627 Adrenocorticotropic Hormone (ACTH) (4-10), human 4037-01-8 98%
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
T16879L SHU 9119 acetate T16879L 98%
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...
TP1004L Beta-MSH (1-22) (human) acetate 98%
β-Melanocyte Stimulating Hormone (MSH), human, a 22-peptide, is an endogenous melanocortin-4 receptor (MC4-R) agonist.
TP1889 MCL0020 475498-26-1 98%
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
T5464 JNJ-10229570 524923-88-4 98%
JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
T7627L Adrenocorticotropic Hormone (ACTH) (4-10) TFA T7627L 98%
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
T8485 THIQ 312637-48-2 98%
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
T9596 AP1189 acetate 959850-74-9 98%
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
TP2212L A-MSH, amide Acetate(581-05-5 free base) TP2212L 98%
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
TP1101 Nonapeptide-1 acetate salt (158563-45-2 free base) TP1101 98%
Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt...
TP1952L PG 106 acetate 98%
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with t...
T7589 Afamelanotide acetate 1566590-77-9 98%
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
T7608 Bremelanotide Acetate 1607799-13-2 98%
Bremelanotide is an agonist of melanocortin receptor (MCR) .
T25310 Dersimelagon 1835256-48-8 98%
Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cyn...
TP1578L Neuropeptide EI, rat acetate TP1578L 98%
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
T12882L Setmelanotide Acetate(920014-72-8 free base) 2759937-80-7 98%
Setmelanotide Acetate is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
TP1248L ACTH 11-24 acetate(4237-93-8 free base) 79190-56-0 98%
ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
TP1893L1 [D-Trp8]-γ-MSH acetate(321351-81-9 free base) TP1893L1 98%
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
Setmelanotide
T12882
Setmelanotide is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
ACTH (1-17) acetate
TP1011L
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
Adrenocorticotropic Hormone (ACTH) (4-10), human
T7627
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
SHU 9119 acetate
T16879L
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...
Beta-MSH (1-22) (human) acetate
TP1004L
β-Melanocyte Stimulating Hormone (MSH), human, a 22-peptide, is an endogenous melanocortin-4 receptor (MC4-R) agonist.
MCL0020
TP1889
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
JNJ-10229570
T5464
JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
T7627L
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
THIQ
T8485
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
AP1189 acetate
T9596
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
a-MSH, amide Acetate(581-05-5 free base)
TP2212L
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
Nonapeptide-1 acetate salt (158563-45-2 free base)
TP1101
Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt...
PG 106 acetate
TP1952L
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with t...
Afamelanotide acetate
T7589
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
Bremelanotide Acetate
T7608
Bremelanotide is an agonist of melanocortin receptor (MCR) .
Dersimelagon
T25310
Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cyn...
Neuropeptide EI, rat acetate
TP1578L
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
Setmelanotide Acetate(920014-72-8 free base)
T12882L
Setmelanotide Acetate is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
ACTH 11-24 acetate(4237-93-8 free base)
TP1248L
ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
TP1893L1
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
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