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Melanocortin Receptor

Melanocortin receptors are members of the rhodopsin family of 7-transmembrane G protein-coupled receptors. There are five known members of the melanocortin receptor system:MC1R,MC2R,MC3R,MC4R,MC5R.
Cat No. product name
TP1952L PG 106 acetate PG 106 acetate 是一种有效的特异性人黑皮质素 3 (hMC3) 受体拮抗剂,IC50 为 210 nM。 PG 106 acetate 对 hMC5 受体和 hMC4 受体没有活性,hMC4 受体的EC50 为 9900 nM。
TP1004L Beta-MSH (1-22) (human) acetate β-Melanocyte Stimulating Hormone (MSH), human, a 22-peptide, is an endogenous melanocortin-4 receptor (MC4-R) agonist.
T7589 Afamelanotide acetate Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
T7627 Adrenocorticotropic Hormone (ACTH) (4-10), human Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
T7627L Adrenocorticotropic Hormone (ACTH) (4-10) TFA Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
TP1011L ACTH (1-17) acetate ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
T20501 Undecylenoyl phenylalanine Undecylenoyl phenylalanine is a novel, skin-lightening agent. It acting as α-melanocyte-stimulating hormone and beta-adrenergic receptor antagonist.
T9596 AP1189 acetate AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
T7813 α-MSH α-MSH is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
T8485 THIQ THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
T7608 Bremelanotide Acetate Bremelanotide is an agonist of melanocortin receptor (MCR) .
TP2212L A-MSH, amide Acetate(581-05-5 free base) a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
TP1101 Nonapeptide-1 acetate salt (158563-45-2 free base) Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt...
TP1578L Neuropeptide EI, rat acetate Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
TP1893L1 [D-Trp8]-γ-MSH acetate(321351-81-9 free base) Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
TP1889 MCL0020 Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
TP1898 HS024 Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). In...
TP2015L HS 014 acetate(207678-81-7 free base) HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 re...
TP1324 Melanotan (MT)-II Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
TP1248L ACTH 11-24 acetate(4237-93-8 free base) ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
T5464 JNJ-10229570 JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
T16879L SHU 9119 acetate SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...
PG 106 acetate
TP1952L
PG 106 acetate 是一种有效的特异性人黑皮质素 3 (hMC3) 受体拮抗剂,IC50 为 210 nM。 PG 106 acetate 对 hMC5 受体和 hMC4 受体没有活性...
Beta-MSH (1-22) (human) acetate
TP1004L
β-Melanocyte Stimulating Hormone (MSH), human, a 22-peptide, is an endogenous melanocortin-4 receptor (MC4-R) agonist.
Afamelanotide acetate
T7589
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pr...
Adrenocorticotropic Hormone (ACTH) (4-10), human
T7627
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
T7627L
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
ACTH (1-17) acetate
TP1011L
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
Undecylenoyl phenylalanine
T20501
Undecylenoyl phenylalanine is a novel, skin-lightening agent. It acting as α-melanocyte-stimulating hormone and beta-adrenergic receptor antagonist.
AP1189 acetate
T9596
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
α-MSH
T7813
α-MSH is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
THIQ
T8485
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
Bremelanotide Acetate
T7608
Bremelanotide is an agonist of melanocortin receptor (MCR) .
a-MSH, amide Acetate(581-05-5 free base)
TP2212L
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
Nonapeptide-1 acetate salt (158563-45-2 free base)
TP1101
Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate sa...
Neuropeptide EI, rat acetate
TP1578L
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
TP1893L1
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
MCL0020
TP1889
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
HS024
TP1898
Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). In...
HS 014 acetate(207678-81-7 free base)
TP2015L
HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 re...
Melanotan (MT)-II
TP1324
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
ACTH 11-24 acetate(4237-93-8 free base)
TP1248L
ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
JNJ-10229570
T5464
JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
SHU 9119 acetate
T16879L
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...