T12882 |
Setmelanotide
|
920014-72-8
|
98%
|
|
Setmelanotide is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
|
TP1011L |
ACTH (1-17) acetate
|
|
98%
|
|
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
|
T7627 |
Adrenocorticotropic Hormone (ACTH) (4-10), human
|
4037-01-8
|
98%
|
|
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
|
T16879L |
SHU 9119 acetate
|
T16879L
|
98%
|
|
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...
|
TP1004L |
Beta-MSH (1-22) (human) acetate
|
|
98%
|
|
β-Melanocyte Stimulating Hormone (MSH), human, a 22-peptide, is an endogenous melanocortin-4 receptor (MC4-R) agonist.
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TP1889 |
MCL0020
|
475498-26-1
|
98%
|
|
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
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T5464 |
JNJ-10229570
|
524923-88-4
|
98%
|
|
JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
|
T7627L |
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
|
T7627L
|
98%
|
|
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
|
T8485 |
THIQ
|
312637-48-2
|
98%
|
|
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
|
T9596 |
AP1189 acetate
|
959850-74-9
|
98%
|
|
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
|
TP2212L |
A-MSH, amide Acetate(581-05-5 free base)
|
TP2212L
|
98%
|
|
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
|
TP1101 |
Nonapeptide-1 acetate salt (158563-45-2 free base)
|
TP1101
|
98%
|
|
Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt...
|
TP1952L |
PG 106 acetate
|
|
98%
|
|
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with t...
|
T7589 |
Afamelanotide acetate
|
1566590-77-9
|
98%
|
|
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
|
T7608 |
Bremelanotide Acetate
|
1607799-13-2
|
98%
|
|
Bremelanotide is an agonist of melanocortin receptor (MCR) .
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T25310 |
Dersimelagon
|
1835256-48-8
|
98%
|
|
Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cyn...
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TP1578L |
Neuropeptide EI, rat acetate
|
TP1578L
|
98%
|
|
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
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T12882L |
Setmelanotide Acetate(920014-72-8 free base)
|
2759937-80-7
|
98%
|
|
Setmelanotide Acetate is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
|
TP1248L |
ACTH 11-24 acetate(4237-93-8 free base)
|
79190-56-0
|
98%
|
|
ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
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TP1893L1 |
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
|
TP1893L1
|
98%
|
|
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
|