Home Tools
Log in
Cart

Protease-activated Receptor

Protease-activated receptors (PAR) are a subfamily of related G protein-coupled receptors that are activated by cleavage of part of their extracellular domain. They are highly expressed in platelets, and also on endothelial cells, myocytes and neurons.
Cat. No. Product name CAS No. Purity Chemical Structure
T41190 AY 77 1835734-92-3 98%
AY 77 is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1...
T7380 Protease-Activated Receptor-4 245443-52-1 98%
Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy
T4186 AC-264613 1051487-82-1 98%
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pro...
T7496 Thrombin Receptor Activator for Peptide 5 (TRAP-5) 141685-53-2 98%
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
TP1046 SLIGRL-NH2 171436-38-7 98%
PAR-2 Activating Peptide is an agonist of Protease-Activated Receptor-2 (PAR-2)
T7623L PAR-4 Agonist Peptide, amide acetate T7623L 98%
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
T7573 TFLLR-NH2 197794-83-5 98%
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7013 Vorapaxar 618385-01-6 98%
Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
T8917 PAR-2-IN-1 1690176-75-0 98%
IUN76750 is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
T7740 Protease-Activated Receptor-4 diTFA T7740 98%
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
T2370 AC-55541 916170-19-9 98%
AOB2796 is a novel PAR2 agonist; activated PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assay...
T21699L VKGILS-NH2 Acetate T21699L 98%
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.
T12870 SCH79797 dihydrochloride 1216720-69-2 98%
SCH79797 dihydrochloride is an effective and selective antagonist of protease activated receptor 1 (PAR1) with an IC50 of 70 nM and a Ki of 35 nM. SCH79797 dihyd...
T38852L TRAP-6 amide acetate 98%
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].
TP1046L PAR-2 Activating Peptide acetate TP1046L 98%
PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2).
TQ0012 AZ3451 2100284-59-9 98%
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
T1986 Atopaxar 751475-53-3 98%
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
T38836L Protease-Activated Receptor-1, PAR-1 Agonist acetate 98%
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 ...
T7137 I-191 1690172-25-8 98%
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
T1986L Atopaxar Hydrobromide 474550-69-1 98%
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
AY 77
T41190
AY 77 is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK1/2 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK1...
Protease-Activated Receptor-4
T7380
Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy
AC-264613
T4186
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pro...
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
T7496
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
SLIGRL-NH2
TP1046
PAR-2 Activating Peptide is an agonist of Protease-Activated Receptor-2 (PAR-2)
PAR-4 Agonist Peptide, amide acetate
T7623L
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
TFLLR-NH2
T7573
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
Vorapaxar
T7013
Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
PAR-2-IN-1
T8917
IUN76750 is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
Protease-Activated Receptor-4 diTFA
T7740
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
AC-55541
T2370
AOB2796 is a novel PAR2 agonist; activated PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assay...
VKGILS-NH2 Acetate
T21699L
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.
SCH79797 dihydrochloride
T12870
SCH79797 dihydrochloride is an effective and selective antagonist of protease activated receptor 1 (PAR1) with an IC50 of 70 nM and a Ki of 35 nM. SCH79797 dihyd...
TRAP-6 amide acetate
T38852L
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].
PAR-2 Activating Peptide acetate
TP1046L
PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2).
AZ3451
TQ0012
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
Atopaxar
T1986
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
Protease-Activated Receptor-1, PAR-1 Agonist acetate
T38836L
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 ...
I-191
T7137
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
Atopaxar Hydrobromide
T1986L
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
1 2