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Protease-activated Receptor

Protease-activated receptors (PAR) are a subfamily of related G protein-coupled receptors that are activated by cleavage of part of their extracellular domain. They are highly expressed in platelets, and also on endothelial cells, myocytes and neurons.
Cat No. product name
T21699L VKGILS-NH2 Acetate VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.
T22933L LRGILS-NH2 acetate LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
T2370 AC-55541 AOB2796 is a novel PAR2 agonist; activated PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assay...
TP1046 SLIGRL-NH2 PAR-2 Activating Peptide is an agonist of Protease-Activated Receptor-2 (PAR-2)
T7623L PAR-4 Agonist Peptide, amide acetate PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
T1893 Parmodulin 2 ML 161 is the inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50: 0.26 μM for the inhibition of platelet P-selectin expression ...
T1986L Atopaxar Hydrobromide Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
T1986 Atopaxar Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
T8917 PAR-2-IN-1 IUN76750 is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
T7496 Thrombin Receptor Activator for Peptide 5 (TRAP-5) Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
T7513 Protease-Activated Receptor-2, amide Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)
T7573L TFLLR-NH2 2TFA(197794-83-5(free base)) TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7573 TFLLR-NH2 TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7380 Protease-Activated Receptor-4 Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy
T7137 I-191 I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
T7013 Vorapaxar Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
T7740 Protease-Activated Receptor-4 diTFA Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
T7674 Thrombin Receptor Activator for Peptide Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
T7623 PAR-4 Agonist Peptide, amide PAR-4 Agonist Peptide, amide is an agonist of proteinase-activated receptor-4 (PAR-4).
T7625 TRAP-6 TRAP-6(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
TQ0012 AZ3451 AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
TP1378 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) 2-Furoyl-LIGRLO-amide is a potent and selective protease-activated receptor 2 (PAR2) agonist.
TP1904L FSLLRY-NH2 TFA(245329-02-6 free base) FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR...
TP1925L TcY-NH2 TFA(327177-34-4 free base) tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
TP1046L PAR-2 Activating Peptide acetate PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2).
TP1065 PAR-4 Agonist Peptide, amide TFA PAR-4 Agonist Peptide, amide TFA is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked...
T4186 AC-264613 AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pro...
T3098 Vorapaxar sulfate Vorapaxar sulfate is a potent and orally active thrombin receptor (PAR-1) antagonist.
T12870 SCH79797 dihydrochloride SCH79797 dihydrochloride 是一种有效的特异性蛋白酶激活受体 1 (PAR1) 拮抗剂,IC50 为 70 nM,Ki 为 35 nM。SCH79797 dihydrochloride 具有抗增殖和促凋亡作用。
T27267 ENMD-1068 HCl ENMD-1068 HCl是一种选择性蛋白酶激活受体(PAR-2)拮抗剂,具有抗血管生成和抗炎活性。
VKGILS-NH2 Acetate
T21699L
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.
LRGILS-NH2 acetate
T22933L
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
AC-55541
T2370
AOB2796 is a novel PAR2 agonist; activated PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assay...
SLIGRL-NH2
TP1046
PAR-2 Activating Peptide is an agonist of Protease-Activated Receptor-2 (PAR-2)
PAR-4 Agonist Peptide, amide acetate
T7623L
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
Parmodulin 2
T1893
ML 161 is the inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50: 0.26 μM for the inhibition of platelet P-selectin expression...
Atopaxar Hydrobromide
T1986L
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
Atopaxar
T1986
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
PAR-2-IN-1
T8917
IUN76750 is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
T7496
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
Protease-Activated Receptor-2, amide
T7513
Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)
TFLLR-NH2 2TFA(197794-83-5(free base))
T7573L
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
TFLLR-NH2
T7573
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
Protease-Activated Receptor-4
T7380
Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy
I-191
T7137
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
Vorapaxar
T7013
Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
Protease-Activated Receptor-4 diTFA
T7740
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
Thrombin Receptor Activator for Peptide
T7674
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
PAR-4 Agonist Peptide, amide
T7623
PAR-4 Agonist Peptide, amide is an agonist of proteinase-activated receptor-4 (PAR-4).
TRAP-6
T7625
TRAP-6(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
AZ3451
TQ0012
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
TP1378
2-Furoyl-LIGRLO-amide is a potent and selective protease-activated receptor 2 (PAR2) agonist.
FSLLRY-NH2 TFA(245329-02-6 free base)
TP1904L
FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR...
tcY-NH2 TFA(327177-34-4 free base)
TP1925L
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
PAR-2 Activating Peptide acetate
TP1046L
PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2).
PAR-4 Agonist Peptide, amide TFA
TP1065
PAR-4 Agonist Peptide, amide TFA is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked...
AC-264613
T4186
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pro...
Vorapaxar sulfate
T3098
Vorapaxar sulfate is a potent and orally active thrombin receptor (PAR-1) antagonist.
SCH79797 dihydrochloride
T12870
SCH79797 dihydrochloride 是一种有效的特异性蛋白酶激活受体 1 (PAR1) 拮抗剂,IC50 为 70 nM,Ki 为 35 nM。SCH79797 dihydrochloride 具有抗...
ENMD-1068 HCl
T27267
ENMD-1068 HCl是一种选择性蛋白酶激活受体(PAR-2)拮抗剂,具有抗血管生成和抗炎活性。