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Acyltransferase

Acyltransferase is a type of transferase enzyme that acts upon acyl groups.
Cat. No. Product name CAS No. Purity Chemical Structure
T6937 PF-04620110 1109276-89-2 98%
PF-04620110 is an orally active, selective and potent diglyceride acyltransferase-1 (DGAT1) inhibitor with IC50 of 19 nM.
T12426 PF-06424439 1469284-78-3 98%
PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).
T13373 YM17E 124900-72-7 98%
YM17E is an inhibitor of ACAT with IC50 of 44 nM in rabbit liver microsomes in vitro.
T12767 RP 70676 136609-26-2 98%
RP 70676 is a potent ACAT inhibitor(rat and rabbit ACAT with IC50 of 25 and 44 nM ).
T23521 VULM 1457 228544-65-8 98%
Acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor
T10035 10,12-Tricosadiynoic acid 66990-30-5
10,12-Tricosadiynoic acid is a highly selective and orally active inhibitor of acyl-CoA oxidase-1 (ACOX1). It can treat the high-fat diet- or obesity-induced met...
T5544 2-Furoic acid 88-14-2 100%
2-Furoic acid, an orally active selective human cathepsin K inhibitor, may have the therapeutic potential for the treatment of diseases characterized by excessiv...
T16409 OSMI-1 1681056-61-0 96.79%
OSMI-1 inhibits protein O-linked N-acetylglucosamine (O-GlcNAcylation) in several mammalian cell lines without qualitatively altering cell surface N- or O-linked...
T6365 A 922500 959122-11-3 97.34%
A922500 is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel o...
T8236 RHC 80267 83654-05-1 98%
RHC 80267 is a selective inhibitor of DAGL (IC50 : 4 µM in canine platelets)
T8314 RP-64477 135239-65-5 99.16%
RP64477 is the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) inhibitor.
T0504 Cyclandelate 456-59-7 99.21%
Cyclandelate, a direct-acting smooth muscle relaxant, is used to dilate blood vessels.
T12225L Nevanimibe hydrochloride 133825-81-7 99.25%
Nevanimibe hydrochloride is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
T3342 Xanthohumol 6754-58-1 99.36%
Xanthohumol, also known as 2', 4, 4'-trihydroxy-6'-methoxy-3'-prenylchalcone or desmethylxanthohumol, is a member of the class of compounds known as 3-prenylated...
T22665 PD 128042 114289-47-3 99.44%
acyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor
TN1691 Glabrol 59870-65-4 99.72%
Glabrol is a PTP1B inhibitor, it is also a CYP1B1 inhibitor, it shows inhibition of CYP1B1 in live cell assay with the IC50 value of 15uM.
T12425 PF-06424439 methanesulfonate 1469284-79-4 99.79%
PF-06424439 methanesulfonate is an oral, potent and selective imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) inhibitor(IC50 of 14 nM)[1]. PF-06424439 m...
T11733 K-604 dihydrochloride 217094-32-1 99.88%
K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.
T4681 T863 701232-20-4 99.88%
T-863(DGAT-1 inhibitor) is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA bi...
T2753 Avasimibe 166518-60-1 99.91%
Avasimibe is an orally bioavailable inhibitor of acyl-Coenzyme A: cholesterol acyltransferase (ACAT, IC50: 3.3 μM) that prevents cholesterol deposition in the ar...
PF-04620110
T6937
PF-04620110 is an orally active, selective and potent diglyceride acyltransferase-1 (DGAT1) inhibitor with IC50 of 19 nM.
PF-06424439
T12426
PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).
YM17E
T13373
YM17E is an inhibitor of ACAT with IC50 of 44 nM in rabbit liver microsomes in vitro.
RP 70676
T12767
RP 70676 is a potent ACAT inhibitor(rat and rabbit ACAT with IC50 of 25 and 44 nM ).
VULM 1457
T23521
Acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor
10,12-Tricosadiynoic acid
T10035
10,12-Tricosadiynoic acid is a highly selective and orally active inhibitor of acyl-CoA oxidase-1 (ACOX1). It can treat the high-fat diet- or obesity-induced met...
2-Furoic acid
T5544
2-Furoic acid, an orally active selective human cathepsin K inhibitor, may have the therapeutic potential for the treatment of diseases characterized by excessiv...
OSMI-1
T16409
OSMI-1 inhibits protein O-linked N-acetylglucosamine (O-GlcNAcylation) in several mammalian cell lines without qualitatively altering cell surface N- or O-linked...
A 922500
T6365
A922500 is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel o...
RHC 80267
T8236
RHC 80267 is a selective inhibitor of DAGL (IC50 : 4 µM in canine platelets)
RP-64477
T8314
RP64477 is the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) inhibitor.
Cyclandelate
T0504
Cyclandelate, a direct-acting smooth muscle relaxant, is used to dilate blood vessels.
Nevanimibe hydrochloride
T12225L
Nevanimibe hydrochloride is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
Xanthohumol
T3342
Xanthohumol, also known as 2', 4, 4'-trihydroxy-6'-methoxy-3'-prenylchalcone or desmethylxanthohumol, is a member of the class of compounds known as 3-prenylated...
PD 128042
T22665
acyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor
Glabrol
TN1691
Glabrol is a PTP1B inhibitor, it is also a CYP1B1 inhibitor, it shows inhibition of CYP1B1 in live cell assay with the IC50 value of 15uM.
PF-06424439 methanesulfonate
T12425
PF-06424439 methanesulfonate is an oral, potent and selective imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) inhibitor(IC50 of 14 nM)[1]. PF-06424439 m...
K-604 dihydrochloride
T11733
K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.
T863
T4681
T-863(DGAT-1 inhibitor) is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA bi...
Avasimibe
T2753
Avasimibe is an orally bioavailable inhibitor of acyl-Coenzyme A: cholesterol acyltransferase (ACAT, IC50: 3.3 μM) that prevents cholesterol deposition in the ar...
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