FAAH

Fatty acid amide hydrolase or FAAH (oleamide hydrolase, anandamide amidohydrolase) is a member of the serine hydrolase family of enzymes. It was first shown to break down anandamide in 1993. In humans, it is encoded by the gene FAAH.FAAH is an integral membrane hydrolase with a single N-terminal transmembrane domain. In vitro, FAAH has esterase and amidase activity.In vivo, FAAH is the principal catabolic enzyme for a class of bioactive lipids called the fatty acid amides (FAAs).

Cat No.	product name
T28353	PDP-EA	PDP-EA 是脂肪酸酰胺水解酶 (FAAH) 的激活剂，可增强 FAAH 的酰胺水解酶活性。
TN1965	N-Benzyllinolenamide	N-Benzyllinolenamide is a natural product. It is an inhibitor of fatty acid amide hydrolase (FAAH, IC50 of 41.8 μM).
T3354	BIA 10-2474	BIA10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH) that increases levels of the neurotransmitter anandamide in the central ner...
T2859	Biochanin A	Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a naturally occurring fatty ...
T3215	JNJ-42165279	JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-42165279...
T4859	1-Monomyristin	1-Myristoyl-rac-glycerol, a 1-monoglyceride of myristic acid, has antibacterial activity against several Gram-positive bacterial strains. 1-Myristoyl-rac-glycero...
T6714	URB-597	URB597 is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets.
T15268	FAAH-IN-2	FAAH-IN-2 is a potent inhibitor of FAAH(fatty acid amide hydrolase).
T6043	PF-3845	PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
T4323	PF-04457845	PF-04457845 is a greatly and effctive FAAH inhibitor, and for hFAAH(IC50=7.2±0.63 nM) and rFAAH(IC50=7.4±0.62 nM).
T2338	JZL195	JZL195 is a selective and efficacious dual FAAH/MAGL inhibitor.
T3S2105	N-Benzylpalmitamide	N-benzylpalmitamide inhibits fatty acid amide hydrolase (FAAH) in a time-dependent manner and could potentially offer a good alternative for the treatment of pai...
T1325	Carprofen	Carprofen is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic activities.
T9374	AA38-3	AA38-3 inhibites three SHs (ABHD6, ABHD11, and FAAH)
T2684	JNJ-1661010	JNJ-1661010 is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.
T8646	URB937	URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM).
T8927	WWL 154	WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor.
T7688	4-Nonylphenylboronic acid	4-Nonylphenylboronic acid is a inhibitor of FAAH.
T12826	SA57	SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).
T11255	FAAH-IN-1	FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.
T12139	N-(3-Methoxybenzyl)Palmitamide	N-(3-Methoxybenzyl)Palmitamide is a promising FAAH inhibitor, treatment of pain, inflammation and CNS degenerative disorders.
T5357	ARN272	ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).
T16847	SA 47	SA 47 is a selective and effective inhibitor of fatty acid amide hydrolase and carbamate.
T16515	PF 750	PF 750 is a selective and covalent fatty acid amide hydrolase inhibitor, It shows IC50s varied from 16.2-595 nM in different pre-incubation times.
T15802	LY2183240	LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 27...