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FAAH

Fatty acid amide hydrolase or FAAH (oleamide hydrolase, anandamide amidohydrolase) is a member of the serine hydrolase family of enzymes. It was first shown to break down anandamide in 1993. In humans, it is encoded by the gene FAAH.FAAH is an integral membrane hydrolase with a single N-terminal transmembrane domain. In vitro, FAAH has esterase and amidase activity.In vivo, FAAH is the principal catabolic enzyme for a class of bioactive lipids called the fatty acid amides (FAAs).
Cat. No. Product name CAS No. Purity Chemical Structure
T11255 FAAH-IN-1 1242441-47-9 98%
FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.
T16847 SA 47 792236-07-8 98%
SA 47 is a selective and effective inhibitor of fatty acid amide hydrolase and carbamate.
T67745 CB2R/FAAH modulator-2 2876918-68-0 98%
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-2 acts as a CB2R agonist and FAAH inhibitor, the Ki value...
T12826 SA57 1346169-63-8 98%
SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).
T63536 Dual FAAH/sEH-IN-1 2756099-59-7 98%
Dual FAAH/sEH-IN-1 (compound 3) is a high affinity dual inhibitor of FAAH (fatty acid amide hydrolase) and sEH (soluble epoxide hydrolase), with IC50 values of 7...
T67747 CB2R/FAAH modulator-3 2876918-67-9 98%
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are...
T28353 PDP-EA 861891-72-7 98%
PDP-EA is an activator of fatty acid amide hydrolase(FAAH) and enhances the amidohydrolase activity of FAAH.
T16515 PF 750 959151-50-9 98%
PF 750 is a selective and covalent inhibitor of FAAH. PF 750 shows IC50s varying from 16.2 to 595 nM in different incubation times.
T9374 AA38-3 65815-76-1
AA38-3 inhibites three SHs (ABHD6, ABHD11, and FAAH)
T6714 URB-597 546141-08-6 97.84%
URB597 is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets.
T2859 Biochanin A 491-80-5 98%
Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a naturally occurring fatty ...
T11256 FAAH inhibitor 1 326866-17-5 98.05%
FAAH inhibitor 1 is an effective FAAH inhibitor with an IC50 of 18 nM.
T15802 LY2183240 874902-19-9 98.17%
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 27...
T5357 ARN272 488793-85-7 98.23%
ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).
T7688 4-Nonylphenylboronic acid 256383-45-6 99.13%
4-Nonylphenylboronic acid is a inhibitor of FAAH.
T15268 FAAH-IN-2 184475-71-6 99.18%
FAAH-IN-2 is a potent inhibitor of FAAH(fatty acid amide hydrolase).
T1325 Carprofen 53716-49-7 99.45%
Carprofen is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic activities.
T8646 URB937 1357160-72-5 99.55%
URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM).
T4859 1-Monomyristin 589-68-4 99.58%
1-Myristoyl-rac-glycerol, a 1-monoglyceride of myristic acid, has antibacterial activity against several Gram-positive bacterial strains. 1-Myristoyl-rac-glycero...
T6043 PF-3845 1196109-52-0 99.58%
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
FAAH-IN-1
T11255
FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.
SA 47
T16847
SA 47 is a selective and effective inhibitor of fatty acid amide hydrolase and carbamate.
CB2R/FAAH modulator-2
T67745
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-2 acts as a CB2R agonist and FAAH inhibitor, the Ki value...
SA57
T12826
SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).
Dual FAAH/sEH-IN-1
T63536
Dual FAAH/sEH-IN-1 (compound 3) is a high affinity dual inhibitor of FAAH (fatty acid amide hydrolase) and sEH (soluble epoxide hydrolase), with IC50 values of 7...
CB2R/FAAH modulator-3
T67747
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are...
PDP-EA
T28353
PDP-EA is an activator of fatty acid amide hydrolase(FAAH) and enhances the amidohydrolase activity of FAAH.
PF 750
T16515
PF 750 is a selective and covalent inhibitor of FAAH. PF 750 shows IC50s varying from 16.2 to 595 nM in different incubation times.
AA38-3
T9374
AA38-3 inhibites three SHs (ABHD6, ABHD11, and FAAH)
URB-597
T6714
URB597 is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets.
Biochanin A
T2859
Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a naturally occurring fatty ...
FAAH inhibitor 1
T11256
FAAH inhibitor 1 is an effective FAAH inhibitor with an IC50 of 18 nM.
LY2183240
T15802
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 27...
ARN272
T5357
ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).
4-Nonylphenylboronic acid
T7688
4-Nonylphenylboronic acid is a inhibitor of FAAH.
FAAH-IN-2
T15268
FAAH-IN-2 is a potent inhibitor of FAAH(fatty acid amide hydrolase).
Carprofen
T1325
Carprofen is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic activities.
URB937
T8646
URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM).
1-Monomyristin
T4859
1-Myristoyl-rac-glycerol, a 1-monoglyceride of myristic acid, has antibacterial activity against several Gram-positive bacterial strains. 1-Myristoyl-rac-glycero...
PF-3845
T6043
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
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