T2338 |
JZL195 |
JZL195 is a selective and efficacious dual FAAH/MAGL inhibitor. |
T2684 |
JNJ1661010 |
JNJ-1661010 is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2. |
T2859 |
Biochanin A |
Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a naturally occurring fatty...
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T3215 |
JNJ42165279 |
JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-4216527...
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T3354 |
BIA10-2474 |
BIA10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH) that increases levels of the neurotransmitter anandamide in the central ne...
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T6043 |
PF3845 |
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2. |
T6714 |
URB597 |
URB597 is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets. |
T4323 |
PF04457845 |
PF-04457845 is a greatly and effctive FAAH inhibitor, and for hFAAH(IC50=7.2±0.63 nM) and rFAAH(IC50=7.4±0.62 nM). |
T7688 |
4-Nonylphenylboronic acid |
4-Nonylphenylboronic acid is a inhibitor of FAAH. |
T12826 |
SA57 |
SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH). |
T11255 |
FAAH-IN-1 |
FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively. |
T16515 |
PF 750 |
PF 750 is a selective and covalent fatty acid amide hydrolase inhibitor, It shows IC50s varied from 16.2-595 nM in different pre-incubation times. |
T16847 |
SA 47 |
SA 47 is a selective and effective inhibitor of fatty acid amide hydrolase and carbamate. |
T8646 |
URB937 |
URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM). |
T15268 |
FAAH-IN-2 |
FAAH-IN-2 is a potent inhibitor of FAAH(fatty acid amide hydrolase). |
T8927 |
WWL 154 |
WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor. |