TN3806 |
Dehydroglyasperin C
|
199331-35-6
|
98%
|
|
Dehydroglyasperin C is a potent NAD(P)H:oxidoquinone reductase (NQO1) and phase 2 enzyme inducer. Dehydroglyasperin C possesses potent antioxidant, cancer chemop...
|
T16361 |
Nucleocidin
|
24751-69-7
|
98%
|
|
Nucleocidin is an antitrypanosomal antibiotic. Nucleocidin inhibiting the transfer of labeled amino acid from S-RNA to protein.
|
T64376 |
WAY-652509
|
854355-54-7
|
98%
|
|
WAY-652509 is a Quinone reductase 2 inhibitor with IC50 of 0.6μM.
|
T39635 |
Obafistat
|
2160582-57-8
|
98%
|
|
Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4).
|
T38684 |
AKR1C3-IN-4
|
1284180-11-5
|
98%
|
|
AKR1C3-IN-4 is a potent and selective inhibitor of aldo-keto reductase 1C3 (AKR1C3) with an IC50 of 0.56 μM. AKR1C3-IN-4 has the potential for castrate resistant...
|
T0342 |
Carvedilol phosphate hemihydrate
|
610309-89-2
|
100%
|
|
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intri...
|
T1314 |
Triclosan
|
3380-34-5
|
100%
|
|
Triclosan is an antibacterial and antifungal agent.
|
T7374 |
2-HBA
|
131359-24-5
|
95.01%
|
|
2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.
|
T6099 |
Setanaxib
|
1218942-37-0
|
96.72%
|
|
GKT137831 is a potent, specific dual NADPH oxidase (NOX1/4) inhibitor.
|
T4529 |
ASP-9521
|
1126084-37-4
|
96.96%
|
|
ASP-9521 is an effective, specific and orally available AKR1C3 inhibitor (IC50: 11 nM, for human).
|
TN2126 |
Quercetin-3-O-glucose-6''-acetate
|
54542-51-7
|
97.48%
|
|
Quercetin-3-O-glucose-6''-acetate is an inhibitor of NADPH oxidase. Quercetin-3-O-glucose-6''-acetate has antioxidant activities.
|
T4359 |
VAS2870
|
722456-31-7
|
97.49%
|
|
VAS2870 is an inhibitor of NADPH oxidase (NOX).
|
T7191 |
Diphenyleneiodonium chloride
|
4673-26-1
|
98%
|
|
Diphenyleneiodonium chloride(DPI) is an irreversible inhibitor of iNOS and eNOS (IC50 values of 50 nM and 0.3 µM, respectively),and displays broad-spectrum bacte...
|
T7406 |
AKR1C3-IN-1
|
327092-81-9
|
98%
|
|
AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).
|
T0441 |
Pasiniazid
|
2066-89-9
|
98%
|
|
Pasiniazid is an anti-TB and anti-leprosy drug.
|
T8408 |
GKT136901
|
955272-06-7
|
98.29%
|
|
GKT136901 is an inhibitor of NOX1/4.It acts as Selective and Direct Scavenger of Peroxynitrite
|
T15433 |
GSK2795039
|
1415925-18-6
|
98.68%
|
|
GSK2795039 inhibits reactive oxygen species (ROS) production and NADPH consumption. GSK2795039 decreases apoptosis. GSK2795039 is an inhibitor of NADPH oxidase 2...
|
T10353 |
APX-115 free base
|
1270084-92-8
|
99.03%
|
|
APX-115 free base (Ewha-18278 free base) is a potent, orally active pan NADPH oxidase (Nox) inhibitor (Kis: 1.08 μM, 0.57 μM, and 0.63 μM for Nox1, Nox2, and Nox...
|
T16342 |
KL1333
|
1800405-30-4
|
99.27%
|
|
KL1333 enhances energy metabolism and mitochondrial dysfunction in MELAS fibroblasts. Elevated NAD+ levels trigger the activation of SIRT1 and AMPK, and subseque...
|
T14151 |
AKR1C1-IN-1
|
4906-68-7
|
99.46%
|
|
AKR1C1-IN-1 is a human 20α-hydroxysteroid dehydrogenase (AKR1C1) inhibitor (Ki: 4 nM for AKR1C1).
|