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AhR

The aryl hydrocarbon receptor (AHR) is a member of the basic helix-loop-helix-period-aryl hydrocarbon receptor nuclear translocator-single-minded (bHLH-PAS) family of transcription factors, which act as biological sensors by initiating gene expression programs in response to endogenous and exogenous signals.
Cat. No. Product name CAS No. Purity Chemical Structure
T20625 Prochloraz 67747-09-5 98%
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
T5541 PDM11 1032508-03-4
PDM 11 is an antagonist of aryl hydrocarbon receptor (AhR)
T23151 Phortress 328087-38-3 100%
Phortress is a high affinity AhR ligand that elicits antitumor activity by inducing transcription of CYP1A1.
T4607 CAY 10465 688348-33-6 100%
CAY 10465 is a selective and high-affinity AhR agonist, with a Ki of 0.2 nM, and shows no effect on estrogen receptor (Ki >100000 nM).
T4644 Tapinarof 79338-84-4 100%
Tapinarof is targeted as a topical cream treatment for psoriasis, a chronic autoimmune skin disease.
T10938 D-Kynurenine 13441-51-5 97.08%
D-Kynurenine is a metabolite of D-tryptophan and an agonist of GPR109B. D-Kynurenine activates AhR and promotes the conversion of the epithelium to mesenchyme. D...
T5622 BAY-218 2162982-11-6 98%
AHR antagonist 1 is an aryl hydrocarbon receptor (AHR) antagonist , has an IC50 of 39.9 nM in human cell line.
T7202 ITE 448906-42-1 98%
ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR) (Ki : 3 nM), has immunosuppressive activity.
T4928 L-Kynurenine 2922-83-0 98.44%
L-Kynurenine is a key intermediate in the breakdown pathway of tryptophan. L-Kynurenine is a substrate of kynureninase, KMO, and KAT associated with the suppress...
T1046 Mexiletine hydrochloride 5370-01-4 98.44%
Mexiletine Hydrochloride is the hydrochloride salt form of mexiletine, a local anesthetic and antiarrhythmic (Class IB) agent structurally related to lidocaine. ...
TN1451 Brevifolincarboxylic acid 18490-95-4 99.42%
Brevifolincarboxylic acid is a natural product isolated from Polygonum capitatum, it has inhibitory effect on the aryl hydrocarbon receptor (AhR). Brevifolincarb...
T4608 PDM2 688348-25-6 99.57%
PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.
T9822 WAY-605471 378223-81-5 99.57%
WAY-605471 is a AHR antagonist with IC50 of 0.5 - 1 μM.
T2448 CH-223191 301326-22-7 99.58%
CH-223191 is a potent and specific antagonist for aryl hydrocarbon receptor (AhR).
T10007 1,4-Chrysenequinone 100900-16-1 99.65%
1,4-Chrysenequinone acts as an activator of aryl hydrocarbon receptor (AhR).
T0343 Nimodipine 66085-59-4 99.71%
Nimodipine, a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.
T5281 Skatole 83-34-1 99.74%
Skatole is produced by intestinal bacteria. Skatole regulates intestinal epithelial cellular functions through activating aryl hydrocarbon receptors and p38.
T1960 YL-109 36341-25-0 99.77%
YL-109, a novel anticancer agent, can inhibit breast Y cell growth and invasiveness in vitro and in vivo.
T4938 Potassium 1H-indol-3-yl sulfate 2642-37-7 99.87%
Indoxyl sulfate (potassium salt) is an agonist for the human aryl hydrocarbon receptor (AHR). The aryl hydrocarbon receptor (AhR) has recently emerged as a patho...
T1159 Leflunomide 75706-12-6 99.9%
Leflunomide is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis.
Prochloraz
T20625
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
PDM11
T5541
PDM 11 is an antagonist of aryl hydrocarbon receptor (AhR)
Phortress
T23151
Phortress is a high affinity AhR ligand that elicits antitumor activity by inducing transcription of CYP1A1.
CAY 10465
T4607
CAY 10465 is a selective and high-affinity AhR agonist, with a Ki of 0.2 nM, and shows no effect on estrogen receptor (Ki >100000 nM).
Tapinarof
T4644
Tapinarof is targeted as a topical cream treatment for psoriasis, a chronic autoimmune skin disease.
D-Kynurenine
T10938
D-Kynurenine is a metabolite of D-tryptophan and an agonist of GPR109B. D-Kynurenine activates AhR and promotes the conversion of the epithelium to mesenchyme. D...
BAY-218
T5622
AHR antagonist 1 is an aryl hydrocarbon receptor (AHR) antagonist , has an IC50 of 39.9 nM in human cell line.
ITE
T7202
ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR) (Ki : 3 nM), has immunosuppressive activity.
L-Kynurenine
T4928
L-Kynurenine is a key intermediate in the breakdown pathway of tryptophan. L-Kynurenine is a substrate of kynureninase, KMO, and KAT associated with the suppress...
Mexiletine hydrochloride
T1046
Mexiletine Hydrochloride is the hydrochloride salt form of mexiletine, a local anesthetic and antiarrhythmic (Class IB) agent structurally related to lidocaine. ...
Brevifolincarboxylic acid
TN1451
Brevifolincarboxylic acid is a natural product isolated from Polygonum capitatum, it has inhibitory effect on the aryl hydrocarbon receptor (AhR). Brevifolincarb...
PDM2
T4608
PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.
WAY-605471
T9822
WAY-605471 is a AHR antagonist with IC50 of 0.5 - 1 μM.
CH-223191
T2448
CH-223191 is a potent and specific antagonist for aryl hydrocarbon receptor (AhR).
1,4-Chrysenequinone
T10007
1,4-Chrysenequinone acts as an activator of aryl hydrocarbon receptor (AhR).
Nimodipine
T0343
Nimodipine, a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.
Skatole
T5281
Skatole is produced by intestinal bacteria. Skatole regulates intestinal epithelial cellular functions through activating aryl hydrocarbon receptors and p38.
YL-109
T1960
YL-109, a novel anticancer agent, can inhibit breast Y cell growth and invasiveness in vitro and in vivo.
Potassium 1H-indol-3-yl sulfate
T4938
Indoxyl sulfate (potassium salt) is an agonist for the human aryl hydrocarbon receptor (AHR). The aryl hydrocarbon receptor (AhR) has recently emerged as a patho...
Leflunomide
T1159
Leflunomide is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis.
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