Nimodipine, a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells. |
Mexiletine Hydrochloride is the hydrochloride salt form of mexiletine, a local anesthetic and antiarrhythmic (Class IB) agent structurally related to lidocaine....
Leflunomide is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis. |
StemRegenin 1 is an aryl hydrocarbon receptor (AhR) inhibitor. |
YL-109, a novel anticancer agent, can inhibit breast Y cell growth and invasiveness in vitro and in vivo. |
CH-223191 is a potent and specific antagonist for aryl hydrocarbon receptor (AhR). |
Tapinarof is targeted as a topical cream treatment for psoriasis, a chronic autoimmune skin disease. |
||Indoxyl sulfate potassium salt
Indoxyl sulfate (potassium salt) is an agonist for the human aryl hydrocarbon receptor (AHR). The aryl hydrocarbon receptor (AhR) has recently emerged as a path...
L-Kynurenine is a key intermediate in the breakdown pathway of tryptophan. L-Kynurenine is a substrate of kynureninase, KMO, and KAT associated with the suppres...
||AHR antagonist 1
AHR antagonist 1 is an aryl hydrocarbon receptor (AHR) antagonist , has an IC50 of 39.9 nM in human cell line. |
ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR) (Ki : 3 nM), has immunosuppressive activity. |
PDM 11 is an antagonist of aryl hydrocarbon receptor (AhR) |
1,4-Chrysenequinone acts as an activator of aryl hydrocarbon receptor (AhR). |