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Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Cat No. product name
T35337L Teduglutide acetate Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
TP1863L Glucagon (19-29), human acetate Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
T15389L Glucagon (1-29), bovine, human, porcine hydrochloride Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphorylatio...
TP2071L Bay 55-9837 acetate Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
TP1039 Secretin (33-59), rat Secretin (33-59), rat is a 27-aa peptide, acts on secretin receptor, enhances the secretion of bicarbonate, enzymes, and K+ from the pancreas.
TP1103 Cotadutide acetate Cotadutide acetate (MEDI0382 acetate) is a potent peptide dual agonist of glucagon-like peptide-1 (GLP-1) and glucagon receptor with EC50 values of 6.9 pM and 10...
TP2252 GLP-1 (9-36) amide antagonist at the human GLP-1 receptor
TP1376 GLP-1(7-37) acetate(106612-94-6 free base) Glp-1 (7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
T9579 GLP-1 receptor agonist 9 1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
TP1148L Glucagon-like peptide 1 (1-37), human acetate Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
T0294 6α-Methylprednisolone 21-hemisuccinate sodium salt METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
T35337 Teduglutide Teduglutide (ALX-0600, Gattex, Revestive, TAK 633)是人胰高血糖素样肽-2 (GLP-2)的类似物,可与GLP-2 receptors结合。Teduglutide 在动物模型中可延长 GLP-2 的肠道营养特性。
T19850 Semaglutide Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
T8355 Exenatide acetate Exendin-4 is a glucagon-like protein-1 (GLP-1) receptor agonist
T8748 Exendin-4 acetate Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
T9226 CCG-143140 CCG-143140 is a GLP-1 receptor inverse agonists.
T8876 PF-06882961 Tris PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
T7364 NNC-0640 NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
T12878 Semaglutide TFA (910463-68-2 free base) Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T12431 PF-06882961 PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
T11408 GLP-1 receptor agonist 1 GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
T11845 LGD-6972 LGD-6972 is an antagonist of glucagon receptor.
TP1111L Tirzepatide Acetate(2023788-19-2 free base) Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.
TP1452L1 HAEGTFTSD acetate(926018-45-3 free base) HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
TP1469 Lixisenatide acetate (320367-13-3 free base) Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
TP1419L HAEGTFT acetate(926018-95-3 free base) HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
TP2100 Avexitide Avexitide (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
TP1796 Albiglutide TFA (782500-75-8 free base) Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
TQ0124 BETP BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
TQ0239 PF-06291874 PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
T6876 Liraglutide Liraglutide is a long-acting GLP-1 receptor agonist.
T3896 Shanzhiside methyl ester Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 ...
T3422 GRA Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor.
T3984 GLP-1(7-36), amide GLP-1 (7-36) amide is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays vari...
T3967 Exendin-4 Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer ...
Teduglutide acetate
T35337L
Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
Glucagon (19-29), human acetate
TP1863L
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
Glucagon (1-29), bovine, human, porcine hydrochloride
T15389L
Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphoryla...
Bay 55-9837 acetate
TP2071L
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
Secretin (33-59), rat
TP1039
Secretin (33-59), rat is a 27-aa peptide, acts on secretin receptor, enhances the secretion of bicarbonate, enzymes, and K+ from the pancreas.
Cotadutide acetate
TP1103
Cotadutide acetate (MEDI0382 acetate) is a potent peptide dual agonist of glucagon-like peptide-1 (GLP-1) and glucagon receptor with EC50 values of 6.9 pM...
GLP-1 (9-36) amide
TP2252
antagonist at the human GLP-1 receptor
GLP-1(7-37) acetate(106612-94-6 free base)
TP1376
Glp-1 (7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
GLP-1 receptor agonist 9
T9579
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
Glucagon-like peptide 1 (1-37), human acetate
TP1148L
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
6α-Methylprednisolone 21-hemisuccinate sodium salt
T0294
METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
Teduglutide
T35337
Semaglutide
T19850
Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
Exenatide acetate
T8355
Exendin-4 is a glucagon-like protein-1 (GLP-1) receptor agonist
Exendin-4 acetate
T8748
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
CCG-143140
T9226
CCG-143140 is a GLP-1 receptor inverse agonists.
PF-06882961 Tris
T8876
PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
NNC-0640
T7364
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
Semaglutide TFA (910463-68-2 free base)
T12878
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
PF-06882961
T12431
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
GLP-1 receptor agonist 1
T11408
GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
LGD-6972
T11845
LGD-6972 is an antagonist of glucagon receptor.
Tirzepatide Acetate(2023788-19-2 free base)
TP1111L
Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.
HAEGTFTSD acetate(926018-45-3 free base)
TP1452L1
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
Lixisenatide acetate (320367-13-3 free base)
TP1469
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
HAEGTFT acetate(926018-95-3 free base)
TP1419L
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
Avexitide
TP2100
Avexitide (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
Albiglutide TFA (782500-75-8 free base)
TP1796
Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
BETP
TQ0124
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
PF-06291874
TQ0239
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
Liraglutide
T6876
Liraglutide is a long-acting GLP-1 receptor agonist.
Shanzhiside methyl ester
T3896
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38...
GRA Ex-25
T3422
GRA-Ex-25 is an inhibitor of glucagon receptor.
GLP-1(7-36), amide
T3984
GLP-1 (7-36) amide is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays vari...
Exendin-4
T3967
Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer ...