T10572L |
BMT-124110 Formate
|
T10572L
|
98%
|
|
BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase ...
|
T24152 |
HTH-01-091
|
2000209-42-5
|
98%
|
|
HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK...
|
T16931 |
SRPKIN-1
|
2089226-94-6
|
98%
|
|
SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
|
T8957 |
CRT0066101
|
956121-30-5
|
98%
|
|
CRT0066101 is an inhibitor of PKD.
|
T8362 |
Benzamidine hydrochloride
|
1670-14-0
|
98%
|
|
Benzamidine HCl is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 µM, respectively).
|
T8535 |
GAK inhibitor 49
|
319492-82-5
|
98%
|
|
GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
|
TQ0104 |
CRT0066101 dihydrochloride
|
1883545-60-5
|
98%
|
|
CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).
|
T9276 |
SBC-115337
|
423148-46-3
|
98%
|
|
SBC-115337 is a PCSK9 inhibitor.
|
T6283 |
Wortmannin
|
19545-26-7
|
98%
|
|
Wortmannin is the first described PI3K inhibitor with IC50 of 3 nM, with little selectivity within the PI3K family. Also blocks autophagosome formation and poten...
|
T5169 |
SGC-GAK-1
|
2226517-76-4
|
98%
|
|
SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
|
T2458 |
CID755673
|
521937-07-5
|
98%
|
|
CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective PKD1 inhibition when compared with PLK1, AKT, CAMKIIα, CA...
|
T2391 |
Camostat mesylate
|
59721-29-8
|
98%
|
|
Camostat is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.
|
T4524 |
SBC-110736
|
1629166-02-4
|
98%
|
|
SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitor
|
T3050 |
ML-7 hydrochloride
|
110448-33-4
|
98%
|
|
ML-7 Hcl is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM); also inhibits smooth-musc...
|
TP1890L1 |
MLCK inhibitor peptide 18 acetate
|
TP1890L1
|
98%
|
|
MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinas...
|
T7444 |
6-(Dimethylamino)purine
|
938-55-6
|
98%
|
|
6-(Dimethylamino)purine is a serine threonine protein kinase and CDK inhibitor
|
T0610 |
Piceatannol
|
10083-24-6
|
98%
|
|
Piceatannol is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine kinases and inhibits NF-κB activat...
|
TN2082 |
Pinostrobin
|
480-37-5
|
98%
|
|
Pinostrobin, a potent flavonoid inducer, exerts a neuroprotective effect against Aα²(25-35)-induced neurotoxicity in PC12 cells, at least in part, via inhibiting...
|
T5194 |
SPHINX31
|
1818389-84-2
|
98%
|
|
SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).
|
T2153 |
1-NM-PP1
|
221244-14-0
|
98%
|
|
1 nM-PP1 is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.
|