Serine/threonin kinase

Serine threonine kinase belongs to protein kinase, which can phosphorylate the OH group of serine or threonine residues. Serine threonine kinases contain Rho kinase, Aurora kinase, AMP kinase, RAF kinase, Polo like kinase, PIM kinase, ATM kinase and other kinases. The cAMP/cGMP, Ca2+/calmodulin and diacylglycerol and multiple chenmical signals can regulate the activity of serine threonine kinases.

Cat. No.	Product name	CAS No.	Purity
T10572L	BMT-124110 Formate	T10572L	98%
T10572L	BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase ...
T24152	HTH-01-091	2000209-42-5	98%
T24152	HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK...
T16931	SRPKIN-1	2089226-94-6	98%
T16931	SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
T8957	CRT0066101	956121-30-5	98%
T8957	CRT0066101 is an inhibitor of PKD.
T8362	Benzamidine hydrochloride	1670-14-0	98%
T8362	Benzamidine HCl is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 µM, respectively).
T8535	GAK inhibitor 49	319492-82-5	98%
T8535	GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
TQ0104	CRT0066101 dihydrochloride	1883545-60-5	98%
TQ0104	CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).
T9276	SBC-115337	423148-46-3	98%
T9276	SBC-115337 is a PCSK9 inhibitor.
T6283	Wortmannin	19545-26-7	98%
T6283	Wortmannin is the first described PI3K inhibitor with IC50 of 3 nM, with little selectivity within the PI3K family. Also blocks autophagosome formation and poten...
T5169	SGC-GAK-1	2226517-76-4	98%
T5169	SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
T2458	CID755673	521937-07-5	98%
T2458	CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective PKD1 inhibition when compared with PLK1, AKT, CAMKIIα, CA...
T2391	Camostat mesylate	59721-29-8	98%
T2391	Camostat is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.
T4524	SBC-110736	1629166-02-4	98%
T4524	SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitor
T3050	ML-7 hydrochloride	110448-33-4	98%
T3050	ML-7 Hcl is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM); also inhibits smooth-musc...
TP1890L1	MLCK inhibitor peptide 18 acetate	TP1890L1	98%
TP1890L1	MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinas...
T7444	6-(Dimethylamino)purine	938-55-6	98%
T7444	6-(Dimethylamino)purine is a serine threonine protein kinase and CDK inhibitor
T0610	Piceatannol	10083-24-6	98%
T0610	Piceatannol is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine kinases and inhibits NF-κB activat...
TN2082	Pinostrobin	480-37-5	98%
TN2082	Pinostrobin, a potent flavonoid inducer, exerts a neuroprotective effect against Aα²(25-35)-induced neurotoxicity in PC12 cells, at least in part, via inhibiting...
T5194	SPHINX31	1818389-84-2	98%
T5194	SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).
T2153	1-NM-PP1	221244-14-0	98%
T2153	1 nM-PP1 is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.