Cat. No. | Product name | CAS No. | Purity | Chemical Structure |
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T13383 | Zamicastat | 1080028-80-3 | 98% |
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Zamicastat is an inhibitor of dopamine β-hydroxylase (DBH), and is also a concentration-dependent dual inhibitor of P-gp and BCRP(IC50 values of 73.8 μM and 17.0... | ||||
TN2233 | Spathulenol | 6750-60-3 | 98% |
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Spathulenol has immunomodulatory effect. Spathulenol shows the capacity to inhibit proliferation in the lymphocytes and to induce apoptosis in these cells possib... | ||||
TQ0043 | Dofequidar | 129716-58-1 | 98% |
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Dofequidar (MS-209) is a quinoline compound that can reverse P-glycoprotein (P-gp)-mediated MDR. | ||||
TN5114 | Taxinine | 3835-52-7 | 98% |
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Taxinine and Taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells. | ||||
TN1048 | Cnidilin | 14348-22-2 | 98% |
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Cnidilin has high BBB permeability and has pharmacokinetic potentials for the treatment of central nervous system diseases. | ||||
TN3937 | Ent-16alpha,17-Dihydroxyatisan-3-one | 112523-91-8 | 98% |
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ent-16alpha,17-Dihydroxyatisan-3-one and ent-16alpha,17-dihydroxykauran-3-one have apoptosis induction activities on L5178 human MDR1 gene-transfected mouse lymp... | ||||
TN1099 | Dihydroevocarpine | 15266-35-0 | 98% |
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Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is a... | ||||
TN4410 | Lappaol C | 64855-00-1 | 98% |
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Lappaol C has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. Lappaol C also ... | ||||
TN2726 | Jatrophane 5 | 210108-89-7 | 98% |
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Jatrophane 5 demonstrates the most powerful inhibition of P-gp, higher than R(+)-verapamil and tariquidar in colorectal multi-drug resistant (MDR) cells (DLD1-Tx... | ||||
T2A2486 | 3',4',5',5,7-Pentamethoxyflavone | 53350-26-8 | 98% |
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3',4',5',5,7-Pentamethoxyflavone has anti-inflammatory and cancer chemopreventive activities. 3',4',5',5,7-Pentamethoxyflavone could be used as an effective adju... | ||||
TN5124 | Taxuspine X | 194782-02-0 | 98% |
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Taxuspine X may have p-glycoprotein inhibitory activity. | ||||
TN1525 | Convallatoxin | 508-75-8 | 98% |
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Convallatoxin is a natural product | ||||
TN2263 | Tenacigenin B | 80508-42-5 | 98% |
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Standard reference | ||||
TN4819 | (-)-Praeruptorin A | 14017-71-1 | 98% |
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(-)-Praeruptorin A has anti-inflammatory, anti-contractile and anti-hyperplasia activities, it exerts distinct relaxant effects on isolated rat aorta rings depen... | ||||
TN2554 | 1-Monopalmitin | 542-44-9 | 98% |
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1-Monopalmitin has dielectric properties. 1-Monopalmitin inhibits the P-glycoprotein activity in intestinal Caco-2 cells. | ||||
TN4411 | Lappaol F | 69394-17-8 | 98% |
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1. Lappaol F has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. 2. Lap... |
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TN2257 | Tanshinone IIB | 17397-93-2 | 98% |
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Co-treatment with Tanshinone IIB (TSB) significantly inhibits the DNA laddering, cytotoxicity and apoptosis of rat cortical neurons induced by staurosporine in a... | ||||
TN2727 | Jatrophane 2 | 210108-86-4 | 98% |
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2,5,7,8,9,14-Hexaacetoxy-3-benzoyloxy-15-hydroxyjatropha-6(17),11E-diene (Jatrophane 2 ) exhibits significant antifeedant activity against a generalist plant-fee... | ||||
TN4749 | Pepluanin A | 670257-89-3 | 98% |
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Pepluanin A, shows a very high activity for a jatrophane diterpene, outperforming cyclosporin A by a factor of at least 2 in the inhibition of Pgp-mediated dauno... | ||||
TCS2336 | Evodine | 6989-38-4 | 98% |
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1. Evodine has antinociceptive activity. |