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Estrogen/progestogen Receptor

Estrogen receptors are a group of proteins found inside cells. They are receptors that are activated by the hormone estrogen (17β-estradiol). Two classes of estrogen receptor exist: ER, which is a member of the nuclear hormone family of intracellular receptors, and GPER (GPR30), which is a member of the rhodopsin-like family of G protein-coupled receptors.The progesterone receptor (PR), also known as NR3C3 or nuclear receptor subfamily 3, group C, member 3, is a protein found inside cells. It is activated by the steroid hormone progesterone.
Cat. No. Product name CAS No. Purity Chemical Structure
T11231 ERRγ Inverse Agonist 1 2316832-86-5 98%
ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].
T11222 ERB-196 550997-55-2 98%
Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.
T0171 Norethynodrel 68-23-5 98%
Norethynodrel is a synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uteri...
TN1679 Genistein 7,4'-di-O-β-D-glucoside 36190-98-4 98%
Genistein 7,4'-di-O-beta-D-glucopyranoside shows significant estrogenic proliferative effect in MCF-7 cell in sub-cytotoxic concentration range.
T12312 OP-1074 1443752-76-8 98%
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
T12329 Ospemifene D4 T12329 98%
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
T16351 NSC16168 6837-93-0 98%
NSC16168 inhibits DNA repair and potentiates CDDP efficacy in cancer. NSC16168 is a specific ERCC1-XPF inhibitor (IC50: 0.42 μM).
TQ0163 Sagittatoside A 118525-35-2 98%
Sagittatoside A selectively activates estrogen response element (ERE)-luciferase activity via ERα.
TN1690 Glabrene 60008-03-9 98%
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely t...
T6827 Endoxifen Z-isomer hydrochloride 1032008-74-4 98%
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
TN2200 Segetalin A 161875-97-4 98%
Segetalin A has estrogen-like activity.
T12278 NXT629 1454925-59-7 98%
NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 nM).
T6404 Bazedoxifene hydrochloride 198480-56-7 98%
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
TN2288 Uralenol 139163-15-8 98%
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as s...
TQ0149 Prinaberel 524684-52-4 98%
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
TN2045 Pelargonidin-3-O-glucoside chloride 18466-51-8 98%
Pelargonidin-3-O-glucopyranoside is the glucoside of Pelargonidin, an potential antidiabetic agent. Pelargonidin-3-O-glucopyranoside has antioxidant, anti-inflam...
T3645 Endoxifen E-isomer hydrochloride 1197194-61-8 98%
Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
T20720 Norethisterone enanthate 3836-23-5 98%
Norethindrone enanthate has antigonadotropic effects and can be used as a hormonal contraceptive. It is also a useful compound to study chem.-chem. interaction f...
T11230 ERRα antagonist-1 1072145-33-5 98%
ERRα antagonist-1 is a selective and high affinity estrogen-related receptor α (ERRα) antagonist. ERRα antagonist-1 inhibits interaction of ERRα with Proliferato...
T1579 Mestranol 72-33-3 98%
Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
ERRγ Inverse Agonist 1
T11231
ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].
ERB-196
T11222
Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.
Norethynodrel
T0171
Norethynodrel is a synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uteri...
Genistein 7,4'-di-O-β-D-glucoside
TN1679
Genistein 7,4'-di-O-beta-D-glucopyranoside shows significant estrogenic proliferative effect in MCF-7 cell in sub-cytotoxic concentration range.
OP-1074
T12312
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
Ospemifene D4
T12329
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
NSC16168
T16351
NSC16168 inhibits DNA repair and potentiates CDDP efficacy in cancer. NSC16168 is a specific ERCC1-XPF inhibitor (IC50: 0.42 μM).
Sagittatoside A
TQ0163
Sagittatoside A selectively activates estrogen response element (ERE)-luciferase activity via ERα.
Glabrene
TN1690
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely t...
Endoxifen Z-isomer hydrochloride
T6827
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
Segetalin A
TN2200
Segetalin A has estrogen-like activity.
NXT629
T12278
NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 nM).
Bazedoxifene hydrochloride
T6404
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
Uralenol
TN2288
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as s...
Prinaberel
TQ0149
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
Pelargonidin-3-O-glucoside chloride
TN2045
Pelargonidin-3-O-glucopyranoside is the glucoside of Pelargonidin, an potential antidiabetic agent. Pelargonidin-3-O-glucopyranoside has antioxidant, anti-inflam...
Endoxifen E-isomer hydrochloride
T3645
Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
Norethisterone enanthate
T20720
Norethindrone enanthate has antigonadotropic effects and can be used as a hormonal contraceptive. It is also a useful compound to study chem.-chem. interaction f...
ERRα antagonist-1
T11230
ERRα antagonist-1 is a selective and high affinity estrogen-related receptor α (ERRα) antagonist. ERRα antagonist-1 inhibits interaction of ERRα with Proliferato...
Mestranol
T1579
Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
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