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Glucocorticoid Receptor

The glucocorticoid receptor (GR, or GCR) also known as NR3C1 (nuclear receptor subfamily 3, group C, member 1) is the receptor to which cortisol and other glucocorticoids bind. The GR is expressed in almost every cell in the body and regulates genes controlling the development, metabolism, and immune response.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TN3910 Ecdysone 3604-87-3 100%
Ecdysone
Ecdysone is a major steroid hormone in insects and herbs. Ecdysone triggers mineralocorticoid receptor activation and induces cellular apoptosis. Ecdysone signal...
T78073 HP210 728039-52-9 98%
HP210
HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-re...
T80652 N-Demethyl Mifepristone 104004-96-8 98%
N-Demethyl Mifepristone
N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone's...
T0107 Halcinonide 3093-35-4 99.94%
Halcinonide
Halcinonide (Halciderm), a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.
T9022 AZD9977 1850385-64-6 99.92%
AZD9977
AZD9977 is a novel, selective modulator of mineralocorticoid receptor .
T0977 Medrysone 2668-66-8 99.91%
Medrysone
Medrysone (6α-Methyl-11β-hydroxyprogesterone) is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone ex...
T0261 Amcinonide 51022-69-6 99.9%
Amcinonide
Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.
T2526 Ciclesonide 126544-47-6 99.89%
Ciclesonide
Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
T0947L Dexamethasone Phosphate disodium 2392-39-4 99.88%
Dexamethasone Phosphate disodium
Dexamethasone Phosphate disodium (EGP437. Dex-Phos) is a water-soluble form of the synthetic glucocorticoid dexamethasone.
T2748 Cortodoxone 152-58-9 99.87%
Cortodoxone
Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
T1541 Drospirenone 67392-87-4 99.85%
Drospirenone
Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T0820 Triamcinolone acetonide 76-25-5 99.84%
Triamcinolone acetonide
Triamcinolone acetonide (Azmacort) is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is...
T1560 Prednisolone 50-24-8 99.83%
Prednisolone
Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
T0354 Canrenone 976-71-6 99.8%
Canrenone
Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity.
T3962 TPI-1 79756-69-7 99.79%
TPI-1
TPI-1 is a SHP-1 inhibitor.
T1076 Dexamethasone 50-02-2 99.77%
Dexamethasone
Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist and an IL receptor modulator. Dexamethasone has anti-inflammatory and immunosuppressive activit...
T6503 Fluorometholone Acetate 3801-06-7 99.77%
Fluorometholone Acetate
Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.
T1102 Mifepristone 84371-65-3 99.74%
Mifepristone
Mifepristone (C-1073) is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
T1559 Betamethasone dipropionate 5593-20-4 99.74%
Betamethasone dipropionate
Betamethasone Dipropionate is the 17, 21-dipropionate ester of betamethasone, a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory ...
T1284 Megestrol acetate 595-33-5 99.72%
Megestrol acetate
Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic pr...
Ecdysone
TN3910
Ecdysone is a major steroid hormone in insects and herbs. Ecdysone triggers mineralocorticoid receptor activation and induces cellular apoptosis. Ecdysone signal...
HP210
T78073
HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-re...
N-Demethyl Mifepristone
T80652
N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone's...
Halcinonide
T0107
Halcinonide (Halciderm), a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.
AZD9977
T9022
AZD9977 is a novel, selective modulator of mineralocorticoid receptor .
Medrysone
T0977
Medrysone (6α-Methyl-11β-hydroxyprogesterone) is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone ex...
Amcinonide
T0261
Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.
Ciclesonide
T2526
Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
Dexamethasone Phosphate disodium
T0947L
Dexamethasone Phosphate disodium (EGP437. Dex-Phos) is a water-soluble form of the synthetic glucocorticoid dexamethasone.
Cortodoxone
T2748
Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
Drospirenone
T1541
Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
Triamcinolone acetonide
T0820
Triamcinolone acetonide (Azmacort) is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is...
Prednisolone
T1560
Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
Canrenone
T0354
Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity.
TPI-1
T3962
TPI-1 is a SHP-1 inhibitor.
Dexamethasone
T1076
Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist and an IL receptor modulator. Dexamethasone has anti-inflammatory and immunosuppressive activit...
Fluorometholone Acetate
T6503
Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.
Mifepristone
T1102
Mifepristone (C-1073) is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
Betamethasone dipropionate
T1559
Betamethasone Dipropionate is the 17, 21-dipropionate ester of betamethasone, a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory ...
Megestrol acetate
T1284
Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic pr...
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TargetMol