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Glucocorticoid Receptor

The glucocorticoid receptor (GR, or GCR) also known as NR3C1 (nuclear receptor subfamily 3, group C, member 1) is the receptor to which cortisol and other glucocorticoids bind. The GR is expressed in almost every cell in the body and regulates genes controlling the development, metabolism, and immune response.
Cat No. product name
T2748 Cortodoxone Cortodoxone is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
T0034 Cortisone acetate Cortisone Acetate is the acetate salt form of cortisone, a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal...
T15389L Glucagon (1-29), bovine, human, porcine hydrochloride Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphorylatio...
T0276 Hydrocortisone Valerate Hydrocortisone Valerate has anti-inflammatory, antipruritic and vasoconstrictive properties.
T1076 Dexamethasone Dexamethasone is a glucocorticoid receptor agonist and an IL receptor modulator.Dexamethasone inhibits production of exosomes containing inflammatory microRNA-15...
T0977 Medrysone Medrysone is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone exerts its effect by interacting with ...
T0107 Halcinonide Halcinonide, a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.
T4277 Osilodrostat Osilodrostat (LCI699) is an effective inhibitor of human 11β-hydroxylase (IC50: 2.5 nM) and aldosterone synthase (IC50: 0.7 nM).
T6580 Meprednisone Betapar(Meprednisone) is a glucocorticoid and a methylated derivative of prednisone.
T0947L Dexamethasone Phosphate disodium Dexamethasone disodium phosphate is a water-soluble form of the synthetic glucocorticoid dexamethasone.
T1102 Mifepristone Mifepristone is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
T1284 Megestrol acetate Megestrol acetate is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic properties. ...
T14981 Clobetasone butyrate Clobetasone butyrate can be used to relieve corticosteroid-responsive dermatoses, including atopic dermatitis and psoriasis. Clobetasone butyrate is a synthetic ...
T1561 Clobetasol propionate Clobetasol propionate exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediated gene expre...
T2810 (20S)-Protopanaxatriol (20S)-Protopanaxatriol(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid receptor.
T0947 Dexamethasone acetate Dexamethasone Acetate is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addition to bind...
T0188 Fluticasone (propionate) Fluticasone propionate, derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR (glucocorticoid receptor) agonist....
T0181 Loteprednol etabonate Loteprednol Etabonate is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.
T1683 Actriol Actriol is always used as Glucocorticoid Receptor agonist.
T6503 Fluorometholone Acetate Fluorometholone Acetate is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.
T0948L Corticosterone Corticosterone is a sensitive inhibitor of monoamine transport.
T15102 Dexamethasone palmitate Dexamethasone palmitate is a prodrug of Dexamethasone and a glucocorticoid receptor agonist. It shows a 47-fold lower affinity for the glucocorticoid receptor th...
T1541 Drospirenone Drospirenone is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T4602 Hydrocortisone hemisuccinate Hydrocortisone 21-hemisuccinate is a corticosteroid used as an analytical and chromatography reagent.
T0270 Hydrocortisone 17-butyrate Hydrocortisone Butyrate is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
T3962 TPI-1 TPI-1 is a SHP-1 inhibitor.
T0354 Canrenone Canrenone is an aldosterone antagonist with potassium-sparing diuretic activity.
T0343 Nimodipine Nimodipine, a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.
TN3910 Ecdysone Ecdysone signaling through Ecdysone receptor isoform B1 is required cell autonomously for the muscle death. A nctional Bombyx Ecdysone receptor binds to EcRE-D a...
T2884 Cortisone Cortisone is a corticosteroid with potent glucocorticoid activity.
T1261 Medroxyprogesterone Acetate Medroxyprogesterone acetate is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally...
T1243 Hydrocortisone acetate Hydrocortisone acetate is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive properties.
T1614 Hydrocortisone Hydrocortisone, a glucocorticoid receptor agonist, promotes protein catabolism, gluconeogenesis, capillary wall stability, renal excretion of calcium, and suppre...
T0476 Spironolactone Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
T0294 6α-Methylprednisolone 21-hemisuccinate sodium salt METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
T1560 Prednisolone Prednisolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
T3033 Deoxycorticosterone acetate Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
T22367 Methylprednisolone succinate Methylprednisolone sodium succinate is a glucocorticoid used to treat a variety health issues including asthma, severe allergic reactions, gastrointestinal dise...
T21395 Finerenone Finerenone is a third-generation, selective, and orally available nonsteroidal mineralocorticoid receptor (MR) antagonist with IC50 of 18 nM for the treatment of...
T2548 Diflorasone Diflorasone is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive properties. Like other glucocorticoids, diflorasone enters the cell by dif...
T2526 Ciclesonide Ciclesonide(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
T9022 AZD9977 AZD 9977 is a novel, selective modulator of mineralocorticoid receptor .
T8777 Beclometasone BecloMethasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma...
T8396 Prednisone acetate Prednisone acetate is a glucocorticoid receptor agonist with immunomodulating properties and anti-inflammatory.
T0798 Triamcinolone Triamcinolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Upon cell entry, triamcinolone binds to and activates the gl...
T0820 Triamcinolone acetonide Triamcinolone acetonide is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is an anti-in...
T0367 Fluocinolone (Acetonide) Fluocinolone acetonide is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, ...
T0337 Prednisolone acetate Prednisolone Acetate is the acetate salt form of prednisolone, a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
T0261 Amcinonide Amcinonide is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.
T1124 Flumethasone Flumethasone is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.
Cortodoxone
T2748
Cortodoxone is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
Cortisone acetate
T0034
Cortisone Acetate is the acetate salt form of cortisone, a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal...
Glucagon (1-29), bovine, human, porcine hydrochloride
T15389L
Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphoryla...
Hydrocortisone Valerate
T0276
Hydrocortisone Valerate has anti-inflammatory, antipruritic and vasoconstrictive properties.
Dexamethasone
T1076
Dexamethasone is a glucocorticoid receptor agonist and an IL receptor modulator.Dexamethasone inhibits production of exosomes containing inflammatory microRNA-15...
Medrysone
T0977
Medrysone is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone exerts its effect by interacting with ...
Halcinonide
T0107
Halcinonide, a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.
Osilodrostat
T4277
Osilodrostat (LCI699) is an effective inhibitor of human 11β-hydroxylase (IC50: 2.5 nM) and aldosterone synthase (IC50: 0.7 nM).
Meprednisone
T6580
Betapar(Meprednisone) is a glucocorticoid and a methylated derivative of prednisone.
Dexamethasone Phosphate disodium
T0947L
Dexamethasone disodium phosphate is a water-soluble form of the synthetic glucocorticoid dexamethasone.
Mifepristone
T1102
Mifepristone is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
Megestrol acetate
T1284
Megestrol acetate is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic properties. ...
Clobetasone butyrate
T14981
Clobetasone butyrate can be used to relieve corticosteroid-responsive dermatoses, including atopic dermatitis and psoriasis. Clobetasone butyrate is a synthetic ...
Clobetasol propionate
T1561
Clobetasol propionate exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediated gene expre...
(20S)-Protopanaxatriol
T2810
(20S)-Protopanaxatriol(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid receptor.
Dexamethasone acetate
T0947
Dexamethasone Acetate is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addition to bind...
Fluticasone (propionate)
T0188
Fluticasone propionate, derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR (glucocorticoid receptor) agonist....
Loteprednol etabonate
T0181
Loteprednol Etabonate is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.
Actriol
T1683
Actriol is always used as Glucocorticoid Receptor agonist.
Fluorometholone Acetate
T6503
Fluorometholone Acetate is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.
Corticosterone
T0948L
Corticosterone is a sensitive inhibitor of monoamine transport.
Dexamethasone palmitate
T15102
Dexamethasone palmitate is a prodrug of Dexamethasone and a glucocorticoid receptor agonist. It shows a 47-fold lower affinity for the glucocorticoid receptor th...
Drospirenone
T1541
Drospirenone is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
Hydrocortisone hemisuccinate
T4602
Hydrocortisone 21-hemisuccinate is a corticosteroid used as an analytical and chromatography reagent.
Hydrocortisone 17-butyrate
T0270
Hydrocortisone Butyrate is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
TPI-1
T3962
TPI-1 is a SHP-1 inhibitor.
Canrenone
T0354
Canrenone is an aldosterone antagonist with potassium-sparing diuretic activity.
Nimodipine
T0343
Nimodipine, a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.
Ecdysone
TN3910
Ecdysone signaling through Ecdysone receptor isoform B1 is required cell autonomously for the muscle death. A nctional Bombyx Ecdysone receptor binds to EcRE-D a...
Cortisone
T2884
Cortisone is a corticosteroid with potent glucocorticoid activity.
Medroxyprogesterone Acetate
T1261
Medroxyprogesterone acetate is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally...
Hydrocortisone acetate
T1243
Hydrocortisone acetate is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive properties.
Hydrocortisone
T1614
Hydrocortisone, a glucocorticoid receptor agonist, promotes protein catabolism, gluconeogenesis, capillary wall stability, renal excretion of calcium, and suppre...
Spironolactone
T0476
Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
6α-Methylprednisolone 21-hemisuccinate sodium salt
T0294
METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
Prednisolone
T1560
Prednisolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
Deoxycorticosterone acetate
T3033
Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
Methylprednisolone succinate
T22367
Methylprednisolone sodium succinate is a glucocorticoid used to treat a variety health issues including asthma, severe allergic reactions, gastrointestinal dise...
Finerenone
T21395
Finerenone is a third-generation, selective, and orally available nonsteroidal mineralocorticoid receptor (MR) antagonist with IC50 of 18 nM for the treatment of...
Diflorasone
T2548
Diflorasone is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive properties. Like other glucocorticoids, diflorasone enters the cell by dif...
Ciclesonide
T2526
Ciclesonide(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
AZD9977
T9022
AZD 9977 is a novel, selective modulator of mineralocorticoid receptor .
Beclometasone
T8777
BecloMethasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma...
Prednisone acetate
T8396
Prednisone acetate is a glucocorticoid receptor agonist with immunomodulating properties and anti-inflammatory.
Triamcinolone
T0798
Triamcinolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Upon cell entry, triamcinolone binds to and activates the gl...
Triamcinolone acetonide
T0820
Triamcinolone acetonide is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is an anti-in...
Fluocinolone (Acetonide)
T0367
Fluocinolone acetonide is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, ...
Prednisolone acetate
T0337
Prednisolone Acetate is the acetate salt form of prednisolone, a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
Amcinonide
T0261
Amcinonide is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.
Flumethasone
T1124
Flumethasone is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.
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