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Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling
MAPK Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Cat. No. Product name CAS No. Purity Chemical Structure
T22849 ICI 199,441 hydrochloride 115199-84-3 98%
ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
TN3367 Akuammidine 639-36-1 98%
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
T11478L GSK1521498 free base 1007573-18-3 98%
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
T11198 Endomorphin 2 TFA 1276124-00-5 98%
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
T13419 ROCK-IN-1 934387-35-6 98%
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
T7404 Dermorphin 77614-16-5 98%
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
T7567 Adrenorphin 88377-68-8 98%
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
TN3368 Akuammigine 642-17-1 98%
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T4633 Asimadoline 153205-46-0 98%
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
TP2036 DPDPE 88373-73-3 98%
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
T7306 Valorphin 144313-54-2 98%
Valorphin has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
T12169 Naltrindole hydrochloride 111469-81-9 98%
Naltrindole hydrochloride is a selective and non-peptide δ opioid receptor antagonist(Ki = 0.02 nM).
T7576 β-Casomorphin, bovine 72122-62-4 98%
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
T12241 Norbinaltorphimine dihydrochloride 113158-34-2 98%
Norbinaltorphimine dihydrochloride is a potent and selective antagonist of κ opioid receptor.
TN5017 Sideritoflavone 70360-12-2 98%
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
T15165 DPI-3290 182417-73-8 98%
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
T13438 (R,S)-Ivosidenib 2070009-31-1 98%
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
TP1367L [D-Ala2]leucine-enkephalin acetate TP1367L 98%
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
T11479 GSK1521498 1426543-84-1 98%
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
T12314 Opioid receptor modulator 1 77514-44-4 98%
Opioid receptor modulator 1 is a modulator of opioid receptor.
ICI 199,441 hydrochloride
T22849
ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
Akuammidine
TN3367
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
GSK1521498 free base
T11478L
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
Endomorphin 2 TFA
T11198
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
ROCK-IN-1
T13419
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
Dermorphin
T7404
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
Adrenorphin
T7567
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
Asimadoline
T4633
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
DPDPE
TP2036
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
Valorphin
T7306
Valorphin has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
Naltrindole hydrochloride
T12169
Naltrindole hydrochloride is a selective and non-peptide δ opioid receptor antagonist(Ki = 0.02 nM).
β-Casomorphin, bovine
T7576
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
Norbinaltorphimine dihydrochloride
T12241
Norbinaltorphimine dihydrochloride is a potent and selective antagonist of κ opioid receptor.
Sideritoflavone
TN5017
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
DPI-3290
T15165
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
(R,S)-Ivosidenib
T13438
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
[D-Ala2]leucine-enkephalin acetate
TP1367L
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
GSK1521498
T11479
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
Opioid receptor modulator 1
T12314
Opioid receptor modulator 1 is a modulator of opioid receptor.
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