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Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Cat No. product name
T41284 Nalfurafine Nalfurafine 是一种有效且特异性的 G 蛋白偏倚 κ-阿片受体激动剂,具有高转化潜力。 Nalfurafine 增强了 MOR 靶向镇痛药的生物学作用,可用于尿毒症瘙痒症的相关研究。
T38193L β-Endorphin (1-27) (human) acetate β-Endorphin (1-27) (human) acetate 存在于大脑垂体和下丘脑中,具有镇痛活性。 β-Endorphin (1-27) (human) acetate 是一种阿片受体激动剂,对 μ-阿片受体和 δ-阿片受体具有较好的亲和力。
T20166L Deltorphin acetate Deltorphin acetate 是一种从青蛙 Phyllomedusa bicolor 的皮肤分泌物中获得的物质,对 δ-阿片受体具有高选择性和亲和力。
T2921 Sinomenine hydrochloride Sinomenine hydrochloride is extracted from Sinomenium Acutum Rehderett Wilson.
T0478 Progesterone Progesterone is the major progestational steroid that is secreted primarily by the CORPUS LUTEUM and the PLACENTA. Progesterone acts on the UTERUS, the MAMMARY G...
T0137 Mirtazapine Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T4633 Asimadoline Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
T7173 [Leu5]-Enkephalin [Leu5]-Enkephalin is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
T22752L (D-Ser2)-Leu-Enkephalin-Thr (D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.
T0929 Docusate sodium Docusate is an orally available, over-the-counter laxative and stool softener used to treat or prevent constipation. Docusate has not been linked to serum enzyme...
T23076L Nociceptin (1-7) acetate Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor. Nociceptin (1-7) combines with nociceptin reduces hyperalgesia and has a...
TP1940L1 Ac-RYYRIK-NH2 acetate Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial ag...
T0209 Loperamide hydrochloride Loperamide Hydrochloride is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
T21660L B-Casomorphin (1-3) Acetate b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
T2726 Sinomenine Sinomenine is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
T26869 BMS-986122 BMS-986122 is a positive allosteric modulator of the μ-Opioid Receptor.
T7748 Dermorphin TFA Dermorphin TFA is a new class of opioids-like peptides
T5158 N-Desmethylclozapine N-Desmethylclozapine is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 receptors, an agonist a...
T1407 (-)-Menthol L-Menthol is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local anesthetic proper...
T39284 EST73502 EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
T0783 Mianserin hydrochloride Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
T1197 Trimebutine maleate Trimebutine maleate is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate receptors ser...
TP2501 Difelikefalin acetate Difelikefalin acetate is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into the brain.
T5S2360 Corydaline 1. Corydaline, an isoquinoline alkaloid, is one of the major active constituents in a new prokinetic botanical agent. 2. Corydaline promotes gastric emptying and...
T2870 Matrine Matrine, an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
T3417 Amentoflavone Amentoflavone, as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for drug metabolism in t...
TP1941L1 Ac-RYYRWK-NH2 acetate Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.
T5S0581 Sec-O-Glucosylhamaudol Sec-O-glucosylhamaudol has anti-inflammatory effect through regulation of p38 Mitogen-Activated Protein Kinase in Lipopolysaccharide-stimulated RAW264.7 cell lin...
TP2052L CTOP acetate CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.
T21757 BRL 52537 hydrochloride BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury[1]. It is used for res...
TP2036 DPDPE DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
T21422 Methylnaltrexone bromide Methylnaltrexone, used in form of methylnaltrexone bromide, is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone acts to reve...
T2071 MCOPPB triHydrochloride MCOPPB trihydrochlride is a nociceptin receptor agonist.
T20435L Leuphasyl TFA Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway o...
T23306 Salvinorin A Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
T2388 Nalfurafine hydrochloride Nalfurafine(TRK-820) is an opioid κ-selective agonist; has been approved in Japan for treatment of itch in patients with chronic kidney disease.
T8992 BMS986188 BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.
T8991 BMS986187 BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
T8557 N-terminally acetylated Leu-enkephalin Leu-enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.N-terminally acetylated Leu-enkephalin is the N-terminally ace...
T8455 Spinorphin Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
T7665 [Leu5]-Enkephalin TFA(58822-25-6(free bas)) [Leu5]-Enkephalin is the most potent δ-receptor ago
T7613 β-Casomorphin, human β-Casomorphin, human(TFA) is an opioid receptor agonist.
T7639 Deltorphin 2 Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM)
T7637 Deltorphin I Deltorphin I(TFA) is an agonist of δ-opioid receptor.
T7173L [Leu5]-Enkephalin acetate(58822-25-6 free base) [Leu5]-Enkephalin acetate is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respecti...
T7218 Endomorphin 2 Endomorphins-2 (EM-2) could decrease both the frequency and amplitude of the sEPSC of the motoneurons in lamina IX, which was reversed by the MOR antagonist CTOP...
T7211 Tyr-Gly-Gly-Phe-Met-OH Tyr-Gly-Gly-Phe-Met-OH, is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.
T7576L β-Casomorphin, bovine TFA(72122-62-4(free base)) β-Casomorphin, bovine TFA is an opioid peptide isolated from casein peptone
T7576 β-Casomorphin, bovine β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
T7567L Adrenorphin 3TFA(88377-68-8(free base)) Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Nalfurafine
T41284
β-Endorphin (1-27) (human) acetate
T38193L
Deltorphin acetate
T20166L
Deltorphin acetate 是一种从青蛙 Phyllomedusa bicolor 的皮肤分泌物中获得的物质,对 δ-阿片受体具有高选择性和亲和力。
Sinomenine hydrochloride
T2921
Sinomenine hydrochloride is extracted from Sinomenium Acutum Rehderett Wilson.
Progesterone
T0478
Progesterone is the major progestational steroid that is secreted primarily by the CORPUS LUTEUM and the PLACENTA. Progesterone acts on the UTERUS, the MAMMARY G...
Mirtazapine
T0137
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
Asimadoline
T4633
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
[Leu5]-Enkephalin
T7173
[Leu5]-Enkephalin is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
(D-Ser2)-Leu-Enkephalin-Thr
T22752L
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.
Docusate sodium
T0929
Docusate is an orally available, over-the-counter laxative and stool softener used to treat or prevent constipation. Docusate has not been linked to serum enzyme...
Nociceptin (1-7) acetate
T23076L
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor. Nociceptin (1-7) combines with nociceptin reduces hyperalgesia and has a...
Ac-RYYRIK-NH2 acetate
TP1940L1
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial ag...
Loperamide hydrochloride
T0209
Loperamide Hydrochloride is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
b-Casomorphin (1-3) Acetate
T21660L
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
Sinomenine
T2726
Sinomenine is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
BMS-986122
T26869
BMS-986122 is a positive allosteric modulator of the μ-Opioid Receptor.
Dermorphin TFA
T7748
Dermorphin TFA is a new class of opioids-like peptides
N-Desmethylclozapine
T5158
N-Desmethylclozapine is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 receptors, an agonist a...
(-)-Menthol
T1407
L-Menthol is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local anesthetic proper...
EST73502
T39284
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
Mianserin hydrochloride
T0783
Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
Trimebutine maleate
T1197
Trimebutine maleate is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate receptors ser...
Difelikefalin acetate
TP2501
Difelikefalin acetate is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into the brain.
Corydaline
T5S2360
1. Corydaline, an isoquinoline alkaloid, is one of the major active constituents in a new prokinetic botanical agent. 2. Corydaline promotes gastric emptying and...
Matrine
T2870
Matrine, an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
Amentoflavone
T3417
Amentoflavone, as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for drug metabolism in t...
Ac-RYYRWK-NH2 acetate
TP1941L1
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.
Sec-O-Glucosylhamaudol
T5S0581
Sec-O-glucosylhamaudol has anti-inflammatory effect through regulation of p38 Mitogen-Activated Protein Kinase in Lipopolysaccharide-stimulated RAW264.7 cell lin...
CTOP acetate
TP2052L
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.
BRL 52537 hydrochloride
T21757
BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury[1]. It is used for res...
DPDPE
TP2036
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antino...
Methylnaltrexone bromide
T21422
Methylnaltrexone, used in form of methylnaltrexone bromide, is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone acts to rev...
MCOPPB triHydrochloride
T2071
MCOPPB trihydrochlride is a nociceptin receptor agonist.
Leuphasyl TFA
T20435L
Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway ...
Salvinorin A
T23306
Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
Nalfurafine hydrochloride
T2388
Nalfurafine(TRK-820) is an opioid κ-selective agonist; has been approved in Japan for treatment of itch in patients with chronic kidney disease.
BMS986188
T8992
BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.
BMS986187
T8991
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
N-terminally acetylated Leu-enkephalin
T8557
Leu-enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.N-terminally acetylated Leu-enkephalin is the N-terminally ace...
Spinorphin
T8455
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
T7665
[Leu5]-Enkephalin is the most potent δ-receptor ago
β-Casomorphin, human
T7613
β-Casomorphin, human(TFA) is an opioid receptor agonist.
Deltorphin 2
T7639
Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM)
Deltorphin I
T7637
Deltorphin I(TFA) is an agonist of δ-opioid receptor.
[Leu5]-Enkephalin acetate(58822-25-6 free base)
T7173L
[Leu5]-Enkephalin acetate is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respec...
Endomorphin 2
T7218
Endomorphins-2 (EM-2) could decrease both the frequency and amplitude of the sEPSC of the motoneurons in lamina IX, which was reversed by the MOR antagonist CTOP...
Tyr-Gly-Gly-Phe-Met-OH
T7211
Tyr-Gly-Gly-Phe-Met-OH, is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.
β-Casomorphin, bovine TFA(72122-62-4(free base))
T7576L
β-Casomorphin, bovine TFA is an opioid peptide isolated from casein peptone
β-Casomorphin, bovine
T7576
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
Adrenorphin 3TFA(88377-68-8(free base))
T7567L
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
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