T10821 |
Cirsiliol
|
34334-69-5
|
98%
|
|
Cirsiliol is a selective inhibitor of 5-lipoxygenase and a competitive low-affinity ligand of benzodiazepine receptors.
|
TN1871 |
Ligustroside
|
35897-92-8
|
98%
|
|
Ligustroside shows little antioxidant, and anti-inflammatory properties, it shows a significant inhibition effect on prostaglandin E2 (PGE2)-release. Ligustrosid...
|
T10719 |
CCT365623 hydrochloride
|
2126136-98-7
|
98%
|
|
CCT365623 hydrochloride is an orally active inhibitor of lysyl oxidase (LOX) (IC50: 0.89 μM). It suppresses EGFR (pY1068) and AKT phosphorylation driven by EGF.
|
T11196 |
Enazadrem
|
107361-33-1
|
98%
|
|
Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.
|
TN5020 |
(+/-)-Sigmoidin A
|
176046-04-1
|
98%
|
|
Sigmoidin A has moderate antioxidant, antimicrobial and anti-inflammatory activity.
|
TN4783 |
Picralinal
|
20045-06-1
|
98%
|
|
Picralinal has anti-inflammatory and analgesic effects.
|
TN4331 |
Isotachioside
|
31427-08-4
|
98%
|
|
Isotachioside has15-lipoxygenase (15-LO) inhibitory activities.
|
T10438 |
AZD 4407
|
166882-70-8
|
98%
|
|
AZD 4407 is a potent inhibitor of 5-lipoxygenase.
|
T34624 |
Setileuton
|
910656-27-8
|
98%
|
|
Setileuton is a specific 5-LOX inhibitor and can be used in research on asthma and atherosclerosis.
|
TN5174 |
Trichosanatine
|
169626-16-8
|
98%
|
|
Trichosanatine and squamosamide, as potential candidates as lead compounds for further study in drug development process with the PP2A- α protein. Trichosanatine...
|
TL0014 |
Pinusolide
|
31685-80-0
|
98%
|
|
Pinusolide is a platelet activating factor ( PAF) antagonist, it may prove of therapeutic value in the treatment of hypotension, it has antileukemic potential, a...
|
T4571 |
Balsalazide
|
80573-04-2
|
98%
|
|
Balsalazide is an anti-inflammatory compound used in the treatment of Inflammatory Bowel Disease.
|
T13764 |
Lycopodine
|
466-61-5
|
98%
|
|
Lycopodine inhibits proliferation of HeLa cells through induction of apoptosis via caspase-3 activation. Lycopodine, a pharmacologically important bioactive comp...
|
T10151 |
5-Lipoxygenase-In-1
|
125235-15-6
|
98%
|
|
5-Lipoxygenase-In-1 (compound example 4.10) is a 5-Lipoxygenase inhibitor extracted from patent EP 331232 A2.
|
T39986 |
LOX-IN-3 dihydrochloride
|
2409964-23-2
|
98%
|
|
LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX). LOX-IN-3 dihydrochloride inhibited bovine LOX (IC50<10 μM) and human LOXL2 (IC50<1 μM)activities...
|
T9878 |
Croconazole
|
77175-51-0
|
98%
|
|
Croconazole exhibited dose-dependent inhibitory activity on the 5-lipoxygenase (5-LOX) of neutrophils. Croconazole is an antimycotic agent. The IC50s for the syn...
|
T21838 |
1-Naphthyl 3,5-dinitrobenzoate
|
93261-39-3
|
98%
|
|
1-Naphthyl 3,5-dinitrobenzoate is an inhibitor of 5-LOX can be used in studies about inflammatory therapy.
|
T5759 |
S-(+)-Marmesin
|
13849-08-6
|
|
|
Marmesin is a coumarin originally isolated from the mature bark of A. marmelos,exhibiting COX-2/5-LOX dual inhibitory activity.
|
T22054 |
BW 755C
|
66000-40-6
|
|
|
BW 755C is a dual inhibitor of 5-lipoxygenase (5-LO) and cyclooxygenase (COX) pathways.
|
TN1255 |
3-O-Acetyl-11-hydroxy-beta-boswellic acid
|
146019-25-2
|
|
|
3-O-Acetyl-11-hydroxy-beta-boswellic acid is the precursor of 3-O-acetyl-9, 11-dehydro-beta-boswellic acid(a 5-lipoxygenase inhibitor ).
|