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Neurokinin receptor

The tachykinin receptor 1 (TACR1) also known as neurokinin 1 receptor (NK1R) or substance P receptor (SPR) is a G protein coupled receptor found in the central nervous system and peripheral nervous system. The endogenous ligand for this receptor is Substance P, although it has some affinity for other tachykinins.
Cat. No. Product name CAS No. Purity Chemical Structure
T10688 Casopitant mesylate 414910-30-8 98%
Casopitant mesylate (GW679769B) is a selective, brain permeable, and orally active antagonist of neurokinin 1 (NK1) receptor. It is a second in the class of anti...
T13329L Vofopitant dihydrochloride 168266-51-1 98%
Vofopitant dihydrochloride is a selective and orally available antagonist of tachykinin neurokinin 1(NK1) receptor (pKi: 9.5 and 10.6 in rat and human membranes ...
T7631 Eledoisin Related Peptide 2990-43-4 98%
Eledoisin Related Peptide(2TFA) is a tachykinin receptor ligand.
T19518 Physalaemin 2507-24-6 98%
Physalaemin is a non-mammalian tachykinin.
T35344 Maropitant citrate 359875-09-5 98%
TQ0087 NKP608 177707-12-9 98%
NKP608 is a selective and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50: 2.6 nM) and in vivo.
TP1177 Eledoisin 69-25-0 98%
Eledoisin is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin family of neuropeptides.
T10892 CS-003 Free base 191672-52-3 98%
CS-003 free base (CS-003) is a triple tachykinin receptor antagonist with high affinity for human (neurokinin) NK1, NK2 and NK3 receptors, with Ki values of 2.3 ...
T24697 R 396 129809-09-2 98%
R 396 is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.
T16406 Orvepitant maleate 579475-24-4 98%
Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant...
T7396 Substance P(1-7) 68060-49-1 98%
Substance P 1-7 is the major bioactive metabolite formed after proteolytic degradation of the tachykinin substance P (SP),with anti-inflammatory, anti-nociceptiv...
T7559 Neurokinin A(4-10) 97559-35-8 98%
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
T13329 Vofopitant 168266-90-8 98%
Vofopitant is a potent antagonist of the tachykinin NK1 receptor (pKis: 10.6, 9.5, and 9.8 for the human, rat, and ferret NK1 receptor, respectively).
T23316 SB 218795 174635-53-1 98%
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
T24446L MEN 10207 acetate 98%
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.
T17156 Tradipitant 622370-35-8 98%
Tradipitant is an antagonist of neurokinin-1.
T38144 Elinzanetant 929046-33-3 98%
Elinzanetant is a neurokinin receptors antagonist used for the research of Schizophrenia[1]. [1]. Alvaro, Giuseppe; Andreotti, Daniele; Belvedere, Sandro; Di Fab...
T24697L R 396 acetate 98%
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.
T20413L Spantide acetate T20413L 98%
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
T19518L Physalaemin acetate 98%
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
Casopitant mesylate
T10688
Casopitant mesylate (GW679769B) is a selective, brain permeable, and orally active antagonist of neurokinin 1 (NK1) receptor. It is a second in the class of anti...
Vofopitant dihydrochloride
T13329L
Vofopitant dihydrochloride is a selective and orally available antagonist of tachykinin neurokinin 1(NK1) receptor (pKi: 9.5 and 10.6 in rat and human membranes ...
Eledoisin Related Peptide
T7631
Eledoisin Related Peptide(2TFA) is a tachykinin receptor ligand.
Physalaemin
T19518
Physalaemin is a non-mammalian tachykinin.
Maropitant citrate
T35344
NKP608
TQ0087
NKP608 is a selective and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50: 2.6 nM) and in vivo.
Eledoisin
TP1177
Eledoisin is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin family of neuropeptides.
CS-003 Free base
T10892
CS-003 free base (CS-003) is a triple tachykinin receptor antagonist with high affinity for human (neurokinin) NK1, NK2 and NK3 receptors, with Ki values of 2.3 ...
R 396
T24697
R 396 is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.
Orvepitant maleate
T16406
Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant...
Substance P(1-7)
T7396
Substance P 1-7 is the major bioactive metabolite formed after proteolytic degradation of the tachykinin substance P (SP),with anti-inflammatory, anti-nociceptiv...
Neurokinin A(4-10)
T7559
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
Vofopitant
T13329
Vofopitant is a potent antagonist of the tachykinin NK1 receptor (pKis: 10.6, 9.5, and 9.8 for the human, rat, and ferret NK1 receptor, respectively).
SB 218795
T23316
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
MEN 10207 acetate
T24446L
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.
Tradipitant
T17156
Tradipitant is an antagonist of neurokinin-1.
Elinzanetant
T38144
Elinzanetant is a neurokinin receptors antagonist used for the research of Schizophrenia[1]. [1]. Alvaro, Giuseppe; Andreotti, Daniele; Belvedere, Sandro; Di Fab...
R 396 acetate
T24697L
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.
Spantide acetate
T20413L
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
Physalaemin acetate
T19518L
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
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