T10688 |
Casopitant mesylate
|
414910-30-8
|
98%
|
|
Casopitant mesylate (GW679769B) is a selective, brain permeable, and orally active antagonist of neurokinin 1 (NK1) receptor. It is a second in the class of anti...
|
T13329L |
Vofopitant dihydrochloride
|
168266-51-1
|
98%
|
|
Vofopitant dihydrochloride is a selective and orally available antagonist of tachykinin neurokinin 1(NK1) receptor (pKi: 9.5 and 10.6 in rat and human membranes ...
|
T7631 |
Eledoisin Related Peptide
|
2990-43-4
|
98%
|
|
Eledoisin Related Peptide(2TFA) is a tachykinin receptor ligand.
|
T19518 |
Physalaemin
|
2507-24-6
|
98%
|
|
Physalaemin is a non-mammalian tachykinin.
|
T35344 |
Maropitant citrate
|
359875-09-5
|
98%
|
|
|
TQ0087 |
NKP608
|
177707-12-9
|
98%
|
|
NKP608 is a selective and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50: 2.6 nM) and in vivo.
|
TP1177 |
Eledoisin
|
69-25-0
|
98%
|
|
Eledoisin is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin family of neuropeptides.
|
T10892 |
CS-003 Free base
|
191672-52-3
|
98%
|
|
CS-003 free base (CS-003) is a triple tachykinin receptor antagonist with high affinity for human (neurokinin) NK1, NK2 and NK3 receptors, with Ki values of 2.3 ...
|
T24697 |
R 396
|
129809-09-2
|
98%
|
|
R 396 is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.
|
T16406 |
Orvepitant maleate
|
579475-24-4
|
98%
|
|
Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant...
|
T7396 |
Substance P(1-7)
|
68060-49-1
|
98%
|
|
Substance P 1-7 is the major bioactive metabolite formed after proteolytic degradation of the tachykinin substance P (SP),with anti-inflammatory, anti-nociceptiv...
|
T7559 |
Neurokinin A(4-10)
|
97559-35-8
|
98%
|
|
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
|
T13329 |
Vofopitant
|
168266-90-8
|
98%
|
|
Vofopitant is a potent antagonist of the tachykinin NK1 receptor (pKis: 10.6, 9.5, and 9.8 for the human, rat, and ferret NK1 receptor, respectively).
|
T23316 |
SB 218795
|
174635-53-1
|
98%
|
|
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
|
T24446L |
MEN 10207 acetate
|
|
98%
|
|
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.
|
T17156 |
Tradipitant
|
622370-35-8
|
98%
|
|
Tradipitant is an antagonist of neurokinin-1.
|
T38144 |
Elinzanetant
|
929046-33-3
|
98%
|
|
Elinzanetant is a neurokinin receptors antagonist used for the research of Schizophrenia[1].
[1]. Alvaro, Giuseppe; Andreotti, Daniele; Belvedere, Sandro; Di Fab...
|
T24697L |
R 396 acetate
|
|
98%
|
|
R 396 acetate is an NK-2 Tachykinin Receptor
Antagonist.
|
T20413L |
Spantide acetate
|
T20413L
|
98%
|
|
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
|
T19518L |
Physalaemin acetate
|
|
98%
|
|
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
|