Moclobemide is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties. |
Modaline was a 2-methyl-3-piperidinopyrazine derivative found to inhibit monoamine oxidase (MAO) and showed a curative effect for the anti-depressant. Similar ...
Pargyline is a monoamine oxidase inhibitor with antihypertensive properties. |
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states. |
Ethaverine hydrochloride is a homologue of papaverine. |
Linezolid, the first of the oxazolidinone class, is a synthetic antibiotic used for the therapy of infections resulted from multi-resistant bacteria including ...
Allylthiourea, a metabolic inhibitor, specifically suppresses ammonia oxidation. |
Furazolidone, a nitrofuran derivative, inhibits AML1-ETO transformed cells with IC50 value of 12.7 μM. It is antibacterial and antiprotozoal activity, |
Iproniazid is a non-selective, irreversible monoamine oxidase inhibitor (MAOI). |
Senna is a herbal laxative that is found in garden rhubarb and green vegetables. |
||Tranylcypromine (2-PCPA) hydrochloride
Tranylcypromine Hydrochloride, a monoamine oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression. It...
Clorgyline hydrochloride, a white powder, is served as monoamine oxidase inhibitor. |
Rasagiline is an inhibitor of monamine oxidase used as adjunctive therapy in combination with levodopa and carbidopa in the management of Parkinsons disease. |
Nialamide is an MAO inhibitor that is used as an antidepressive agent. |
Raloxifene hydrochloride is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estrog...
Pargyline hydrochloride is an irreversible monoamine oxidase(MAO) inhibitor with antihypertensive properties. |
Hydralazine Hydrochloride is the hydrochloride salt of hydralazine, a phthalazine derivative with antihypertensive and potential antineoplastic activities. Hydr...
Harmine is an alkaloid isolated from seeds of Peganum harmala. |
Tedizolid is an Oxazolidinone Antibacterial. The mechanism of action of tedizolid is as a Breast Cancer Resistance Protein Inhibitor. |
Rosmarinic acid has shown to contain antioxidant,anti-inflammatory and antimicrobial activities. Possesses promising physiological actions related to cognitive ...
Paeonol is an active extraction from Paeonia suffruticosa. Paeonol inhibits MAO-A and MAO-B with IC50 of 54.6 μM and 42.5 μM, respectively. |
Tyramine is an indirect sympathomimetic that occurs naturally in cheese and other foods. Tyramine does not directly activate adrenergic receptors, but it can se...
TB5 is a potent, selective and reversible inhibitor of hMAO-B. |
Jatrorrhizine is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species. It was found to have antimicrobial and antifungal ac...
Safinamide Mesylate, a mesylate salt of Safinamide, can reversibly and specifically inhibit MAO-B (IC50: 98 nM), has 5918-fold selectivity against MAO-A. |
Isatin is an endogenous MAO inhibitor. |
Rasagiline Mesylate is a novel MAO-B inhibitor, which can treat idiopathic Parkinson's disease. |
1,4-Naphthoquinone was used as a potential inhibitor of monoamine oxidase and DNA topoisomerase activities. It was also used to inhibit the acetyltransferase...
Selegiline hydrochloride is a selective, reversible inhibitor of MAO-B (Ki = 0.091 μM) over MAO-A (Ki = 9.06 μM). Monoamine oxidase (MAO) inhibitors have util...
Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A). |
MD 69276 (Toloxatone) is a reversible monoamine oxidase A (MAOA) inhibitor. |
N-(2-Aminoethyl)-5-chlor-2-pyridincarbox is a reversible and selective mao-b inhibitor(Ki：7.9nM). |
(Z)-SU4312 is a inhibitor of MAO-B and NOS(IC50 value of 0.2 μM, 19.0μM,respectively). |
Purpurin was a reversible and competitive inhibitor of MAO-A with a Ki value of 0.422μM. it exhibits anti-angiogenic, antifungal, antibiotic, and antioxidative...
3,4-Dihydro-7-hydroxy-2(1H)-quinolinone (7- Hydroxy- 3, 4- dihydro- 2(1H) - quinolinone) is a weak MAO-A inhibitor(with an IC50 of 183 μM) . |
Salvigenin is a potent inhibitor of hMAO-A(monoamine oxidases),with neuroprotective effect and antitumor cytotoxic and immunomodulatory properties. |
LAZABEMIDE(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). |
Glycyrrhizic acid is a triterpenoid saponinl with anti-tumor and anti-diabetic activities. |
Tranylcypromine is an inhibitor of monoamine oxidase (MAO) and lysine-specific demethylase 1 (LSD1) with a rapid onset of activity. |
Osthenol shows antitumor-promoting activity, it also has antifungal and antibacterial activities. |
Glycyrrhisoflavone is a tyrosinase inhibitor, it also shows inhibitory effects on monoamine oxidase. |
Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is ...
4-Hydroxyderricin, the major active ingredients of Angelica keiskei Koidzumi, is a potent selective MAO-B inhibitor (IC50: 3.43 μM). It also mildly inhibits DB...
CR4056 is a selective inhibitor of human recombinant MAO-A (IC50: 202.7 nM) and a ligand of the imidazoline-2 receptor (I2R) (IC50: 596 nM). |
CX-157 is a reversible monoamine oxidase-A (MAO-A) inhibitor (EC50:19.3 ng/mL). |
Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A). |
MAO-IN-1 is an inhibitor of monoamine oxidase B (MAO B; IC50: 20 nM). |
||Ro 41-1049 hydrochloride
Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (Kd: 16.5 and 64.4 nM, respectively). |
Amiflamine is an inhibitor of reversible MAO-A. |
1-Methyl-2-undecyl-4(1H)-quinolone, and dihydroevocarpine should also be served as the chemical markers together with evodiamine for the quality control of Evod...
2'-O-Methylperlatolic acid and confluentic acid are monoamine oxidase B inhibitors in a Brazilian plant, Himatanthus sucuuba. |
5-Hydroxy-1-methoxyxanthone, 1,5-dihydroxyxanthone and 6-deoxyjacareubin are all antifungal against Cladosporium cucumerinum, while they show differing degrees ...
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. |
8alpha-Tigloyloxyhirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. 8alpha-Tigloyloxyhirsutinolide 13-O-acetate has...
Cudraflavone B has anti-proliferative activity, mouse brain monoamine oxidase (MAO) inhibitory effects, apoptotic actions in human gastric carcinoma cells and m...
Echitovenidine shows monoamine oxidase inhibitor activity. |
Glicoricone acts as a partial estrogen antagonist. Glicoricone inhibited the monoamine oxidase with the IC50 values of 6.0 x 10(-5)-1.4 x 10(-4) M. |