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Estrogen Receptor/ERR

The ERRs are orphan nuclear receptors, meaning the identity of their endogenous ligand has yet to be unambiguously determined. They are named because of sequence homology with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones.There are three human estrogen related receptors:ERRα,ERRβand ERRγ .
Cat. No. Product name CAS No. Purity Chemical Structure
T20419 Raloxifene 84449-90-1 98%
Raloxifene is a selective oestrogen receptor modulator. It has effects on bone and breast cancer and cardiovascular disease risk.
T11237L Camizestrant TFA T11237L 98%
Camizestrant TFA is a potent and orally active antagonist of estrogen receptor (ER).
T3645 Endoxifen E-isomer hydrochloride 1197194-61-8 98%
Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
T13674 Elacestrant 722533-56-4 98%
Elacestrant with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
T11237 Camizestrant 2222844-89-3 98%
Camizestrant is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
T6404 Bazedoxifene hydrochloride 198480-56-7 98%
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
T6827 Endoxifen Z-isomer hydrochloride 1032008-74-4 98%
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
T11098 Droloxifene 82413-20-5 98%
Droloxifene, a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells....
T36857L Premarin 481-97-0 98%
Premarin is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.
TN1052 Lindleyin 59282-56-3 98%
Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by the physiological estrogens.
T12654 (Rac)-Acolbifene 151533-34-5 98%
(Rac)-Acolbifene is the racemic form of Acolbifene. Acolbifene is a estrogen receptor antagonist. (Rac)-Acolbifene exhibits anti-estrogenic and estrogenic activi...
T10239 Acolbifene 182167-02-8 98%
Acolbifene is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifen...
T21897L MPP hydrochloride 98%
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
T20625 Prochloraz 67747-09-5 98%
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
T7389 G15 1161002-05-6
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
T6533 Hexestrol 84-16-2 100%
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
T1579 Mestranol 72-33-3 100%
Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
T39710 ARV-471 2229711-68-4 97.15%
ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
T2882 Genistin 529-59-9 97.65%
Genistin is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anti...
T15788 LSZ-102 2135600-76-7 97.84%
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
Raloxifene
T20419
Raloxifene is a selective oestrogen receptor modulator. It has effects on bone and breast cancer and cardiovascular disease risk.
Camizestrant TFA
T11237L
Camizestrant TFA is a potent and orally active antagonist of estrogen receptor (ER).
Endoxifen E-isomer hydrochloride
T3645
Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
Elacestrant
T13674
Elacestrant with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
Camizestrant
T11237
Camizestrant is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
Bazedoxifene hydrochloride
T6404
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
Endoxifen Z-isomer hydrochloride
T6827
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
Droloxifene
T11098
Droloxifene, a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells....
Premarin
T36857L
Premarin is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.
Lindleyin
TN1052
Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by the physiological estrogens.
(Rac)-Acolbifene
T12654
(Rac)-Acolbifene is the racemic form of Acolbifene. Acolbifene is a estrogen receptor antagonist. (Rac)-Acolbifene exhibits anti-estrogenic and estrogenic activi...
Acolbifene
T10239
Acolbifene is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifen...
MPP hydrochloride
T21897L
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
Prochloraz
T20625
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
G15
T7389
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
Hexestrol
T6533
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
Mestranol
T1579
Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
ARV-471
T39710
ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
Genistin
T2882
Genistin is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anti...
LSZ-102
T15788
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
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