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Estrogen Receptor/ERR

The ERRs are orphan nuclear receptors, meaning the identity of their endogenous ligand has yet to be unambiguously determined. They are named because of sequence homology with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones.There are three human estrogen related receptors:ERRα,ERRβand ERRγ .
Cat. No. Product name CAS No. Purity Chemical Structure
T22794 G36 1392487-51-2 98%
G36 is a cell-permeable non-steroidal antagonist of GPER. G36 inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 (IC50 = 112 and 165 n...
T11237 Camizestrant 2222844-89-3 98%
Camizestrant is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
T11098 Droloxifene 82413-20-5 98%
Droloxifene, a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells....
T11237L Camizestrant TFA T11237L 98%
Camizestrant TFA is a potent and orally active antagonist of estrogen receptor (ER).
T60664 Atamestane 96301-34-7 98%
Atamestane is a competitive, irreversible inhibitor of estrogen biosynthesis, a specific aromatase inhibitor that selectively blocks estrogen biosynthesis result...
T11236 Giredestrant tartrate 2407529-33-1 98%
Giredestrant tartrate is a novel, orally active, selective and effective non-steroidal estrogen receptor antagonist. Giredestrant tartrate strongly binds to ER, ...
T9455 4-hydroxyestrone-4-methyl ether 58562-33-7 98%
4-hydroxyestrone-4-methyl ether is the methylation of 4-OHE1, which is catalyzed by COMT.
T6404 Bazedoxifene hydrochloride 198480-56-7 98%
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
T6827 Endoxifen Z-isomer hydrochloride 1032008-74-4 98%
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
TN1567 Delphinidin chloride 528-53-0 98%
Delphinidin chloride, a natural plant pigment found in berries and red wine, is a precursor of certain anthocyanins. Delphinidin chloride induces the release of ...
TN3084 5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone 1353676-65-9 98%
5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone showed strong anti-proliferation effect on ER-positive breast cancer MCF-7 cells in vitro, with an IC50 val...
T9454 4-Hydroxyestrone 3131-23-5 98%
4-Hydroxyestrone, an endogenous estrogen metabolite, can strongly protect neuronal cells against oxidative damage.
T9997 GLL 398 2077980-80-2 98%
GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.
T0760 Cholesterol 57-88-5 98%
Cholesterol is the primary sterol in mammals. The significance of Cholesterol is becoming more appreciated in fundamental cellular processes.
T6306 Erteberel 533884-09-2 98%
LY500307 is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.
T2146 Fulvestrant 129453-61-8 98%
Fulvestrant is a potent Estrogen Receptor antagonist (IC50: 9.4 nM).
T3385 Gypenoside XVII 80321-69-3 98%
Gypenoside XVII confers protection against Aβ25-35-induced neurotoxicity through estrogen receptor-dependent activation of PI3K/Akt pathways, activation of Nrf2/...
T0384 Estradiol benzoate 50-50-0 98%
Estradiol Benzoate is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics...
TN1148 Isopsoralenoside 905954-18-9 98%
Isopsoralenoside shows estrogen-like, osteoblastic proliferation accelerating, antitumor, and antibacterial effects.
T21387L Nafoxidine 1845-11-0 98%
Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.
G36
T22794
G36 is a cell-permeable non-steroidal antagonist of GPER. G36 inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 (IC50 = 112 and 165 n...
Camizestrant
T11237
Camizestrant is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
Droloxifene
T11098
Droloxifene, a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells....
Camizestrant TFA
T11237L
Camizestrant TFA is a potent and orally active antagonist of estrogen receptor (ER).
Atamestane
T60664
Atamestane is a competitive, irreversible inhibitor of estrogen biosynthesis, a specific aromatase inhibitor that selectively blocks estrogen biosynthesis result...
Giredestrant tartrate
T11236
Giredestrant tartrate is a novel, orally active, selective and effective non-steroidal estrogen receptor antagonist. Giredestrant tartrate strongly binds to ER, ...
4-hydroxyestrone-4-methyl ether
T9455
4-hydroxyestrone-4-methyl ether is the methylation of 4-OHE1, which is catalyzed by COMT.
Bazedoxifene hydrochloride
T6404
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
Endoxifen Z-isomer hydrochloride
T6827
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
Delphinidin chloride
TN1567
Delphinidin chloride, a natural plant pigment found in berries and red wine, is a precursor of certain anthocyanins. Delphinidin chloride induces the release of ...
5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone
TN3084
5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone showed strong anti-proliferation effect on ER-positive breast cancer MCF-7 cells in vitro, with an IC50 val...
4-Hydroxyestrone
T9454
4-Hydroxyestrone, an endogenous estrogen metabolite, can strongly protect neuronal cells against oxidative damage.
GLL 398
T9997
GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.
Cholesterol
T0760
Cholesterol is the primary sterol in mammals. The significance of Cholesterol is becoming more appreciated in fundamental cellular processes.
Erteberel
T6306
LY500307 is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.
Fulvestrant
T2146
Fulvestrant is a potent Estrogen Receptor antagonist (IC50: 9.4 nM).
Gypenoside XVII
T3385
Gypenoside XVII confers protection against Aβ25-35-induced neurotoxicity through estrogen receptor-dependent activation of PI3K/Akt pathways, activation of Nrf2/...
Estradiol benzoate
T0384
Estradiol Benzoate is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics...
Isopsoralenoside
TN1148
Isopsoralenoside shows estrogen-like, osteoblastic proliferation accelerating, antitumor, and antibacterial effects.
Nafoxidine
T21387L
Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.
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