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Androgen Receptor

The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding any of the androgenic hormones, including testosterone and dihydrotestosterone in the cytoplasm and then translocating into the nucleus.
Cat. No. Product name CAS No. Purity Chemical Structure
T19449 N-desmethyl Enzalutamide D6 T19449 98%
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
TMA1012 Ganoderiol F 114567-47-4 98%
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
T14843 Bifluranol 34633-34-6 98%
Bifluranol is an anti-androgen.
T14675 BMS-564929 627530-84-1 98%
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
TN4774 Physalin A 23027-91-0 98%
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate canc...
T10946 D4-abiraterone 154229-21-7 98%
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abira...
T15816 LY341495 201943-63-7 98%
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
T15749 LGD-2226 328947-93-9 98%
LGD-2226 is a selective and orally active androgen receptor modulator (EC50: 0.2 nM, Ki: 1.5 nM for the human androgen receptor). LGD-2226 can be used for muscle...
TN1061 Ganoderol B 104700-96-1 98%
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
TN1663 Ganoderic acid DM 173075-45-1 98%
Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 ...
T20625 Prochloraz 67747-09-5 98%
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
TN1067 Galloylpaeoniflorin 122965-41-7 98%
6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
T39695 ARD-2128 2222111-87-5 98%
ARD-2128 is a highly potent, orally bioavailable PROTAC degrader of androgen receptor (AR). ARD-2128 effectively reduces AR protein, suppresses AR-regulated gene...
T8860 DSRM-3716 58142-99-7 98%
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
T24943 VPC-14228 19983-28-9 98%
VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.
T67818 BMS-641988 98%
BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
T2991 3,3'-Diindolylmethane 1968-05-4 98%
DIM (3, 3'-diindolylmethane), a small molecule compound, is a proposed Y preventive agent.
T8117 Metenolone acetate 434-05-9 98%
Methenolone acetate is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow failure.
T75129 Luxdegalutamide 2750830-09-0 98%
Luxdegalutamide is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades the wild-type and...
T6400 AZD3514 1240299-33-5 98%
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.
N-desmethyl Enzalutamide D6
T19449
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
Ganoderiol F
TMA1012
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
Bifluranol
T14843
Bifluranol is an anti-androgen.
BMS-564929
T14675
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
Physalin A
TN4774
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate canc...
D4-abiraterone
T10946
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abira...
LY341495
T15816
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
LGD-2226
T15749
LGD-2226 is a selective and orally active androgen receptor modulator (EC50: 0.2 nM, Ki: 1.5 nM for the human androgen receptor). LGD-2226 can be used for muscle...
Ganoderol B
TN1061
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
Ganoderic acid DM
TN1663
Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 ...
Prochloraz
T20625
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
Galloylpaeoniflorin
TN1067
6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
ARD-2128
T39695
ARD-2128 is a highly potent, orally bioavailable PROTAC degrader of androgen receptor (AR). ARD-2128 effectively reduces AR protein, suppresses AR-regulated gene...
DSRM-3716
T8860
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
VPC-14228
T24943
VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.
BMS-641988
T67818
BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
3,3'-Diindolylmethane
T2991
DIM (3, 3'-diindolylmethane), a small molecule compound, is a proposed Y preventive agent.
Metenolone acetate
T8117
Methenolone acetate is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow failure.
Luxdegalutamide
T75129
Luxdegalutamide is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades the wild-type and...
AZD3514
T6400
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.
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