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Androgen Receptor

The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding any of the androgenic hormones, including testosterone and dihydrotestosterone in the cytoplasm and then translocating into the nucleus.
Cat No. product name
T21740 RD162 RD162 是一种与雄激素受体 (AR) 特异性结合的非甾体抗雄激素 (NSAA)。
T2321 Protodioscin Protodioscin is a major steroidal saponin in dioscoreae rhizome, with anti-hyperlipidemia, anti-cancer properties.
T7440 P,p'-DDE 4,4'-DDE is a metabolite and degradation product of the organochlorine pesticide DDT
T3137 Boldenone Undecylenate Boldenone undecylenate is a synthetic steroid.
T8117 Metenolone acetate Methenolone acetate is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow failure.
T0380 Bicalutamide Bicalutamide, a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the receptor bind...
T15445 Proxalutamide Proxalutamide is a potent antagonist of the androgen receptor (AR).
T9752 3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile 3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.
T9035 Testosterone undecanoate Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.
T8860 DSRM-3716 Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
T19470 Nandrolone propionate Nandrolone propionate is an anabolic steroid action primarily consisting of androgenic and nitrogen-retentive properties.
T29111 VPC-13566 VPC-13566 is a BF3-specific small molecule, which effectively inhibited AR transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-1356...
T6829 EPI-001 EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ~6 μM and a selective PPAR-gamma modulator.
T20761 RU 59063 RU 59063 is a prototype of high-affinity nonsteroidal androgen receptor (AR) ligands.
T2207 Adrenosterone Adrenosterone is a steroid hormone isolated from the adrenal cortex.
T5100 DJ-V-159 DJ-V159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A).
T6002 Enzalutamide Enzalutamide (MDV 3100) is a non-steroidal androgen receptor (AR) antagonist (IC50: 36 nM in LNCaP prostate cells).
T20789 S-23 S-23 is a novel nonsteroidal agonist and has tissue selective.
T1541 Drospirenone Drospirenone is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T2991 3,3'-Diindolylmethane DIM (3, 3'-diindolylmethane), a small molecule compound, is a proposed Y preventive agent.
T6889 MI-136 MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.
TN1067 Galloylpaeoniflorin 6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
T20625 Prochloraz Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
T12146 N-Desmethyl-Apalutamide N-Desmethyl Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
T14116 ACP-105 ACP-105 is a selective amd potent androgen receptor modulator (SARM). For AR wild type and T877A mutant, the pEC50s values are 9.0 and 9.3 , respectively.
T26539 AC-262536 AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.
T1596 Chlormadinone acetate Chlormadinone acetate is an orally active synthetic progestational hormone used often in combinations as an oral contraceptive.
T1261 Medroxyprogesterone Acetate Medroxyprogesterone acetate is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally...
T9179 CLP-3094 CLP-3094 is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selecti...
T2895 Lupeol Lupeol is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
T0476 Spironolactone Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
T8217 Enzalutamide carboxylic acid Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
T12928 SK33 SK33 is a potent and tissue selective anti-androgen,and is a trifluoromethylated enobosarm analog, SK33 reduces androgen receptor (AR) transcriptional activity.
T19449 N-desmethyl Enzalutamide D6 N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
T19450 N-desmethyl Enzalutamide N-desmethyl Enzalutamide is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and sec...
T2408 Ostarine Ostarine is a non-steroidal agent with anabolic activity. Selective androgen receptor modulator (SARM) GTx-024 is designed to work like testosterone, thus promot...
T2339 Apalutamide Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
T22263 Bavdegalutamide ARV-110 is an oral degrader of androgen receptor PROTAC for prostate cancer treatment.
T2236 RU 58841 RU 58841 is a specific androgen receptor antagonist or anti-androgen; RU 58841 has a significant effect on hair regrowth.
T7690 2-hydroxy Flutamide 2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer
T7358 YK11 YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when use...
T9246 JNJ-63576253 JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).
TCS1372 Atraric acid Atraric acid derivatives as a new chemical lead structure for novel therapeutic compounds as AR antagonists, that can be used for prophylaxis or treatment of pro...
T8933 JNJ-63576253 free base JNJ-63576253 is a potent and orally active full antagonist of androgen receptor (AR), with IC50s of 37 and 54 nM for F877L mutant AR and wild-type AR in LNCaP ce...
T8709 Nandrolone phenylpropionate Nandrolone phenpropionate is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis
T8592 CTK8A3536 CTK8A3536 is an inhibitor of Androgen receptor.
TMA1012 Ganoderiol F Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
TN1061 Ganoderol B Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
TN1370 Allura Red AC Allura Red AC and amaranth are very important food azo dyes used in food, drug, paper, cosmetic and textile industries.
TN2245 Sunset Yellow FCF Sunset yellow FCF and Brilliant Blue FCF are used as colorant food additives in many food products, they can have cytotoxic and genotoxic potential, it care must...
RD162
T21740
RD162 是一种与雄激素受体 (AR) 特异性结合的非甾体抗雄激素 (NSAA)。
Protodioscin
T2321
Protodioscin is a major steroidal saponin in dioscoreae rhizome, with anti-hyperlipidemia, anti-cancer properties.
p,p'-DDE
T7440
4,4'-DDE is a metabolite and degradation product of the organochlorine pesticide DDT
Boldenone Undecylenate
T3137
Boldenone undecylenate is a synthetic steroid.
Metenolone acetate
T8117
Methenolone acetate is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow failure.
Bicalutamide
T0380
Bicalutamide, a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the receptor bind...
Proxalutamide
T15445
Proxalutamide is a potent antagonist of the androgen receptor (AR).
3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
T9752
3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.
Testosterone undecanoate
T9035
Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.
DSRM-3716
T8860
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
Nandrolone propionate
T19470
Nandrolone propionate is an anabolic steroid action primarily consisting of androgenic and nitrogen-retentive properties.
VPC-13566
T29111
VPC-13566 is a BF3-specific small molecule, which effectively inhibited AR transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-1356...
EPI-001
T6829
EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ~6 μM and a selective PPAR-gamma modulator.
RU 59063
T20761
RU 59063 is a prototype of high-affinity nonsteroidal androgen receptor (AR) ligands.
Adrenosterone
T2207
Adrenosterone is a steroid hormone isolated from the adrenal cortex.
DJ-V-159
T5100
DJ-V159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A).
Enzalutamide
T6002
Enzalutamide (MDV 3100) is a non-steroidal androgen receptor (AR) antagonist (IC50: 36 nM in LNCaP prostate cells).
S-23
T20789
S-23 is a novel nonsteroidal agonist and has tissue selective.
Drospirenone
T1541
Drospirenone is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
3,3'-Diindolylmethane
T2991
DIM (3, 3'-diindolylmethane), a small molecule compound, is a proposed Y preventive agent.
MI-136
T6889
MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.
Galloylpaeoniflorin
TN1067
6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
Prochloraz
T20625
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
N-Desmethyl-Apalutamide
T12146
N-Desmethyl Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
ACP-105
T14116
ACP-105 is a selective amd potent androgen receptor modulator (SARM). For AR wild type and T877A mutant, the pEC50s values are 9.0 and 9.3 , respectively.
AC-262536
T26539
AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.
Chlormadinone acetate
T1596
Chlormadinone acetate is an orally active synthetic progestational hormone used often in combinations as an oral contraceptive.
Medroxyprogesterone Acetate
T1261
Medroxyprogesterone acetate is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally...
CLP-3094
T9179
CLP-3094 is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a select...
Lupeol
T2895
Lupeol is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
Spironolactone
T0476
Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
Enzalutamide carboxylic acid
T8217
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
SK33
T12928
SK33 is a potent and tissue selective anti-androgen,and is a trifluoromethylated enobosarm analog, SK33 reduces androgen receptor (AR) transcriptional activity.
N-desmethyl Enzalutamide D6
T19449
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
N-desmethyl Enzalutamide
T19450
N-desmethyl Enzalutamide is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and sec...
Ostarine
T2408
Ostarine is a non-steroidal agent with anabolic activity. Selective androgen receptor modulator (SARM) GTx-024 is designed to work like testosterone, thus promot...
Apalutamide
T2339
Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
Bavdegalutamide
T22263
ARV-110 is an oral degrader of androgen receptor PROTAC for prostate cancer treatment.
RU 58841
T2236
RU 58841 is a specific androgen receptor antagonist or anti-androgen; RU 58841 has a significant effect on hair regrowth.
2-hydroxy Flutamide
T7690
2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer
YK11
T7358
YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when use...
JNJ-63576253
T9246
JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).
Atraric acid
TCS1372
Atraric acid derivatives as a new chemical lead structure for novel therapeutic compounds as AR antagonists, that can be used for prophylaxis or treatment of pro...
JNJ-63576253 free base
T8933
JNJ-63576253 is a potent and orally active full antagonist of androgen receptor (AR), with IC50s of 37 and 54 nM for F877L mutant AR and wild-type AR in LNCaP ce...
Nandrolone phenylpropionate
T8709
Nandrolone phenpropionate is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis
CTK8A3536
T8592
CTK8A3536 is an inhibitor of Androgen receptor.
Ganoderiol F
TMA1012
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
Ganoderol B
TN1061
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prost...
Allura Red AC
TN1370
Allura Red AC and amaranth are very important food azo dyes used in food, drug, paper, cosmetic and textile industries.
Sunset Yellow FCF
TN2245
Sunset yellow FCF and Brilliant Blue FCF are used as colorant food additives in many food products, they can have cytotoxic and genotoxic potential, it care must...
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