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Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T23535	Xanthine amine congener	96865-92-8	99.7%
T23535	Xanthine amine congener is an Adenosine receptor antagonist.
T37793	A2B receptor antagonist 2	784-90-7	100%
T37793	A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T11762	Kira8 Hydrochloride	2250019-92-0	98%
T11762	Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
T78084	PSB 0777 ammonium hydrate		98%
T78084	PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for hu...
T79027	A1/A3 AR antagonist 3	2665804-57-7	98%
T79027	A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in the...
T79372	A3AR agonist 1		98%
T79372	A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective conc...
T79373	A3AR agonist 2		98%
T79373	Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. Thi...
T13008	ST3932	1246018-21-2	98%
T13008	ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
T72626	A2AR-antagonist-1	2922920-71-4	98%
T72626	A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability...
T16281	Nelonicline	1026134-63-3	98%
T16281	Nelonicline is a selective agonist of neuronal nicotinic receptors.
TQ0136	GR79236	124555-18-6	98%
TQ0136	GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T16158	PF-02575799	863491-70-7	98%
T16158	PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
T8598	CHEMBL241987	109740-09-2	99.98%
T8598	CHEMBL241987 targets the Adenosine receptor A3 (human)
T12161	N6-Ethyladenosine	14357-08-5	99.98%
T12161	N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
T6745	5-Iodotubercidin	24386-93-4	99.98%
T6745	5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinas...
T2205	Acefylline	652-37-9	99.95%
T2205	Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhyd...
T23336	SCH442416	316173-57-6	99.95%
T23336	SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.0...
T1681	Aminophylline	317-34-0	99.94%
T1681	Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.
T12163	N6-(2-Phenylethyl)adenosine	20125-39-7	99.94%
T12163	N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for ra...
T22744	DPCPX	102146-07-6	99.93%
T22744	DPCPX (PD 116948) is an A1 adenosine receptor antagonist