T16158 |
PF-02575799
|
863491-70-7
|
98%
|
|
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
|
T27509 |
GW-493838
|
253124-46-8
|
98%
|
|
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or...
|
T22031 |
ANR 94
|
634924-89-3
|
98%
|
|
ANR94 is a potent and selective adenosine A 2A receptor (AA 2A R) antagonist with an K i of 46 nM for hAA 2A R. ANR94 has the potential for the research of Parki...
|
T11762 |
Kira8 Hydrochloride
|
2250019-92-0
|
98%
|
|
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
|
TQ0136 |
GR79236
|
124555-18-6
|
98%
|
|
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
|
T13008 |
ST3932
|
1246018-21-2
|
98%
|
|
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
|
T16281 |
Nelonicline
|
1026134-63-3
|
98%
|
|
Nelonicline is a selective agonist of neuronal nicotinic receptors.
|
T12163 |
N6-(2-Phenylethyl)adenosine
|
20125-39-7
|
98%
|
|
N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
|
T21620 |
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine
|
133240-06-9
|
98%
|
|
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine is an adenosine receptor antagonist.
|
T28861 |
ST-1535
|
496955-42-1
|
98%
|
|
ST 1535 is a potent and orally active antagonist of A2A adenosine receptor with antiparkinsonian activity and antitremorigenic effects. ST 1535 exhibits the pote...
|
T15418 |
GS-6201
|
752222-83-6
|
98%
|
|
GS-6201 is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors (Ki: 22 nM). GS-62...
|
T37792 |
A2A receptor antagonist 1
|
443103-97-7
|
98%
|
|
A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
|
T37793 |
A2B receptor antagonist 2
|
784-90-7
|
98%
|
|
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
|
T27629 |
ISAM-140
|
932191-62-3
|
98%
|
|
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
|
T23016 |
MRS1220
|
183721-15-5
|
98%
|
|
MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
|
T16140 |
MRS 1754
|
264622-58-4
|
98%
|
|
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
|
T23201 |
PSB 1115
|
152529-79-8
|
98%
|
|
human A2B adenosine receptor antagonist
|
T29112 |
VPC171
|
1018830-99-3
|
98%
|
|
VPC171 is a positive allosteric modulator (PAM) of the adenosine A1 receptor (A1R).
|
T8613 |
1-Ethyl-6-aminouracil
|
41862-09-3
|
|
|
1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosi...
|
T14078 |
AB928
|
2239273-34-6
|
100%
|
|
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
|