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Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.
Cat. No. Product name CAS No. Purity Chemical Structure
T16158 PF-02575799 863491-70-7 98%
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
T27509 GW-493838 253124-46-8 98%
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or...
T22031 ANR 94 634924-89-3 98%
ANR94 is a potent and selective adenosine A 2A receptor (AA 2A R) antagonist with an K i of 46 nM for hAA 2A R. ANR94 has the potential for the research of Parki...
T11762 Kira8 Hydrochloride 2250019-92-0 98%
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
TQ0136 GR79236 124555-18-6 98%
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T13008 ST3932 1246018-21-2 98%
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
T16281 Nelonicline 1026134-63-3 98%
Nelonicline is a selective agonist of neuronal nicotinic receptors.
T12163 N6-(2-Phenylethyl)adenosine 20125-39-7 98%
N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
T21620 2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine 133240-06-9 98%
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine is an adenosine receptor antagonist.
T28861 ST-1535 496955-42-1 98%
ST 1535 is a potent and orally active antagonist of A2A adenosine receptor with antiparkinsonian activity and antitremorigenic effects. ST 1535 exhibits the pote...
T15418 GS-6201 752222-83-6 98%
GS-6201 is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors (Ki: 22 nM). GS-62...
T37792 A2A receptor antagonist 1 443103-97-7 98%
A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
T37793 A2B receptor antagonist 2 784-90-7 98%
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T27629 ISAM-140 932191-62-3 98%
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
T23016 MRS1220 183721-15-5 98%
MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
T16140 MRS 1754 264622-58-4 98%
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
T23201 PSB 1115 152529-79-8 98%
human A2B adenosine receptor antagonist
T29112 VPC171 1018830-99-3 98%
VPC171 is a positive allosteric modulator (PAM) of the adenosine A1 receptor (A1R).
T8613 1-Ethyl-6-aminouracil 41862-09-3
1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosi...
T14078 AB928 2239273-34-6 100%
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
PF-02575799
T16158
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
GW-493838
T27509
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or...
ANR 94
T22031
ANR94 is a potent and selective adenosine A 2A receptor (AA 2A R) antagonist with an K i of 46 nM for hAA 2A R. ANR94 has the potential for the research of Parki...
Kira8 Hydrochloride
T11762
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
GR79236
TQ0136
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
ST3932
T13008
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
Nelonicline
T16281
Nelonicline is a selective agonist of neuronal nicotinic receptors.
N6-(2-Phenylethyl)adenosine
T12163
N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine
T21620
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine is an adenosine receptor antagonist.
ST-1535
T28861
ST 1535 is a potent and orally active antagonist of A2A adenosine receptor with antiparkinsonian activity and antitremorigenic effects. ST 1535 exhibits the pote...
GS-6201
T15418
GS-6201 is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors (Ki: 22 nM). GS-62...
A2A receptor antagonist 1
T37792
A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
A2B receptor antagonist 2
T37793
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
ISAM-140
T27629
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
MRS1220
T23016
MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
MRS 1754
T16140
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
PSB 1115
T23201
human A2B adenosine receptor antagonist
VPC171
T29112
VPC171 is a positive allosteric modulator (PAM) of the adenosine A1 receptor (A1R).
1-Ethyl-6-aminouracil
T8613
1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosi...
AB928
T14078
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
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