TN2641 |
15-Methoxypinusolidic acid
|
769928-72-5
|
98%
|
|
15-Methoxypinusolidic acid has anti-inflammatory effects, it inhibits LPS-induced iNOS expression and NO production, independent on MAPK and NF-kappaB. 15-Methox...
|
T8447 |
Ro 8-4304
|
195988-65-9
|
98%
|
|
Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM
|
TN5263 |
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one
|
569-83-5
|
98%
|
|
Xanthohumol, prenylchacone flavonoid, is a natural product with multi-biofunctions purified from Hops Humulus lupulus. Xanthohumol is effective against HIV-1 and...
|
T16473 |
Perzinfotel
|
144912-63-0
|
98%
|
|
Perzinfotel displays high affinity (IC50=30 nM) for the glutamate site. Perzinfotel is an effective, selective, and competitive NMDA receptor antagonist with neu...
|
T22654 |
Selfotel
|
110347-85-8
|
98%
|
|
NMDA receptor antagonist
|
T7778 |
Glypromate
|
32302-76-4
|
98%
|
|
Glypromate is a neuroprotective agent, is a weak NMDA receptor agonist
|
T16332 |
NKH477
|
138605-00-2
|
98%
|
|
NKH477 is a novel water-soluble forskolin derivative that improves cardiac failure mainly through its beneficial effects on diastolic cardiac function. NKH477 sh...
|
T3407 |
Rapastinel
|
117928-94-6
|
98%
|
|
Rapastinel (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.
|
T60237 |
L-Cysteine S-sulfate
|
1637-71-4
|
98%
|
|
L-Cysteine S-sulfate is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist. L-Cysteine S-sulfate is the substrate for cystine lyase [1].
|
T22900 |
L-701252
|
151057-13-5
|
98%
|
|
L-701252 is a potent antagonist of glycine site NMDA receptor with an IC50 of 420 nM. L-701252 provides a small degree of neuroprotection in global cerebral isch...
|
T22517 |
5,7-Dichlorokynurenic acid
|
131123-76-7
|
98%
|
|
NMDA receptor antagonist
|
T12234 |
NMDA-IN-1
|
700878-19-9
|
98%
|
|
NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).
|
T25196 |
BZAD01
|
305339-41-7
|
98%
|
|
BZAD01 is an antagonist of GluN2B subtype-selective NMDA.
|
T3407L |
Rapastinel acetate
|
491872-39-0
|
98%
|
|
Rapastinel acetate is a modulator of N-methyl-D-aspartate (NMDA) receptor and a partial agonist of glycine site long-lasting antidepressant effects.
|
TQ0279 |
Ibotenic acid
|
2552-55-8
|
98%
|
|
Ibotenic acid has agonist activity at both the NMDA and trans-ACPD or metabotropic quisqualate receptors.
|
T20571 |
Cis-PDA
|
46026-75-9
|
98%
|
|
cis-PDA, a general ionotropic receptor antagonist, acts by blocking NMDA, AMPA, and kainate mediated responses. It also acts as a partial NMDA receptor agonist.
|
T22733 |
DL-AP5
|
76326-31-3
|
|
|
NMDA antagonist
|
T4096 |
Quinolinic acid
|
89-00-9
|
|
|
Quinolinic acid is an endogenous N-methyl-D-aspartate (NMDA) receptor agonist synthesized from L-tryptophan via the kynurenine pathway.
|
T22542 |
1-Aminocyclobutanecarboxylic acid
|
22264-50-2
|
|
|
1-Aminocyclobutanecarboxylic acid is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].
|
T7867 |
Flutriafol
|
76674-21-0
|
100%
|
|
Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist
|