Search Result

Search Results for " transferase "

Targets

Histone Methyltransferase DNA Methyltransferase Histone Acetyltransferase Methionine Adenosyltransferase (MAT) Acyltransferase Transferase N-Acetylglucosaminyltransferase NF-κB Rho

144

Compounds

Natural Products

Recombinant Proteins

Cat No.	Product Name	Synonyms	Targets
T25450	GGTI 2147	GGTI2147,Geranylgeranyl transferase inhibitor-2147,GGTI-2147	NF-κB , Rho
	GGTI 2147 decreased Rac1 activity, down-regulated p65 expression, and ameliorated OGD/R-induced neuronal apoptosis.		NF-κB , Rho
T82343	Gamma-Glutamyl Transferase-IN-1
	Gamma-Glutamyl Transferase-IN-1 (compound 4de), a β-carboline 1-hydrazide inhibitor, exhibits antifungal and antibacterial properties by targeting glutamyltransferase. Its mechanism of action involves inducing the accumu...
T82342	Gamma-Glutamyl Transferase-IN-2
	Gamma-Glutamyl Transferase-IN-2 (compound 4dq), a β-carboline 1-hydrazide inhibitor, exhibits both antifungal and antibacterial properties by targeting glutamyltransferase. Its mode of action includes inducing reactive o...
T11282	FGTI-2734		Transferase
	FGTI-2734 is a dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT-1) inhibitor, exhibiting IC50 values of 250 nM and 520 nM for FT and GGT-1, respectively. It effectively prevents the membrane localizat...		Transferase
T9626	Cycloleucine		NMDAR
	Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM. Cycloleucine is also a competitive inhibitor of S-adenosyl-methionine mediated methylation with anxiolytic and cytostatic ef...		NMDAR
T11505	GSTO1-IN-1		Glutathione Peroxidase , GST
	GSTO1-IN-1 is a potent glutathione S-transferase omega 1 inhibitor (GSTO1; IC50: 31 nM).		Glutathione Peroxidase , GST
T6302	Lonafarnib	Sarasar,Sch66336	Raf , Transferase , Autophagy , Ras
	Lonafarnib (Sch66336) is an orally bioavailable FPTase inhibitor for H-ras, K-ras-4B, and N-ras (IC50: 1.9/5.2/2.8 nM).		Raf , Transferase , Autophagy , Ras
T4335	GNE-617	GNE617	NAMPT
	GNE-617, a specific NAMPT inhibitor(IC50=5 nM), shows potency in xenograft models of cancer.		NAMPT
T2678	LB42708		Transferase
	LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).		Transferase
T12171	Nampt-IN-5		P450 , NAMPT
	Nampt-IN-5 is a potent and orally active inhibitor of nicotinamide phosphoribosyltransferase (NAMPT) .		P450 , NAMPT
T6682	STF-118804	STF 118804,STF118804	Apoptosis , NAMPT
	STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 <10 nM.		Apoptosis , NAMPT
T4376	Nampt-IN-1	LSN3154567	c-Fms , NAMPT , CSF-1R
	Nampt-IN-1 (LSN3154567) (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an IC50 of 3.1 nM.		c-Fms , NAMPT , CSF-1R
T3182	L-778123 hydrochloride	L 778123	Telomerase , Transferase
	The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.		Telomerase , Transferase
T6271	Tipifarnib	R115777,Zarnestra,IND 58359	Transferase
	Tipifarnib (IND 58359) is a nonpeptidomimetic quinolinone with potential antineoplastic activity. Tipifarnib binds to and inhibits the enzyme farnesyl protein transferase, an enzyme involved in protein processing (farnes...		Transferase
T16409	OSMI-1		Others , Acyltransferase
	OSMI-1 is an O-GlcNAc transferase (OGT) inhibitor (IC50=2.7 μM) that is orally active and cell-permeable. OSMI-1 inhibits protein O-GlcNA acetylation without qualitatively altering cell-surface N- or O- linked glycans.		Others , Acyltransferase
T2700	FTI-277 hydrochloride	FTI 277 HCl	Apoptosis , Transferase , Ras
	FTI-277 hydrochloride (FTI 277 HCl) is an effective and specific farnesyltransferase (FTase) inhibitor (IC50: 500 pM); this selectivity is about 100-fold than the closely related GGTase I.		Apoptosis , Transferase , Ras
T38050	CP-609754		Transferase
	CP-609754 (LNK-754) is a potent and reversible farnesyltransferase inhibitor with potential anticancer activity.The IC50 for inhibiting farnesylation of recombinant human H-Ras is 0.57 ng/mL and recombinant K-Ras is 46 n...		Transferase
T1998	CHS-828	CHS 828,GMX1778	Apoptosis , NAMPT
	CHS-828 (GMX1778), a pyridyl cyanoguanidine, is an effective inhibitor of NAD+ biosynthesis enzyme NAMPT (IC50 <25 nM).		Apoptosis , NAMPT
T4564	Ethacrynic acid	Edecrin,Etacrynic Acid,Hydromedin	Others , Calcium Channel , NF-κB , GST
	Ethacrynic acid (Edecrin) is a nonsulfonamide loop diuretic that inhibits the activity of the Na+/K+/2Cl- cotransporter NKCC2 in the thick ascending limb of the loop of Henle. It also inhibits glutathione S-transferase a...		Others , Calcium Channel , NF-κB , GST
T5097	Ezatiostat	TER199(free base),TLK199	Apoptosis , Glutathione Peroxidase , GST
	Ezatiostat (TER199(free base)) is a tripeptide analog of glutathione that can selectively inhibit GSTP1-1 catalytic activity.		Apoptosis , Glutathione Peroxidase , GST
T22665	PD 128042	CI 976	Acyltransferase
	PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor. CI 976 inhibits Golgi-associated LPAT activity (IC50: 15 μM) and multi...		Acyltransferase
T17102	Tipifarnib (S enantiomer)	Tipifarnib S enantiomer,(S)-(-)-R-115777,(S)-Tipifarnib,IND-58359 S enantiomer	Transferase
	Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).		Transferase
T12854	SBI-797812		NAMPT
	SBI-797812 is structurally similar to active-site directed inhibitor of NAMPT(NAMPT with EC50 of 0.37 μM).		NAMPT
T2644	(E)-Daporinad	Daporinad,(E)-N-[4-(1-BENZOYL-PIPERIDIN-4-YL)-BUTYL]-3-PYRIDIN-3-YL-ACRYLAMIDE,APO866,FK866	NAMPT , Transferase , Autophagy
	(E)-Daporinad (FK866) is a small molecule inhibitor of nicotinamide phosphoribosyltransferase (NMPRTase), with potential antineoplastic and antiangiogenic activities.		NAMPT , Transferase , Autophagy
T22776	Ezatiostat hydrochloride	TLK199 HCl,TER199	Glutathione Peroxidase
	Ezatiostat hydrochloride (TLK199 HCl) is an effective inhibitor of glutathione S-transferase. Ezatiostat hydrochloride is a novel glutathione analog and the potential treatment of cytopenias. In addition, Ezatiostat hydr...		Glutathione Peroxidase
T61037	Glycosyltransferase-IN-1		Others
	Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.		Others
T11563	Histone Acetyltransferase Inhibitor II		Epigenetic Reader Domain , Histone Acetyltransferase
	Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity in mammalian cells.		Epigenetic Reader Domain , Histone Acetyltransferase
T77560	Histone acetyltransferase p300 Inhibitor 4c		Carbonic Anhydrase , AChE
	Histone acetyltransferase p300 Inhibitor 4c is a 2-aminothiazole derivative. Histone acetyltransferase p300 Inhibitor 4c inhibited hCA I, hCA II, AChE and BChE with Ki values of 0.008 ± 0.001, 0.124 ± 0.017, 0.129 ± 0.03...		Carbonic Anhydrase , AChE
T75416	Alpha-1,3-N-Acetylgalactosaminyltransferase (Pm1138)
	Alpha-1,3-N-Acetylgalactosaminyltransferase (Pm1138) (EC 2.4.1.40(Pm1138)), also known as the ABO system transferase, exhibits glycosyl transferase activity [1].
T76158	Phosphate acetyltransferase
	Phosphate acetyltransferase, a transferase enzyme utilized in biochemical research, catalyzes the reversible acetylation of CoA from acetyl-P, yielding acetyl-CoA and inorganic phosphate. This process is integral to acet...
T63738	Purine phosphoribosyltransferase-IN-2
	Purine phosphoribosyltransferase-IN-2 is a potent inhibitor of Plasmodium falciparum (Pf), Plasmodium vivax (Pv), and Trypanosoma brucei (Tbr) 6-oxopurine phosphoribosyltransferase (PRT) with Ki values of 30, 20, and 2 n...
T75421	Alpha-2,3-Sialyltransferase (PmST3)
	alpha-2,3-Sialyltransferase (PmST3) is a beta-galactoside. alpha-2,3-Sialyltransferase (PmST3) catalyzes the transfer of sialic acid to carbohydrate groups of glycoproteins and glycolipids [1] .
T63737	Purine phosphoribosyltransferase-IN-1
	Purinephosphoribosyltransferase-IN-1 (Compound (S,R)-48) is a potent inhibitor of Plasmodium falciparum (Pf), Plasmodium vivax (Pv) and Trypanosoma brucei (Tbr) 6-oxopurine phosphate ribosyltransferase (PRT) with Ki valu...
T75418	Alpha-1,3-Galactosyltransferase (GTB)
	Alpha-1,3-Galactosyltransferase (GTB) (alpha 1,3GT) is responsible for catalyzing the synthesis of the α-galactose (α-Gal) epitope, known as a xenoantigen. This enzyme facilitates the transfer of galactose from UDP-Gal t...
T75419	Alpha-2,8-Sialyltransferase (CstII)
	Alpha-2,8-Sialyltransferase (CstII) (ST8Sia VI), belonging to the alpha2,8-sialyltransferase (ST8Sia) family, primarily catalyzes the elongation of the α2,8-linked oligo/polysialic acid chain on the sialic acid (Sia) res...
T75399	GlcNAc 1-P uridyltransferase (CjGlmU)
	GlcNAc 1-P uridyltransferase (CjGlmU), a sugar nucleotidyltransferase (SNT), employs UTP and GlcNAc-1-P to synthesize UDP-GlcNAc, with potential implications in antimicrobial agent research [1].
T75413	Beta-1,4-Galactosyltransferase (LgtB)
	Beta-1,4-Galactosyltransferase (LgtB) (B4GALT1(LgtB)), a key enzyme in biochemical research, catalyzes the transfer of UDP-galactose to N-acetylglucosamine, resulting in the synthesis of galactose beta-1,4-N-acetylglucos...
T13429	α-2,3-sialyltransferase-IN-1	Lith-O-Asp analog	Others
	α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).		Others
T11037	Diacylglycerol acyltransferase inhibitor-1		Others
	Diacylglycerol Acyltransferase Inhibitor-1, a diacylglycerol acyltransferase (DGAT1) inhibitor, effectively suppresses the activity of DGAT1.		Others
T75414	Alpha-1,4-Galactosyltransferase (LgtC)
	Alpha-1,4-Galactosyltransferase (LgtC) (A4GALT), a glycosphingolipid-specific glycosyltransferase, catalyzes the transfer of a galactose molecule to the alpha-1,4 position on lactosylceramide, resulting in the formation ...
T75411	Beta-1, 3-N-Acetylhexaminyltransferase (LgtA)
	Beta-1, 3-N-Acetylhexaminyltransferase (LgtA), a glycosyltransferase, plays a critical role in biochemical studies by catalyzing the transfer of N-acetylglucosamine from UDP-GlcNAc to substrates including N-acetyllactosa...
T75415	Beta-1,3-Galactosyltransferase (CgtB)
	Beta-1,3-Galactosyltransferase (CgtB) (GM1-synthase), an enzyme critical for the production of sialylated lipooligosaccharide (LOS SIAL), plays a key role in biochemical research. This enzyme facilitates the incorporatio...
T78352	N-acetylglucosamine-1-P uridyltransferase (AGX1)	GlcNAc1pUT
	N-acetylglucosamine-1-P uridyltransferase (AGX1) (GlcNAc1pUT) is a bifunctional enzyme that couples with GlcNAc-1-P and UTP to catalyze the synthesis of UDP-GlcNAc through an uridyltransfer reaction. It exhibits acetyltr...
T78353	Alpha-2,6-Sialyltransferase (Pd26ST)
	Alpha-2,6-Sialyltransferase (Pd26ST) efficiently catalyzes the sialylation of both terminal and internal galactose and N-acetylgalactosamine residues, resulting in the production of terminal α2,6-sialosides [1].
T78364	Alanine aminotransferase		Endogenous Metabolite
	Alanine aminotransferase (ALT), a pyridoxal-dependent enzyme, catalyzes the reversible interconversion of L-alanine and 2-oxoglutarate into pyruvate and L-glutamate [1].		Endogenous Metabolite
T75420	Alpha-1,3/4-Fucosyltransferase (α1,3/4FucT)
	alpha-1,3/4-Fucosyltransferase (α1,3/4FucT) (Hp3/4FT) can be found in Helicobacter pylori . alpha-1,3/4-Fucosyltransferase (α1,3/4FucT) catalyzes fucose transfer from donor GDP-beta-l-fucose to the GlcNAc [1] .
T75417	Alpha-1,3-Galactosyltransferase (a1,3GalT)
	Alpha-1,3-Galactosyltransferase (a1,3GalT) (GGTA1) catalyzes the synthesis of the α-gal epitope by transferring a galactose (Gal) molecule in an α1-3 linkage from a uridyl-diphosphate (UDP) donor to the N-acetyllactosami...
T75389	Catechol O-methyltransferase
	Catechol O-methyltransferase (COMT) is a magnesium-dependent enzyme that mediates the transfer of methyl groups from S-adenosyl methionine to the hydroxyl group on dopamine, thus converting it to 3-methoxytyramine. COMT ...
T76178	Aspartate aminotransferase
	Aspartate aminotransferase (AST) is a transaminase enzyme, is often used in biochemical studies. Aspartate aminotransferase catalyzes aspartate and alpha-ketoglutarate converts to oxaloacetate and glutamate. Aspartate am...
T14375	AZD3988		Transferase
	AZD3988 is an inhibitor of diacylglycerol acyl transferase-1 (DGAT-1). For human, rat, mouse, the IC50s values are 6, 5, 11 nM , respectively.		Transferase

Compounds

GGTI 2147

T25450

Synonym: GGTI2147,Geranylgeranyl transferase inhibitor-2147,GGTI-2147

Target: NF-κB, Rho

Gamma-Glutamyl Transferase-IN-1

T82343

Synonym:

Target:

Gamma-Glutamyl Transferase-IN-2

Target: Transferase

Target: Glutathione Peroxidase, GST

Lonafarnib

T6302

Synonym: Sarasar,Sch66336

Target: Raf, Transferase, Autophagy, Ras

Target: Transferase

Synonym: STF 118804,STF118804

Target: Apoptosis, NAMPT

Nampt-IN-1

T4376

Synonym: LSN3154567

Target: c-Fms, NAMPT, CSF-1R

L-778123 hydrochloride

T3182

Synonym: L 778123

Target: Telomerase, Transferase

Tipifarnib

T6271

Synonym: R115777,Zarnestra,IND 58359

Target: Transferase

OSMI-1

T16409

Synonym:

Target: Others, Acyltransferase

FTI-277 hydrochloride

T2700

Synonym: FTI 277 HCl

Target: Apoptosis, Transferase, Ras

CP-609754

T38050

Synonym:

Target: Transferase

CHS-828

T1998

Synonym: CHS 828,GMX1778

Target: Apoptosis, NAMPT

Ethacrynic acid

T4564

Synonym: Edecrin,Etacrynic Acid,Hydromedin

Target: Others, Calcium Channel, NF-κB, GST

Ezatiostat

T5097

Synonym: TER199(free base),TLK199

Target: Apoptosis, Glutathione Peroxidase, GST

PD 128042

T22665

Synonym: CI 976

Target: Acyltransferase

Tipifarnib (S enantiomer)

T17102

Synonym: Tipifarnib S enantiomer,(S)-(-)-R-115777,(S)-Tipifarnib,IND-58359 S enantiomer

Target: Transferase

Synonym: Daporinad,(E)-N-[4-(1-BENZOYL-PIPERIDIN-4-YL)-BUTYL]-3-PYRIDIN-3-YL-ACRYLAMIDE,APO866,FK866

Target: NAMPT, Transferase, Autophagy

Ezatiostat hydrochloride

T22776

Synonym: TLK199 HCl,TER199

Target: Glutathione Peroxidase

Glycosyltransferase-IN-1

T61037

Synonym:

Target: Others

Histone Acetyltransferase Inhibitor II

T11563

Synonym:

Target: Epigenetic Reader Domain, Histone Acetyltransferase

Histone acetyltransferase p300 Inhibitor 4c

T77560

Synonym:

Target: Carbonic Anhydrase, AChE

alpha-1,3-N-Acetylgalactosaminyltransferase (Pm1138)

T75416

Synonym:

Target:

Phosphate acetyltransferase

T76158

Synonym:

Target:

Purine phosphoribosyltransferase-IN-2

T63738

Synonym:

Target:

alpha-2,3-Sialyltransferase (PmST3)

T75421

Synonym:

Target:

Purine phosphoribosyltransferase-IN-1

T63737

Synonym:

Target:

alpha-1,3-Galactosyltransferase (GTB)

T75418

Synonym:

Target:

alpha-2,8-Sialyltransferase (CstII)

T75419

Synonym:

Target:

GlcNAc 1-P uridyltransferase (CjGlmU)

T75399

Synonym:

Target:

beta-1,4-Galactosyltransferase (LgtB)

T75413

Synonym:

Target:

α-2,3-sialyltransferase-IN-1

T13429

Synonym: Lith-O-Asp analog

Target: Others

Diacylglycerol acyltransferase inhibitor-1

T11037

Synonym:

Target: Others

alpha-1,4-Galactosyltransferase (LgtC)

T75414

Synonym:

Target:

beta-1, 3-N-Acetylhexaminyltransferase (LgtA)

T75411

Synonym:

Target:

beta-1,3-Galactosyltransferase (CgtB)

T75415

Synonym:

Target:

N-acetylglucosamine-1-P uridyltransferase (AGX1)

T78352

Synonym: GlcNAc1pUT

Target:

alpha-2,6-Sialyltransferase (Pd26ST)

T78353

Synonym:

Target:

Alanine aminotransferase

T78364

Synonym:

Target: Endogenous Metabolite

alpha-1,3/4-Fucosyltransferase (α1,3/4FucT)

T75420

Synonym:

Target:

alpha-1,3-Galactosyltransferase (a1,3GalT)

T75417

Synonym:

Target:

Catechol O-methyltransferase

T75389

Synonym:

Target:

Aspartate aminotransferase

Target: Transferase

Cat No.	Product Name	Synonyms	Targets
TN6512	Tectol		Transferase , Parasite
	Tectol has anti-plasmodial activity, it as a moderately active growth inhibitor with an IC50 3.44±0.20μM. It exhibited significant activity against human leukemia cell lines HL60 and CEM. Tectol may cause itchy dermatiti...		Transferase , Parasite
TQ0165	Arglabin	(+)-Arglabin	NOD-like Receptor (NLR) , Transferase , NOD , Autophagy
	Arglabin ((+)-Arglabin) is a natural product isolated from Artemisia glabella, is a NLRP3 inflammasome inhibitor, has anti-atherogenic and anticancer effects.		NOD-like Receptor (NLR) , Transferase , NOD , Autophagy
T3S0012	Coniferyl ferulate		P-gp , GST
	Coniferyl ferulate is a strong inhibitor of glutathione S-transferase (GST) isolated from Radix Angelicae sinensis. It shows strong inhibition of human placental GST (IC50: 0.3 μM). It also reverses multidrug resistance ...		P-gp , GST
TN1078	Seneciphylline		P450 , GST
	Seneciphylline, one of the hepatotoxic pyrolizidine alkaloids, has mutagenic activity in Drosophila and their transfer into rat milk.Seneciphylline can significantly increased the activities of epoxide hydrase and glutat...		P450 , GST
T7995	α-Angelica lactone	Alpha-Angelica Lactone	Others , GST
	α-Angelica lactone has cardiotonic activity, may exert their effects by providing an increased contraction-dependent calcium pool to be released upon systolic depolarization.		Others , GST
T3S0541	Curzerene		Apoptosis , GST
	Curzerene, a sesquiterpene compound derived from the rhizome of Curculigo orchioides Gaertn, possesses potent anti-cancer properties. It is known to induce apoptosis in cells[1] and also suppress the expression of glutat...		Apoptosis , GST
TN3270	(R)-3β-Hydroxy steroid sulfotransferase-IN-11		Others
			Others
TN1474	Caulilexin C		Others , Antifungal
	Caulilexin C shows inhibitory activity on human Acyl CoA: cholesterol transferase I (hACATI) and on human Acyl CoA: cholesterol transferase 2 (hACAT2) at 100 mug/ml.		Others , Antifungal
T3314	Perillyl alcohol	Isocarveol,Perilla alcohol	Apoptosis , Endogenous Metabolite
	Perillyl Alcohol is a naturally occurring monoterpene related to limonene with antineoplastic activity. Perillyl alcohol (Isocarveol) inhibits farnesyl transferase and geranylgeranyl transferase, thereby preventing post-...		Apoptosis , Endogenous Metabolite
TJS0405	Lucidin	NSC 30546,Henine	Others
	1. Lucidin (NSC-30546) and its derivatives are genotoxic, it is mutagenic at the hypoxanthine-guanine phosphoribosyl transferase gene locus.		Others
T6758	Anisomycin	Flagecidin,NSC 76712,Wuningmeisu C	Apoptosis , DNA/RNA Synthesis , Antibacterial , Antibiotic , JNK
	Anisomycin (NSC-76712) is an antibiotic isolated from various Streptomyces species. It interferes with protein and DNA synthesis by inhibiting peptidyl transferase or the 80S ribosome system.
T5654	Musk ketone		Others
	Musk ketone can induce the growth repression and the apoptosis of cancer cells. Musk ketone increases activity of glutathione S-transferase and thus may prove to be useful cancer chemoprotectant.		Others
T3S0218	Thonningianin A		Apoptosis , Others
	1. Thonningianin A has anti-cancer activities.2. Thonningianin A represents a new potent glutathione S-transferase in vitro inhibitor.3. Thonningianin A has antioxidant property, involves radical scavenging, anti-superox...		Apoptosis , Others
T11680	Isoasatone A		P450
	Isoasatone A is a natural product isolated from the plant Heterotropa takaoi M., with anti-insect activity.		P450
T6S0071	Fraxinellone		HIF/HIF Prolyl-Hydroxylase , STAT , PD-1/PD-L1
	1. Fraxinellone significantly reduced weight loss and diarrhea in mice and alleviated the macroscopic and microscopic signs of the disease. 2. Fraxinellone exhibited a variety of insecticidal activities including feeding...		HIF/HIF Prolyl-Hydroxylase , STAT , PD-1/PD-L1
T4848	Mandelic acid	acidomandelico,DL-Mandelic acid	Others , Endogenous Metabolite , Antibacterial
	It is an isomer of cresotinic acid (2-hydroxy-3-methylbenzoic acid) and oxymethylbenzoic acid (2-methoxybenzoic acid). Derivatives of mandelic acid are formed as a result of metabolism of adrenaline and noradrenaline by ...		Others , Endogenous Metabolite , Antibacterial
T24412	Lipoxamycin	G 26146,G-26146,G26146,Neoenactin M1
	Lipoxamycin is an inhibitor of serine palmitoyl-transferase.
T11842	Levomecol		Others
	Levomecol, a broad-spectrum antibiotic derived from Streptomyces venezuelae, comprises Chloramphenicol and Methyluracil. It exerts its bacteriostatic effect by binding to the bacterial ribosome, inhibiting protein synthe...		Others
TN2849	3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid		Antifection
	2-O-beta-d-Glucosyloxy-4-methoxybenzenepropanoic acid[3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid] exhibits glutathione S-transferase (GST) inhibitory and antifungal activities.		Antifection
TN4443	Lipiferolide		Telomerase , Antifection
	Lipiferolide is an inhibitor of farnesyl protein transferase(FPTase), it inhibits the FPTase activity in a dose-dependent manner, and shows cell growth inhibitory activity against several tumor cells, it possesses cytoto...		Telomerase , Antifection
T29329	24-Methylenecholesterol	24Methylenecholesterol,24 Methylenecholesterol,Chalinasterol,Ostreasterol	Acyltransferase
	24-Methylenecholesterol (24 Methylenecholesterol) is a natural marine sterol, which stimulates cholesterol acyl transferase (ACAT) in human macrophages.		Acyltransferase
TN2834	27-p-Coumaroyloxyursolic acid		Others
	27-trans-p-Coumaroyloxyursolic acid and 27-cis-p-coumaroyloxyursolic acid show potent inhibitory activity in the acyl CoA cholesteryl acyl transferase (ACAT) assay.		Others
T75696	Ilexoside XLVIII
	Ilexoside XLVIII, a triterpene saponin isolated from the aqueous extract of Ilex kudincha leaves [1], functions as an acyl CoA cholesteryl acyl transferase (ACAT) inhibitor.
TN4345	Jacobine		Others
	Jacobine induces significant dose-dependent DNA-DNA interstrand cross-linking over the entire range of doses. It was catalyzed by guinea pig hepatic glutathione-S-transferase enzymes in in vitro experiments.		Others
T11202	Enniatin complex		Others
	Enniatin complex, a mixture of cyclohexadepsipeptides predominantly derived from various Fusarium species of fungi, exhibits inhibitory effects on enzymes such as acyl-CoA: cholesterol acyl transferase. Furthermore, it h...		Others
T38299	Tunicamycin V
	Tunicamycin 15:1 is a mixture of tunicamycin structural isomers that contains a 15-carbon N-acyl chain with variable branching patterns.References Tunicamycin 15:1 is a mixture of tunicamycin structural isomers that cont...

Natural Products

Tectol

TN6512

Synonym:

Target: Transferase, Parasite

Arglabin

TQ0165

Synonym: (+)-Arglabin

Target: NOD-like Receptor (NLR), Transferase, NOD, Autophagy

Synonym: Alpha-Angelica Lactone

Target: Apoptosis, GST

(R)-3β-Hydroxy steroid sulfotransferase-IN-11

Target: Others, Antifungal

Perillyl alcohol

T3314

Synonym: Isocarveol,Perilla alcohol

Target: Apoptosis, Endogenous Metabolite

Lucidin

TJS0405

Synonym: NSC 30546,Henine

Target: Others

Anisomycin

T6758

Synonym: Flagecidin,NSC 76712,Wuningmeisu C

Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, JNK

Target: Apoptosis, Others

Target: HIF/HIF Prolyl-Hydroxylase, STAT, PD-1/PD-L1

Mandelic acid

T4848

Synonym: acidomandelico,DL-Mandelic acid

Target: Others, Endogenous Metabolite, Antibacterial

Lipoxamycin

T24412

Synonym: G 26146,G-26146,G26146,Neoenactin M1

3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid

Target: Telomerase, Antifection

24-Methylenecholesterol

T29329

Synonym: 24Methylenecholesterol,24 Methylenecholesterol,Chalinasterol,Ostreasterol

Target: Acyltransferase

27-p-Coumaroyloxyursolic acid

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-00539	GSTA1 Protein, Human, Recombinant (His)	Human	HEK293
	GSTA1 (Glutathione S-Transferase Alpha 1) is a Protein Coding gene. This gene encodes a member of a family of enzymes that function to add glutathione to target electrophilic compounds. Glutathione S-transferases (GSTs) ...
TMPH-00164	4'-phosphopantetheinyl transferase ffp Protein, Bacillus subtilis, Recombinant (His & Myc)	Bacillus subtilis	E. coli
	4'-phosphopantetheinyl transferase ffp Protein, Bacillus subtilis, Recombinant (His & Myc) is expressed in E. coli.
TMPH-00569	AtoD Protein, E. coli, Recombinant (His & Myc)	E. coli	E. coli
	atoD Protein, E. coli, Recombinant (His & Myc) is expressed in E. coli.
TMPY-00027	GSTT2B Protein, Human, Recombinant (His)	Human	HEK293
	GSTT2B Protein, Human, Recombinant (His) is expressed in HEK293 with His tag. The predicted molecular weight is 29 kDa. Accession number: P0CG29
TMPY-03332	PRTFDC1 Protein, Human, Recombinant (His)	Human	E. coli
	PRTFDC1 is a member of the purine/pyrimidine phosphoribosyltransferase family. It can bind GMP, IMP and alpha-D-5-phosphoribosyl 1-pyrophosphate (PRPP). The epigenetic silencing of PRTFDC1 by hypermethylation of the CpG ...
TMPY-03338	GSTZ1 Protein, Human, Recombinant (His)	Human	E. coli
	GSTZ1 (Glutathione S-Transferase Zeta 1) is a Protein Coding gene. 3 alternatively spliced human isoforms have been reported. GSTZ1 gene is a member of the glutathione S-transferase (GSTs) super-family which encodes mult...
TMPY-03450	GSTK1 Protein, Human, Recombinant	Human	E. coli
	GSTK1 gene encodes a member of the kappa class of the glutathione transferase superfamily of enzymes that function in cellular detoxification. Glutathione S-transferases (GSTs) are a family of enzymes that catalyze a var...
TMPH-00406	CtfB Protein, Clostridium acetobutylicum, Recombinant (His & Myc)	Clostridium acetobutylicum	E. coli
	ctfB Protein, Clostridium acetobutylicum, Recombinant (His & Myc) is expressed in E. coli.
TMPY-01554	GSTM5 Protein, Human, Recombinant (His)	Human	E. coli
	GSTM5 Protein, Human, Recombinant (His) is expressed in E. coli with His tag. The predicted molecular weight is 27.9 kDa. Accession number: AAH58881.1
TMPH-02379	ArnT Protein, Klebsiella pneumoniae, Recombinant (His)	Klebsiella pneumoniae	E. coli
	Catalyzes the transfer of the L-Ara4N moiety of the glycolipid undecaprenyl phosphate-alpha-L-Ara4N to lipid A. The modified arabinose is attached to lipid A and is required for resistance to polymyxin and cationic antim...
TMPJ-00611	SFP Protein, B.subtilis, Recombinant (His)	B.subtilis	E. coli
	The Bacillus subtilis enzyme Sfp, required for production of the lipoheptapeptide antibiotic surfactin, posttranslationally phosphopantetheinylates a serine residue in each of the seven peptidyl carrier protein domains o...
TMPY-02223	GSTM2 Protein, Human, Recombinant (His)	Human	E. coli
	Glutathione S-transferase Mu 2, also known as GST class-mu 2, GSTM2-2, and GSTM2, is a cytoplasm protein that belongs to the GST superfamily and Mu family. GSTM2 / GST4 contains one GST C-terminal domain and one GST N-te...
TMPH-03438	CHS1 Protein, S. cerevisiae, Recombinant (His)	Saccharomyces cerevisiae	E. coli
	Polymerizes chitin, a structural polymer of the cell wall and septum, by transferring the sugar moiety of UDP-GlcNAc to the non-reducing end of the growing chitin polymer. Required for mitotic division septum formation d...
TMPJ-00765	TDT Protein, Human, Recombinant (His)	Human	E. coli
	Terminal deoxynucleotidyl transferase (TdT) is a highly conserved vertebrate enzyme that possesses the unique ability to catalyze the random addition of deoxynucleoside 5'-triphosphates onto the 3'-hydroxyl group of a si...
TMPJ-00499	GSTP1 Protein, Human, Recombinant	Human	E. coli
	Glutathione S-transferase P (GSTP1) is an enzyme that contains 1 GST C-terminal domain, 1 GST N-terminal domain. GSTP1 belongs to the GST superfamily, the GSTs are a family of enzymes that play an important role in deto...
TMPH-00017	AcpS Protein, Acholeplasma laidlawii, Recombinant (His & Myc)	Acholeplasma laidlawii	E. coli
	Transfers the 4'-phosphopantetheine moiety from coenzyme A to a Ser of acyl-carrier-protein.
TMPK-01001	RNF43 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293
	RNF43 (E3 ubiquitin-protein ligase RNF43 or RING-type E3 ubiquitin transferase RNF43) functions as a tumor suppressor, by exerting a predominant negative feedback mechanism in the Wnt/β-catenin signaling pathway. RNF43 i...
TMPJ-01302	ACAT2 Protein, Human, Recombinant (His)	Human	E. coli
	ACAT2 is a cytoplasmic enzyme which belongs to the thiolase family. ACAT2 takes part in lipid metabolism, lipoprotein assembly, catalyzing cholesterol esterification in mammalian cells. It is responsible for the synthesi...
TMPH-02628	Cathepsin C Protein, Mouse, Recombinant (His & Myc)	Mouse	E. coli
	Thiol protease. Has dipeptidylpeptidase activity. Can act as both an exopeptidase and endopeptidase. Can degrade glucagon. Plays a role in the generation of cytotoxic lymphocyte effector function.
TMPH-03448	EHT1 Protein, S. cerevisiae, Recombinant (His)	Saccharomyces cerevisiae	E. coli
	Displays enzymatic activity both for medium-chain fatty acid (MCFA) ethyl ester synthesis and hydrolysis (esterase activity). MCFA are toxic for yeast and this enzyme could thus be involved in their detoxification by est...
TMPJ-01115	GALNT3 Protein, Human, Recombinant (His)	Human	Human Cells
	Polypeptide N-acetylgalactosaminyltransferase 3(GALNT3) belongs to the glycosyltransferase 2 family and galNAc-T subfamily. It expressed in organs that contain secretory epithelial glands and it highly expressed in pancr...
TMPJ-01223	GALNTL1 Protein, Human, Recombinant (His)	Human	Human Cells
	Putative polypeptide N-acetylgalactosaminyltransferase-like protein 1, also known as Polypeptide GalNAc transferase-like protein 1, Protein-UDP acetylgalactosaminyltransferase-like protein 1, UDP-GalNAc:polypeptide N-ace...
TMPJ-00690	PGDS Protein, Human, Recombinant	Human	E. coli
	Hematopoietic Prostaglandin D Synthase (HPGDS) belongs to the GST superfamily and Sigma family. HPGDS contains one GST C-terminal domain and one GST N-terminal domain. HPGDS is highly expressed in adipose tissue, macroph...
TMPY-05693	SARS-CoV-2 Methyltransferase/ME Protein (His)	SARS-CoV-2	E. coli
	Coronavirus encodes the 2’-O-MTase (2'O Methyltransferase) that is composed of the catalytic subunit nsp16 and the stimulatory subunit nsp10 and plays an important role in virus genome replication and evasion from innate...
TMPH-00573	DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)	E. coli	E. coli
	Catalyzes the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). It is the only animotransferase known to utilize SAM a...
TMPY-03445	Aspartate Aminotransferase Protein, Human, Recombinant (His)	Human	E. coli
	GOT1 (Glutamic-Oxaloacetic Transaminase 1) is a Protein Coding gene. GOT1 belongs to the class-I pyridoxal-phosphate-dependent aminotransferase family. Glutamic-oxaloacetic transaminase is a pyridoxal phosphate-dependent...
TMPJ-01429	SARS-CoV-2 Guanine-N7 methyltransferase Protein (His)	SARS-CoV-2	E. coli
	The nonstructural protein (nsp) 14 of SARS-CoV 2 was identified as a cap (guanine-N7)-methyltransferase (N7-MTase). Nsp14 of coronaviruses two different activities: an exoribonuclease activity acting on both ssRNA and ds...
TMPH-03604	Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His)	Streptomyces hygroscopicus	E. coli
	Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His) is expressed in E. coli.
TMPH-03608	Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His)	Streptomyces viridochromogenes	Yeast
	Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His) is expressed in Yeast.
TMPY-00279	Dengue virus DENV-2 (strain New Guinea C) NS5 (methyltransferase domain)/Nonstructural protein 5 Protein (His)	DENV	E. coli
	Dengue virus DENV-2 (strain New Guinea C) NS5 (methyltransferase domain)/Nonstructural protein 5 Protein (His) is expressed in E. coli with His tag. The predicted molecular weight is 35.5 kDa. Accession number: AAC59275....
TMPH-03609	Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His & SUMO)	Streptomyces viridochromogenes	E. coli
	Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-03600	Glucosyltransferase-SI Protein, S. mutans serotype c, Recombinant (His & Myc)	Streptococcus mutans	E. coli
	Production of extracellular glucans, that are thought to play a key role in the development of the dental plaque because of their ability to adhere to smooth surfaces and mediate the aggregation of bacterial cells and fo...
TMPH-00313	TRNA (guanine-N(7)-)-methyltransferase Protein, Brugia malayi, Recombinant (His)	Brugia malayi	E. coli
	Catalyzes the formation of N(7)-methylguanine at position 46 (m7G46) in tRNA.
TMPY-02279	Nucleoside phosphorylase/PNP Protein, Human, Recombinant (His)	Human	E. coli
	Purine nucleoside phosphorylase (PNP) is a purine-metabolizing enzyme that catalyzes the reversible phosphorolysis of 6-oxypurine (deoxy)nucleosides to their respective bases and (deoxy)ribose-1-phosphate. It is a key en...
TMPY-00365	GALNT7 Protein, Human, Recombinant (His)	Human	HEK293
	GalNAc-transferase-7 (GALNT7) is essential for the regulation of cell proliferation and has been implicated in tumorigenesis. Colorectal cancer (CRC) arises in a multistep molecular network process, which is from either ...
TMPY-02157	GST Protein, Schistosoma japonicum, Recombinant	Schistosoma japonicum	Baculovirus-Insect Cells
	Genetic engineers have used glutathione S-transferase to create the GST gene fusion system. This system is used to purify and detect proteins of interest. In a GST gene fusion system, the GST sequence is incorporated int...
TMPH-00893	AHCY Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Adenosylhomocysteine is a competitive inhibitor of S-adenosyl-L-methionine-dependent methyl transferase reactions; therefore adenosylhomocysteinase may play a key role in the control of methylations via regulation of the...
TMPH-01397	LANCL1 Protein, Human, Recombinant (His & Myc)	Human	E. coli
	Functions as glutathione transferase. Catalyzes conjugation of the glutathione (GSH) to artificial substrates 1-chloro-2,4-dinitrobenzene (CDNB) and p-nitrophenyl acetate. Mitigates neuronal oxidative stress during norma...
TMPJ-00087	VMO1 Protein, Human, Recombinant (His)	Human	Human Cells
	Vitelline membrane outer layer protein 1 homolog (VMO1) belongs to the VMO1 family is a 202 amino acid secreted protein. Exact function not known, component of the outer membrane of the vitelline layer of the egg. Seems ...
TMPY-01856	MGAT5 Protein, Human, Recombinant (His)	Human	HEK293
	Alpha-1,6-mannosylglycoprotein 6-beta-N-acetylglucosaminyltransferase A, also known as Alpha-mannoside beta-1,6-N-acetylglucosaminyl-transferase, Mannoside acetylglucosaminyltransferase 5, N-acetylglucosaminyl-transferas...
TMPJ-00053	PRL-2 Protein, Human, Recombinant (His)	Human	E. coli
	PTP4A2, also known as PRL2 or PTPCAAX2, is short for Protein tyrosine phosphatase type IVA 2. This protein exists in cell membrane, cytoplasm,endosome and membrane. PTP4A2 is often farnesylated during post-translational ...
TMPY-02596	GLT25D2 Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	Glycosyl transferase 25 domain 2 (GLT25D2) is a glucosyltransferase enzyme expressed only at low levels in the nervous system. Glycosyltransferases are enzymes that act as a catalyst for the transfer of a monosaccharide ...
TMPY-02421	PARP3 Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	Poly(ADP-ribose) polymerase 3 (PARP3) is an important member of the PARP family and shares high structural similarities with both PARP1 and PARP2. Poly(ADP-ribose) polymerase 3 (PARP3), a critical player in cellular resp...
TMPH-02292	B3GNT7 Protein, Human, Recombinant (His & Myc)	Human	E. coli
	N-acetyl glucosamine (GlcNAc) transferase that catalyzes the transfer of GlcNAc via a beta1->3 linkage from UDP-GlcNAc to the non-reducing terminal galactose (Gal) in the linearly growing chain of N- and O-linked keratan...
TMPY-06532	ART1 Protein, Human, Recombinant (His)	Human	HEK293
	Mono-ADP-ribosyltransferase (ART) 1 belongs to a family of mammalian ectoenzymes that catalyze the transfer of ADP-ribose from NAD+ to a target protein. ART1 is predominantly expressed in skeletal and cardiac muscle. It...
TMPY-04209	ART1 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293
	Mono-ADP-ribosyltransferase (ART) 1 belongs to a family of mammalian ectoenzymes that catalyze the transfer of ADP-ribose from NAD+ to a target protein. ART1 is predominantly expressed in skeletal and cardiac muscle. It...
TMPY-02640	FAM3B Protein, Human, Recombinant (hFc)	Human	HEK293
	Pancreatic derived factor, also known as FAM3B, is an islet-specific secreted cytokine specifically expressed at high levels in the islets of Langerhans of the endocrine pancreas. FAM3B protein is present in alpha- and b...
TMPY-01480	LTC4S Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	Leukotriene C4 synthase, also known as LTC4 synthase, Leukotriene-C(4) synthase, and LTC4S, is a multi-pass membrane protein that belongs to the MAPEG family. LTC4S is detected in the lung, platelets, and the myelogenous...
TMPY-01285	METTL11A Protein, Human, Recombinant	Human	E. coli
	Methyltransferase-like protein 11A, also known as METTL11A, is a member of the methyltransferase superfamily and METTL11 family. Methyltransferase is a type of transferase enzyme which transfers a methyl group from a don...
TMPY-01284	METTL11A Protein, Human, Recombinant (GST)	Human	E. coli
	Methyltransferase-like protein 11A, also known as METTL11A, is a member of the methyltransferase superfamily and METTL11 family. Methyltransferase is a type of transferase enzyme which transfers a methyl group from a don...
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