T9975 |
GPR183
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3-(3,4-difluorophenyl)-N-[3-fluoro-5-(morpholin-4-yl)phenyl]propanamide |
Others
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GPR183 is a chemotactic receptor known for its role in the maturation of B cells, and the endogenous ligand is the oxyst... |
TP1490 |
Proadrenomedullin (1-20), human
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Endogenous peptide agonist of Mas related GPR X2 (MRGPRX2, EC50 = 251 nM). Also a noncompetitive nicotinic cholinergic a... |
T40517 |
GPR30 agonist-1
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GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects. |
T60466 |
MRGPRX1 agonist 2
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MRGPRX1 agonist 2 (compound 1a) is a potent positive allosteric modulator of Mas-related G protein-coupled receptor X1 (... |
T40271 |
MrgprX2 antagonist-3
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MrgprX2 antagonist-3 is an MrgprX2 antagonist extracted from patent WO2021092240A1, example E117. MrgprX2 antagonist-3 c... |
T40273 |
MrgprX2 antagonist-2
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MrgprX2 antagonist-2 is an MrgprX2 antagonist extracted from patent WO2021092262A1, example E163. MrgprX2 antagonist-2 c... |
T40176 |
MrgprX2 antagonist-5
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MrgprX2 antagonist-5 is an MrgprX2 antagonist extracted from patent WO2020223255A1, example 16. MrgprX2 antagonist-5 can... |
T40270 |
MrgprX2 antagonist-1
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MrgprX2 antagonist-1 is an MrgprX2 antagonist extracted from patent WO2021092264A1, example E23. MrgprX2 antagonist-1 ca... |
T40268 |
MrgprX2 antagonist-4
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MrgprX2 antagonist-4 is an MrgprX2 antagonist extracted from patent US20210128561A1, compound B-51 E117. MrgprX2 antagon... |
T60497 |
MRGPRX1 agonist 3
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MRGPRX1 agonist 3 (compound 1f) is a potent positive allosteric modulator of Mas-related G protein-coupled receptor X1 (... |
T61055 |
GPR40 agonist 6
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GPR40 agonist 6 (Compound 7a) is a potent and selective agonist of free fatty acid receptor 1 ( FFAR1 or GPR40 ) with an... |
T36951 |
N-(p-Tosyl)-GPR-pNA acetate
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Others
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N-(p-Tosyl)-GPR-pNA acetate is a colorimetric substrate for thrombin that can act as a measure of thrombin activity. |
T8558 |
8-Azabicyclo[3.2.1]octan-3-one, 8-methyl
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Others
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8-Azabicyclo[3.2.1]octan-3-one, 8-methyl targets the MAS-related GPR member X1 (human) |
T27724 |
KDT 501 potassium
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Tetrahydroisohumulone , KDT 501 potassium salt , KDT 501 , KDT-501 |
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KDT 501, a PPAR agonist and G protein-coupled receptor (GPR) 120 agonist, is used potentially for the treatment of type ... |
TP1880 |
PAMP-12(human, porcine)
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PAMP-12 (human, porcine) |
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Potent endogenous peptide agonist of Mas related GPR X2 (MRGPRX2, EC50 = 57.2 nM). Corresponds to amino acids 9 to 20 of... |
T11455 |
GPR35 agonist 1
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Others
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GPR35 agonist 1 is a highly effective and specific GPR35/CXCR8 agonist (EC50: 5.8 nM). |
T23434 |
GPR35 agonist 2
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TC-G 1001 |
Others
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GPR35 agonist |
T11459 |
GPR40 agonist 1
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Others
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GPR40 agonist 1 is an effective new GPR40 agonist (EC50s: 17 nM and 2 nM for rGPR40 and hGPR40). |
T11454 |
GPR120 modulator 2
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Others
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GPR120 modulator 2 is useful for modulating GPR120. |
T10507 |
GPR40 Agonist 2
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GPR
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GPR40 Agonist 2 is a GPR40 agonist extracted from patent WO2009054479A1. It can be used in the research of diabetes. |