T40652 |
Meclizine
|
569-65-3
|
98%
|
|
Meclizine (Meclozine) shows antihistamine activity and reversibly inhibits the interaction of histamine at the H1 receptors . Meclizine is a member of the pipera...
|
T9353 |
OXOMEMAZINE
|
3689-50-7
|
98%
|
|
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
|
T10575 |
BMY-25271
|
78441-82-4
|
98%
|
|
BMY-25271 is an antagonist of histamine H2 receptor.
|
T11531 |
H3R-IN-1 Hydrochloride
|
T11531
|
98%
|
|
H3R-IN-1 Hydrochloride is a histamine receptor 3 ( H3R ) inverse agonist extracted from patent WO2013107336A1, compound example 2.
|
T10769 |
Cetirizine D4
|
1219803-84-5
|
98%
|
|
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
|
T11729 |
JTE-952
|
1255303-54-8
|
98%
|
|
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
|
TN1901 |
(-)-Maackiain
|
2035-15-6
|
98%
|
|
(-)-Maackiain, a phytoalexin, which is an anti-allergic compound that suppresses the up-regulation of the histamine H1 receptor (H1R) gene.
|
TN2895 |
3,5-Dicaffeoyl-epi-quinic acid
|
879305-14-3
|
98%
|
|
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
|
T17118 |
Toreforant
|
952494-46-1
|
98%
|
|
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
|
TN3483 |
Bakkenolide D
|
18456-03-6
|
98%
|
|
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
|
T3037 |
Cyclizine dihydrochloride
|
5897-18-7
|
98%
|
|
Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
|
T10770 |
Cetirizine D8
|
774596-22-4
|
98%
|
|
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
|
TN5279 |
Zeorin
|
22570-53-2
|
98%
|
|
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
|
T10794 |
Chlorcyclizine hydrochloride
|
14362-31-3
|
98%
|
|
Chlorcyclizine hydrochloride is an antagonist of histamine H1.
|
TN1913 |
Marmin
|
14957-38-1
|
98%
|
|
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
|
T15565 |
Imetit dihydrobromide
|
32385-58-3
|
98%
|
|
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
|
T15590 |
Iodophenpropit dihydrobromide
|
145196-87-8
|
98%
|
|
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
|
T11088 |
Doxepin D3 Hydrochloride
|
347840-07-7
|
98%
|
|
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
|
T32191 |
Irdabisant
|
1005402-19-6
|
98%
|
|
Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R K...
|
T6562 |
Latrepirdine dihydrochloride
|
97657-92-6
|
98%
|
|
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
|