T16476 |
PF-03654746
|
935840-31-6
|
99.1%
|
|
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
|
T3037 |
Cyclizine dihydrochloride
|
5897-18-7
|
|
|
Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
|
TN3699 |
Corchoionoside C
|
185414-25-9
|
98%
|
|
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
|
T10770 |
Cetirizine D8
|
774596-22-4
|
98%
|
|
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
|
T11729 |
JTE-952
|
1255303-54-8
|
98%
|
|
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
|
T15590 |
Iodophenpropit dihydrobromide
|
145196-87-8
|
98%
|
|
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
|
TN3483 |
Bakkenolide D
|
18456-03-6
|
98%
|
|
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
|
T12630 |
(R)-(-)-α-Methylhistamine dihydrobromide
|
868698-49-1
|
98%
|
|
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
|
TN2155 |
Rhodiocyanoside A
|
168433-86-1
|
98%
|
|
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
|
T11088 |
Doxepin D3 Hydrochloride
|
347840-07-7
|
98%
|
|
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
|
T15722 |
Lavoltidine
|
76956-02-0
|
98%
|
|
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
|
T17118 |
Toreforant
|
952494-46-1
|
98%
|
|
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
|
T12416 |
PF-03654746 Tosylate
|
1039399-17-1
|
98%
|
|
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
|
T12703 |
ReN-1869 hydrochloride
|
170149-76-5
|
98%
|
|
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
|
T19443L |
N-Acetylhistamine acetate
|
|
98%
|
|
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
|
T2S0118 |
Daurinoline
|
2831-75-6
|
98%
|
|
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
|
T12228 |
Niperotidine
|
84845-75-0
|
98%
|
|
Niperotidine is an antagonist of histamine H2-receptor.
|
T10575 |
BMY-25271
|
78441-82-4
|
98%
|
|
BMY-25271 is an antagonist of histamine H2 receptor.
|
TN4918 |
Roseoside
|
54835-70-0
|
98%
|
|
Roseoside possesses strong antioxidant properties, inhibiting lipid oxidation by 86.4, at 50 microg/mL. Roseoside has insulinotropic activity, enhances insulin r...
|
T11532 |
H4R antagonist 1
|
1429375-54-1
|
98%
|
|
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
|