Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T16476	PF-03654746	935840-31-6	99.1%
T16476	PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
T3037	Cyclizine dihydrochloride	5897-18-7
T3037	Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
TN3699	Corchoionoside C	185414-25-9	98%
TN3699	Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T10770	Cetirizine D8	774596-22-4	98%
T10770	Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T11729	JTE-952	1255303-54-8	98%
T11729	JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
T15590	Iodophenpropit dihydrobromide	145196-87-8	98%
T15590	Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
TN3483	Bakkenolide D	18456-03-6	98%
TN3483	Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T12630	(R)-(-)-α-Methylhistamine dihydrobromide	868698-49-1	98%
T12630	(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN2155	Rhodiocyanoside A	168433-86-1	98%
TN2155	Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T11088	Doxepin D3 Hydrochloride	347840-07-7	98%
T11088	Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
T15722	Lavoltidine	76956-02-0	98%
T15722	Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
T17118	Toreforant	952494-46-1	98%
T17118	Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
T12416	PF-03654746 Tosylate	1039399-17-1	98%
T12416	PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
T12703	ReN-1869 hydrochloride	170149-76-5	98%
T12703	ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
T19443L	N-Acetylhistamine acetate		98%
T19443L	N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
T2S0118	Daurinoline	2831-75-6	98%
T2S0118	Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
T12228	Niperotidine	84845-75-0	98%
T12228	Niperotidine is an antagonist of histamine H2-receptor.
T10575	BMY-25271	78441-82-4	98%
T10575	BMY-25271 is an antagonist of histamine H2 receptor.
TN4918	Roseoside	54835-70-0	98%
TN4918	Roseoside possesses strong antioxidant properties, inhibiting lipid oxidation by 86.4, at 50 microg/mL. Roseoside has insulinotropic activity, enhances insulin r...
T11532	H4R antagonist 1	1429375-54-1	98%
T11532	H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...