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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T16476 PF-03654746 935840-31-6 99.1%
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
T3037 Cyclizine dihydrochloride 5897-18-7
Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
TN3699 Corchoionoside C 185414-25-9 98%
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T10770 Cetirizine D8 774596-22-4 98%
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T11729 JTE-952 1255303-54-8 98%
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
T15590 Iodophenpropit dihydrobromide 145196-87-8 98%
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
TN3483 Bakkenolide D 18456-03-6 98%
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T12630 (R)-(-)-α-Methylhistamine dihydrobromide 868698-49-1 98%
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN2155 Rhodiocyanoside A 168433-86-1 98%
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T11088 Doxepin D3 Hydrochloride 347840-07-7 98%
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
T15722 Lavoltidine 76956-02-0 98%
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
T17118 Toreforant 952494-46-1 98%
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
T12416 PF-03654746 Tosylate 1039399-17-1 98%
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
T12703 ReN-1869 hydrochloride 170149-76-5 98%
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
T19443L N-Acetylhistamine acetate 98%
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
T2S0118 Daurinoline 2831-75-6 98%
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
T12228 Niperotidine 84845-75-0 98%
Niperotidine is an antagonist of histamine H2-receptor.
T10575 BMY-25271 78441-82-4 98%
BMY-25271 is an antagonist of histamine H2 receptor.
TN4918 Roseoside 54835-70-0 98%
Roseoside possesses strong antioxidant properties, inhibiting lipid oxidation by 86.4, at 50 microg/mL. Roseoside has insulinotropic activity, enhances insulin r...
T11532 H4R antagonist 1 1429375-54-1 98%
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
PF-03654746
T16476
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease....
Cyclizine dihydrochloride
T3037
Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
Corchoionoside C
TN3699
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
Cetirizine D8
T10770
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
JTE-952
T11729
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
Iodophenpropit dihydrobromide
T15590
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
Bakkenolide D
TN3483
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
(R)-(-)-α-Methylhistamine dihydrobromide
T12630
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
Rhodiocyanoside A
TN2155
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
Doxepin D3 Hydrochloride
T11088
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
Lavoltidine
T15722
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
Toreforant
T17118
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
PF-03654746 Tosylate
T12416
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
ReN-1869 hydrochloride
T12703
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
N-Acetylhistamine acetate
T19443L
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
Daurinoline
T2S0118
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
Niperotidine
T12228
Niperotidine is an antagonist of histamine H2-receptor.
BMY-25271
T10575
BMY-25271 is an antagonist of histamine H2 receptor.
Roseoside
TN4918
Roseoside possesses strong antioxidant properties, inhibiting lipid oxidation by 86.4, at 50 microg/mL. Roseoside has insulinotropic activity, enhances insulin r...
H4R antagonist 1
T11532
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
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