Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T40652	Meclizine	569-65-3	98%
T40652	Meclizine (Meclozine) shows antihistamine activity and reversibly inhibits the interaction of histamine at the H1 receptors . Meclizine is a member of the pipera...
T9353	OXOMEMAZINE	3689-50-7	98%
T9353	Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
T10575	BMY-25271	78441-82-4	98%
T10575	BMY-25271 is an antagonist of histamine H2 receptor.
T11531	H3R-IN-1 Hydrochloride	T11531	98%
T11531	H3R-IN-1 Hydrochloride is a histamine receptor 3 ( H3R ) inverse agonist extracted from patent WO2013107336A1, compound example 2.
T10769	Cetirizine D4	1219803-84-5	98%
T10769	Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T11729	JTE-952	1255303-54-8	98%
T11729	JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
TN1901	(-)-Maackiain	2035-15-6	98%
TN1901	(-)-Maackiain, a phytoalexin, which is an anti-allergic compound that suppresses the up-regulation of the histamine H1 receptor (H1R) gene.
TN2895	3,5-Dicaffeoyl-epi-quinic acid	879305-14-3	98%
TN2895	3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
T17118	Toreforant	952494-46-1	98%
T17118	Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
TN3483	Bakkenolide D	18456-03-6	98%
TN3483	Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T3037	Cyclizine dihydrochloride	5897-18-7	98%
T3037	Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
T10770	Cetirizine D8	774596-22-4	98%
T10770	Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
TN5279	Zeorin	22570-53-2	98%
TN5279	Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
T10794	Chlorcyclizine hydrochloride	14362-31-3	98%
T10794	Chlorcyclizine hydrochloride is an antagonist of histamine H1.
TN1913	Marmin	14957-38-1	98%
TN1913	Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
T15565	Imetit dihydrobromide	32385-58-3	98%
T15565	Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
T15590	Iodophenpropit dihydrobromide	145196-87-8	98%
T15590	Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
T11088	Doxepin D3 Hydrochloride	347840-07-7	98%
T11088	Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
T32191	Irdabisant	1005402-19-6	98%
T32191	Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R K...
T6562	Latrepirdine dihydrochloride	97657-92-6	98%
T6562	Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...