T77516 |
SARS-CoV-2-IN-39
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SARS-CoV
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Antiviral
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SARS-CoV-2-IN-39是一种 SARS-CoV-2 抑制剂,EC50 为 1 μM。 SARS-CoV-2-IN-39 具有抗病毒活性,通过抑制 SKP2 蛋白并稳定 BECN1 来抑制 SARS-CoV-2。 |
T60538 |
SARS-CoV-2-IN-14
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3',5-Dichlorosalicylanilide |
SARS-CoV
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SARS-CoV-2-IN-14 是一种有效的、可口服的 SARS-CoV-2 抑制剂(IC50 :0.39 μM),是一种氯硝柳胺类似物。SARS-CoV-2-IN-14在人血浆和肝 S9 酶测定中比氯硝柳胺稳定性更强。SARS-CoV-... |
T60919 |
SARS-CoV-2-IN-13
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SARS-CoV
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SARS-CoV-2-IN-13 (compound 6) 是氯硝柳胺的类似物。在人血浆和肝S9酶测定中,SARS-CoV-2-IN-13 比氯硝柳胺更稳定。SARS-CoV-2-IN-13 口服给药时可以提高生物利用度和半衰期。SARS-... |
T77510 |
SARS-CoV-2-IN-46
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SARS-CoV
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SARS-CoV-2-IN-46 是一种 SARS-CoV-2 抑制剂。 |
T36654 |
Anti-SARS-CoV-2 Spike mAb (CR3022)
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Anti-SARS-CoV-2 Spike mAb (CR3022) |
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Anti-SARS-CoV-2 Spike mAb (CR3022) is a human monoclonal IgG1 antibody derived from CHO cells. It specifically targets t... |
T36653 |
Anti-SARS-80R mAb
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Anti-SARS-80R mAb (SARS-80R) is a human IgG1 monoclonal antibody that is derived from CHO cells. Its main function is to... |
T61774 |
SARS 3CLpro-IN-1
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SARS 3CLpro-IN-1 (Compound 3b) is a stereo-specific SARS 3CL protease inhibitor that belongs to the octahydroisochromene... |
T38942 |
SARS-CoV-2-IN-9
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SARS-CoV-2-IN-9 is an inhibitor binding to subsites S1 and S2 in SARS-CoV-2 main protease. |
TMPY-06416 |
SARS-CoV-2 NSP8 Protein
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NSP8 is a nonstructural protein of coronavirus. NSP8 acts as a primase in RNA synthesis. NSP8 and NSP7 are essential co-... |
T40340 |
SARS-CoV-2-IN-10
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SARS-CoV-2-IN-10 is a powerful and non-toxic inhibitor of SARS-CoV-2 3CL protease, with IC50 and EC50 values of 0.13 nM ... |
T40341 |
SARS-CoV-2-IN-11
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SARS-CoV-2-IN-11 is a highly potent and non-toxic inhibitor of the 3C-like protease (3CLpro) of SARS-CoV-2, demonstratin... |
T40207 |
SARS-CoV-2-IN-7
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SARS-CoV-2-IN-7 demonstrates potent inhibition of viral replication in SARS-CoV-2-infected Vero E6 cells with an IC50 va... |
T62834 |
SARS-CoV-2-IN-22
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SARS-CoV-2-IN-22 是一种 SARS-CoV-2 pseudovirus 抑制剂 (IC50: 16.96 μM)。 |
T76270 |
SARS-CoV-2-IN-34
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SARS-CoV-2-IN-34 (S-20-1) 是一种具有广谱抑制活性的,可穿透血脑屏障的pan-coronavirus (CoV) fusion 抑制剂。SARS-CoV-2-IN-34 有效抑制伪型和真型 SARS-CoV-2 和其... |
T64184 |
SARS-CoV-2-IN-8
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SARS-CoV-2-IN-8 是一种 SARS-CoV-2 主要的蛋白酶抑制剂 (IC50: 0.75 μM)。 |
T60556 |
SARS-CoV-2-IN-16
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SARS-CoV-2-IN-16 (Compound 12) 是SARS-CoV-2核衣壳蛋白的有效抑制剂,具有强效的抗病毒活性(EC50 = 3.69 μM)。SARS-CoV-2-IN-16 以7.82 μM 的低Kd 值与 NPro ... |
T60962 |
SARS-CoV-2-IN-18
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SARS-CoV-2-IN-18 (Compound 26) 是 SARS-CoV-2 3C-样蛋白酶的有效抑制剂 (IC50 = 45 nM)。 |
T74946 |
SARS-CoV-2-IN-28
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SARS-CoV-2-IN-28 是一种双臂二磷酸 C7 烷基酯和具有扩展长度的分子镊子。SARS-CoV-2-IN-28 具有抗病毒活性,抑制 SARS-CoV-2 活力和病毒尖刺伪粒子转导的 IC50分别为 0.4 μM 和 1.0 μ... |
T74945 |
SARS-CoV-2-IN-27
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SARS-CoV-2-IN-27 是一种双臂二磷酸 C6 烷基酯和具有扩展长度的分子镊子。SARS-CoV-2-IN-27 具有抗病毒活性,抑制 SARS-CoV-2 活力和病毒尖刺伪粒子转导的 IC50分别为 1.0 μM 和 1.7 μ... |
T61613 |
SARS-CoV-2-IN-17
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SARS-CoV-2-IN-17 (Compound 16) is a highly effective inhibitor of SARS-CoV-2 nucleocapsid protein (NPro). It demonstrate... |