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Compounds

Cat No. Product Name
T16105 ML132 NCGC 00185682 Others
ML132 is an effective and selective inhibitor of caspase 1 (IC50: 0.316 nM).
T76665 Z-LEED-FMK
Z-LEED-FMK 是 caspase-13和 caspase-4抑制剂。Z-LEED-FMK 还能抑制S. typhimurium 感染的巨噬细胞中caspase-1的加工。
T73870 Arg-Gly-Asp-Ser TFA
Arg-Gly-Asp-Ser (TFA) 是整联蛋白结合序列,抑制整联蛋白受体 (integrinreceptor) 功能。Arg-Gly-Asp-Ser (TFA) 直接并特异性地结合 pro-caspase-8,pro-caspase...
T21293 MX1013 MX-1013,MX 1013
MX1013, a dipeptide pan-caspase inhibitor, inhibits caspase-1, -3, -6, -7, -8, and -9.
T24903 TRP-601 TRP601
TRP-601 is a caspase inhibitor.
T31040 CP-18 F-18 CP 18 F-18,CP18 F-18,(18F)-CP18
CP-18 F-18 is a DEVD (the caspase 3 substrate recognition motif) that is an imaging tracer for caspase-3 activity in apo...
T16998 Tauroursodeoxycholate dihydrate 牛磺熊去氧胆酸二水合物,UR 906 dihydrate,Taurolite dihydrate,TUDCA dihydrate Caspase , ERK
Tauroursodeoxycholate dihydrate is an endoplasmic reticulum stress inhibitor. Tauroursodeoxycholate also inhibits ERK. T...
T73683 AC-VEID-CHO TFA
AC-VEID-CHO (TFA) 是一种多肽来源的半胱天冬酶抑制剂,对 Caspase-6、Caspase-3 和 Caspase-7 具有抑制作用,IC50值分别为 16.2 nM、13.6 nM 和162.1 nM。AC-VEID-C...
T36341 Ac-DNLD-AMC
Ac-DNLD-AMC is a fluorogenic caspase-3 substrate. Upon enzymatic cleavage by caspase-3, 7-amino-4-methylcoumarin (AMC) i...
T36334 Z-VAD-AMC (acetate)
Z-VAD-AMC is a fluorogenic substrate for caspase-1. Upon enzymatic cleavage by caspase-1, 7-amino-4-methylcoumarin (AMC)...
T36331 Z-AEVD-FMK Z-AEVD-FMK,Z-Ala-Glu-Val-Asp-Fluoromethyl Ketone
Z-AEVD-FMK is an irreversible inhibitor of caspase-10 and related caspases.[1] At 10 µM, it can prevent the initiati...
T36354 Suc-YVAD-AMC (acetate)
Suc-YVAD-AMC is a fluorogenic substrate for caspase-1. Upon enzymatic cleavage by caspase-1, 7-amino-4-methylcoumarin (A...
T36342 Ac-LEHD-AMC (trifluoroacetate salt)
Ac-LEHD-AMC is a fluorogenic substrate for caspase-9.[1] Upon cleavage by caspase-9, 7-amino-4-methylcoumarin (AMC) is ...
T76268 Mca-VDQVDGW-Lys(Dnp)-NH2
Mca-VDQVDGW-Lys(Dnp)-NH2 是 caspase-7 的荧光底物。可用于定量 caspase-7 活性。
T69632 VRT-043198
VRT-043198 是 VX-765 (Belnacasan) 的活性代谢物,是有效的、选择性的、能透过血脑屏障的caspase-1的抑制剂。VRT-043198 对caspase-1和 caspase-4 的 Ki 值分别为 0.8 n...
T23555 Z-VEID-FMK Others
When compared to other caspase inhibitors, Z-DRHD-FMK inhibited caspase 6 activity more effectively than the general cas...
T36333 Z-IETD-AFC
Z-IETD-AFC is a fluorogenic substrate for caspase-8 and granzyme B. Upon enzymatic cleavage by caspase-8 or granzyme B, ...
T76091 Ac-WEHD-AFC TFA
Ac-WEHD-AFC TFA 是一种荧光caspase-1底物。Ac-WEHD-AFC TFA 可检测caspase-1荧光活性,用于肿瘤和炎症的研究。
T36353 Suc-Tyr-Val-Ala-Asp-pNA
Suc-YVAD-pNA, a chromogenic caspase-1 substrate.
T12413 PETCM Others
PETCM is a caspase-3 activator and acts as an cytochrome c (cyto c)-dependent manner.
ML132
T16105
synonym: NCGC 00185682
Target:
Z-LEED-FMK
T76665
synonym:
Target:
Arg-Gly-Asp-Ser TFA
T73870
synonym:
Target:
MX1013
T21293
synonym: MX-1013,MX 1013
Target:
TRP-601
T24903
synonym: TRP601
Target:
CP-18 F-18
T31040
synonym: CP 18 F-18,CP18 F-18,(18F)-CP18
Target:
Tauroursodeoxycholate dihydrate
T16998
synonym: 牛磺熊去氧胆酸二水合物,UR 906 dihydrate,Taurolite dihydrate,TUDCA dihydrate
Target:
AC-VEID-CHO TFA
T73683
synonym:
Target:
Ac-DNLD-AMC
T36341
synonym:
Target:
Z-VAD-AMC (acetate)
T36334
synonym:
Target:
Z-AEVD-FMK
T36331
synonym: Z-AEVD-FMK,Z-Ala-Glu-Val-Asp-Fluoromethyl Ketone
Target:
Suc-YVAD-AMC (acetate)
T36354
synonym:
Target:
Ac-LEHD-AMC (trifluoroacetate salt)
T36342
synonym:
Target:
Mca-VDQVDGW-Lys(Dnp)-NH2
T76268
synonym:
Target:
VRT-043198
T69632
synonym:
Target:
Z-VEID-FMK
T23555
synonym:
Target:
Z-IETD-AFC
T36333
synonym:
Target:
Ac-WEHD-AFC TFA
T76091
synonym:
Target:
Suc-Tyr-Val-Ala-Asp-pNA
T36353
synonym:
Target:
PETCM
T12413
synonym:
Target:
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