T16105 |
ML132
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NCGC 00185682 |
Others
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ML132 is an effective and selective inhibitor of caspase 1 (IC50: 0.316 nM). |
T76665 |
Z-LEED-FMK
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Z-LEED-FMK 是 caspase-13和 caspase-4抑制剂。Z-LEED-FMK 还能抑制S. typhimurium 感染的巨噬细胞中caspase-1的加工。 |
T73870 |
Arg-Gly-Asp-Ser TFA
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Arg-Gly-Asp-Ser (TFA) 是整联蛋白结合序列,抑制整联蛋白受体 (integrinreceptor) 功能。Arg-Gly-Asp-Ser (TFA) 直接并特异性地结合 pro-caspase-8,pro-caspase... |
T21293 |
MX1013
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MX-1013,MX 1013 |
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MX1013, a dipeptide pan-caspase inhibitor, inhibits caspase-1, -3, -6, -7, -8, and -9. |
T24903 |
TRP-601
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TRP601 |
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TRP-601 is a caspase inhibitor. |
T31040 |
CP-18 F-18
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CP 18 F-18,CP18 F-18,(18F)-CP18 |
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CP-18 F-18 is a DEVD (the caspase 3 substrate recognition motif) that is an imaging tracer for caspase-3 activity in apo... |
T16998 |
Tauroursodeoxycholate dihydrate
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牛磺熊去氧胆酸二水合物,UR 906 dihydrate,Taurolite dihydrate,TUDCA dihydrate |
Caspase
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ERK
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Tauroursodeoxycholate dihydrate is an endoplasmic reticulum stress inhibitor. Tauroursodeoxycholate also inhibits ERK. T... |
T73683 |
AC-VEID-CHO TFA
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AC-VEID-CHO (TFA) 是一种多肽来源的半胱天冬酶抑制剂,对 Caspase-6、Caspase-3 和 Caspase-7 具有抑制作用,IC50值分别为 16.2 nM、13.6 nM 和162.1 nM。AC-VEID-C... |
T36341 |
Ac-DNLD-AMC
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Ac-DNLD-AMC is a fluorogenic caspase-3 substrate. Upon enzymatic cleavage by caspase-3, 7-amino-4-methylcoumarin (AMC) i... |
T36334 |
Z-VAD-AMC (acetate)
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Z-VAD-AMC is a fluorogenic substrate for caspase-1. Upon enzymatic cleavage by caspase-1, 7-amino-4-methylcoumarin (AMC)... |
T36331 |
Z-AEVD-FMK
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Z-AEVD-FMK,Z-Ala-Glu-Val-Asp-Fluoromethyl Ketone |
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Z-AEVD-FMK is an irreversible inhibitor of caspase-10 and related caspases.[1] At 10 µM, it can prevent the initiati... |
T36354 |
Suc-YVAD-AMC (acetate)
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Suc-YVAD-AMC is a fluorogenic substrate for caspase-1. Upon enzymatic cleavage by caspase-1, 7-amino-4-methylcoumarin (A... |
T36342 |
Ac-LEHD-AMC (trifluoroacetate salt)
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Ac-LEHD-AMC is a fluorogenic substrate for caspase-9.[1] Upon cleavage by caspase-9, 7-amino-4-methylcoumarin (AMC) is ... |
T76268 |
Mca-VDQVDGW-Lys(Dnp)-NH2
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Mca-VDQVDGW-Lys(Dnp)-NH2 是 caspase-7 的荧光底物。可用于定量 caspase-7 活性。 |
T69632 |
VRT-043198
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VRT-043198 是 VX-765 (Belnacasan) 的活性代谢物,是有效的、选择性的、能透过血脑屏障的caspase-1的抑制剂。VRT-043198 对caspase-1和 caspase-4 的 Ki 值分别为 0.8 n... |
T23555 |
Z-VEID-FMK
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Others
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When compared to other caspase inhibitors, Z-DRHD-FMK inhibited caspase 6 activity more effectively than the general cas... |
T36333 |
Z-IETD-AFC
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Z-IETD-AFC is a fluorogenic substrate for caspase-8 and granzyme B. Upon enzymatic cleavage by caspase-8 or granzyme B, ... |
T76091 |
Ac-WEHD-AFC TFA
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Ac-WEHD-AFC TFA 是一种荧光caspase-1底物。Ac-WEHD-AFC TFA 可检测caspase-1荧光活性,用于肿瘤和炎症的研究。 |
T36353 |
Suc-Tyr-Val-Ala-Asp-pNA
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Suc-YVAD-pNA, a chromogenic caspase-1 substrate. |
T12413 |
PETCM
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Others
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PETCM is a caspase-3 activator and acts as an cytochrome c (cyto c)-dependent manner. |